Quantitative structure-property relationship modeling of remote liposome loading of drugs.
暂无分享,去创建一个
Alexander Golbraikh | Amiram Goldblum | Alexander Tropsha | Yechezkel Barenholz | Ahuva Cern | A. Tropsha | A. Goldblum | Y. Barenholz | A. Golbraikh | Aleck Sedykh | Ahuva Cern | A. Sedykh
[1] T. Redelmeier,et al. Development of a Liposome Formulation of Ethambutol , 2004, Antimicrobial Agents and Chemotherapy.
[2] Lisa Krugner-Higby,et al. A mathematical relationship for hydromorphone loading into liposomes with trans-membrane ammonium sulfate gradients. , 2010, Journal of pharmaceutical sciences.
[3] Tropsha Alexander,et al. Predictive quantitative structure-activity relationships modeling: Development and validation of QSAR models , 2010 .
[4] Amiram Goldblum,et al. Predicting Oral Druglikeness by Iterative Stochastic Elimination , 2010, J. Chem. Inf. Model..
[5] Bee Jen Tan,et al. Liposomal M-V-05: formulation development and activity testing of a novel dihydrofolate reductase inhibitor for breast cancer therapy. , 2010, International journal of oncology.
[6] Hong Wong,et al. Pharmacokinetic comparison of intravenous carbendazim and remote loaded carbendazim liposomes in nude mice. , 2002, Journal of pharmaceutical and biomedical analysis.
[7] Na Zhang,et al. Targeted delivery of levofloxacin-liposomes for the treatment of pulmonary inflammation , 2009, Journal of drug targeting.
[8] Y. Barenholz,et al. Prolonged circulation time and enhanced accumulation in malignant exudates of doxorubicin encapsulated in polyethylene-glycol coated liposomes. , 1994, Cancer research.
[9] Chih-Jen Lin,et al. LIBSVM: A library for support vector machines , 2011, TIST.
[10] Kosuke Shimizu,et al. Cancer chemotherapy by liposomal 6-[12-(dimethylamino)ethyl]aminol-3-hydroxy-7H-indeno[2,1-clquinolin-7-one dihydrochloride (TAS-103), a novel anti-cancer agent. , 2002, Biological & pharmaceutical bulletin.
[11] Qiang Zhang,et al. In vitro cytotoxicity of Stealth liposomes co-encapsulating doxorubicin and verapamil on doxorubicin-resistant tumor cells. , 2005, Biological & pharmaceutical bulletin.
[12] Kosuke Shimizu,et al. Potential usage of liposomal 4beta-aminoalkyl-4'-O-demethyl-4-desoxypodophyllotoxin (TOP-53) for cancer chemotherapy. , 2002, Biological & pharmaceutical bulletin.
[13] Hao Cai,et al. Ammonium sulfate gradient loading of brucine into liposomes: effect of phospholipid composition on entrapment efficiency and physicochemical properties in vitro. , 2010, Drug development and industrial pharmacy.
[14] Bernhard Schölkopf,et al. Shrinking the Tube: A New Support Vector Regression Algorithm , 1998, NIPS.
[15] Amiram Goldblum,et al. Liposome drugs' loading efficiency: a working model based on loading conditions and drug's physicochemical properties. , 2009, Journal of controlled release : official journal of the Controlled Release Society.
[16] I-Ming Chu,et al. Effect of composition on the stability of liposomal irinotecan prepared by a pH gradient method. , 2003, Journal of bioscience and bioengineering.
[17] T. Ishida,et al. Encapsulation of an antivasospastic drug, fasudil, into liposomes, and in vitro stability of the fasudil-loaded liposomes. , 2002, International journal of pharmaceutics.
[18] Alexander Tropsha,et al. Novel Variable Selection Quantitative Structure-Property Relationship Approach Based on the k-Nearest-Neighbor Principle , 2000, J. Chem. Inf. Comput. Sci..
[19] M. Bally,et al. Uptake of adriamycin into large unilamellar vesicles in response to a pH gradient. , 1986, Biochimica et biophysica acta.
[20] Massimo Fresta,et al. Cytotoxic effects of Gemcitabine-loaded liposomes in human anaplastic thyroid carcinoma cells , 2004, BMC Cancer.
[21] Elias Fattal,et al. Therapeutic Potential of New 4-hydroxy-tamoxifen-Loaded pH-gradient Liposomes in a Multiple Myeloma Experimental Model , 2010, Pharmaceutical Research.
[22] Yechezkel Barenholz,et al. Relevancy of Drug Loading to Liposomal Formulation Therapeutic Efficacy , 2003, Journal of liposome research.
[23] 안드레아스 와그너,et al. Liposomal composition comprising an active ingredient for relaxing smooth muscle, the production of this composition and therapeutically use thereof , 2005 .
[24] Li Zhang,et al. Encapsulation of mitoxantrone into pegylated SUVs enhances its antineoplastic efficacy. , 2008, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[25] Yechezkel Barenholz,et al. Amphipathic weak acid glucocorticoid prodrugs remote-loaded into sterically stabilized nanoliposomes evaluated in arthritic rats and in a Beagle dog: a novel approach to treating autoimmune arthritis. , 2008, Arthritis and rheumatism.
[26] S. A. Sande,et al. Formulation and characterisation of primaquine loaded liposomes prepared by a pH gradient using experimental design. , 2000, International journal of pharmaceutics.
[27] M. Bally,et al. Improved retention of idarubicin after intravenous injection obtained for cholesterol-free liposomes. , 2002, Biochimica et biophysica acta.
[28] Silvia Arpicco,et al. Preparation, characterization, cytotoxicity and pharmacokinetics of liposomes containing lipophilic gemcitabine prodrugs. , 2004, Journal of controlled release : official journal of the Controlled Release Society.
