XP-524 is a dual-BET/EP300 inhibitor that represses oncogenic KRAS and potentiates immune checkpoint inhibition in pancreatic cancer
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A. Rana | K. Ratia | J. Trevino | H. Munshi | Suneel D. Kamath | D. Principe | Dinesh Thummuri | Oleksii Dubrovskyi | Zhengnan Shen | R. Xiong | Jiong Zhao | Patrick W. Underwood | Fei Huang | Yangfeng Li | G. Thatcher | Thao N. D. Pham | Zhou Daohong | Yangfeng Li | Daohong Zhou