[29] M. Bally,et al. The accumulation of drugs within large unilamellar vesicles exhibiting a proton gradient: a survey. , 1990, Chemistry and physics of lipids.
[30] Y. Oh,et al. Formulation and efficacy of liposome-encapsulated antibiotics for therapy of intracellular Mycobacterium avium infection , 1995, Antimicrobial agents and chemotherapy.
[31] Mark Voorneveld,et al. Preparation , 2018, Games Econ. Behav..
[32] Vladimir N. Vapnik,et al. The Nature of Statistical Learning Theory , 2000, Statistics for Engineering and Information Science.
[33] Yechezkel Barenholz,et al. Pharmacokinetics of Pegylated Liposomal Doxorubicin , 2003, Clinical pharmacokinetics.
[34] Volker Wagner,et al. The emerging nanomedicine landscape , 2006, Nature Biotechnology.
[35] Y. Barenholz,et al. Fluidity parameters of lipid regions determined by fluorescence polarization. , 1978, Biochimica et biophysica acta.
[36] R. Schubert,et al. Remote loading of doxorubicin into liposomes driven by a transmembrane phosphate gradient. , 2006, Biochimica et biophysica acta.
[37] J. Ross Quinlan,et al. Improved Use of Continuous Attributes in C4.5 , 1996, J. Artif. Intell. Res..
[38] Y. Barenholz,et al. Dynamics of the hydrocarbon layer in liposomes of lecithin and sphingomyelin containing dicetylphosphate. , 1974, The Journal of biological chemistry.
[39] A. Kozubek,et al. The encapsulation of idarubicin within liposomes using the novel EDTA ion gradient method ensures improved drug retention in vitro and in vivo. , 2010, Journal of controlled release : official journal of the Controlled Release Society.
[40] Yechezkel Barenholz,et al. Liposome application: problems and prospects , 2001 .
[41] F. Frézard,et al. Encapsulation of Mithramycin in Liposomes in Response to a Transmembrane Gradient of Calcium Ions , 1997 .
[42] M. Rocchetti,et al. Development and validation of in silico models for estimating drug preformulation risk in PEG400/water and Tween80/water systems. , 2007, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.
[43] Jing Qin,et al. Preparation, Characterization, and Evaluation of Liposomal Ferulic Acid In Vitro and In Vivo , 2008 .
[44] Y. Barenholz,et al. Doxil® — The First FDA-Approved Nano-Drug: From an Idea to a Product , 2021, Handbook of Harnessing Biomaterials in Nanomedicine.
[45] Yi Jin,et al. Preparation and in vitro evaluation of liposomal chloroquine diphosphate loaded by a transmembrane pH-gradient method. , 2008, International journal of pharmaceutics.
[46] Patrick Couvreur,et al. Supramolecular organization of S12363-liposomes prepared with two different remote loading processes. , 2009, Biochimica et biophysica acta.
[47] I V Zhigaltsev,et al. LIPOSOMES CONTAINING DOPAMINE ENTRAPPED IN RESPONSE TO TRANSMEMBRANE AMMONIUM SULFATE GRADIENT AS CARRIER SYSTEM FOR DOPAMINE DELIVERY INTO THE BRAIN OF PARKINSONIAN MICE , 2001, Journal of liposome research.
[48] Sérgio Simões,et al. Liposomal imatinib–mitoxantrone combination: Formulation development and therapeutic evaluation in an animal model of prostate cancer , 2011, The Prostate.
[49] Bernhard Schölkopf,et al. New Support Vector Algorithms , 2000, Neural Computation.
[50] Norbert Maurer,et al. Development of a weak-base docetaxel derivative that can be loaded into lipid nanoparticles. , 2010, Journal of controlled release : official journal of the Controlled Release Society.
[51] T Nagai,et al. Remote loading of diclofenac, insulin and fluorescein isothiocyanate labeled insulin into liposomes by pH and acetate gradient methods. , 1999, International journal of pharmaceutics.
[52] Jing Qin,et al. Preparation, characterization, and evaluation of liposomal ferulic acid in vitro and in vivo. , 2008, Drug development and industrial pharmacy.
[53] Li Zhang,et al. Development of pegylated liposomal vinorelbine formulation using "post-insertion" technology. , 2010, International journal of pharmaceutics.
[54] Lisa Krugner-Higby,et al. Pharmacokinetics and Behavioral Effects of an Extended-Release, Liposome-Encapsulated Preparation of Oxymorphone in Rhesus Macaques , 2009, Journal of Pharmacology and Experimental Therapeutics.
[55] S Du,et al. Studies on the Encapsulation of Oxymatrine into Liposomes by Ethanol Injection and pH Gradient Method , 2006, Drug development and industrial pharmacy.
[56] A. Filho,et al. Rifabutin encapsulated in liposomes exhibits increased therapeutic activity in a model of disseminated tuberculosis. , 2008, International journal of antimicrobial agents.
[57] K. Edwards,et al. 449 PH GRADIENT LOADING OF ANTHRACYCLINES INTO CHOLESTEROL-FREE LIPOSOMES: ENHANCING DRUG LOADING RATES THROUGH USE OF ETHANOL. , 2001, Journal of Investigative Medicine.
[58] Amiram Goldblum,et al. A stochastic algorithm for global optimization and for best populations: A test case of side chains in proteins , 2002, Proceedings of the National Academy of Sciences of the United States of America.
[59] D. Klatzmann,et al. Liposomal encapsulation of ganciclovir enhances the efficacy of herpes simplex virus type 1 thymidine kinase suicide gene therapy against hepatic tumors in rats. , 1999, Human gene therapy.