Synthesis of 2,4,5-trisubstituted thiazoles with a 5-(N,N-dimethylaminomethyl) substituent
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[1] Russ N. Fitzgerald,et al. An efficient synthesis of a potent PPARpan agonist. , 2006, The Journal of organic chemistry.
[2] H. Sham,et al. Synthesis and Structure−Activity Relationships of N-{3-[2-(4-Alkoxyphenoxy)thiazol-5-yl]-1- methylprop-2-ynyl}carboxy Derivatives as Selective Acetyl-CoA Carboxylase 2 Inhibitors , 2006 .
[3] M. Drew,et al. A new route to furanoeremophilane sesquiterpenoids. Synthesis of Senecio metabolites (±)-6-hydroxyeuryopsin, (±)-1,10-epoxy-6-hydroxyeuryopsin, (±)-toluccanolide A and (±)-toluccanolide C , 2006 .
[4] C. Moody,et al. Total synthesis of the thiopeptide antibiotic amythiamicin D. , 2005, Journal of the American Chemical Society.
[5] F. Qing,et al. Sodium carbonate as carbon dioxide source for the synthesis of cyclic carbonates containing the trifluoromethyl group , 2003 .
[6] E. Sotelo,et al. Pyridazine derivatives. Part 33: Sonogashira approaches in the synthesis of 5-substituted-6-phenyl-3(2H)-pyridazinones☆ , 2003 .
[7] F. Al-Obeidi,et al. Synthesis of 2,5-dihalothiazole-4-carboxylates , 2002 .
[8] Z. Xia,et al. Total synthesis of dendroamide A, a novel cyclic peptide that reverses multiple drug resistance. , 2001, The Journal of organic chemistry.
[9] P. Knochel,et al. Preparation of new polyfunctional magnesiated heterocycles using a chlorine-, bromine-, or iodine-magnesium exchange , 2000, The Journal of organic chemistry.
[10] G. H. Coombs,et al. Enzymes of parasite thiol metabolism as drug targets. , 1999, Parasitology today.
[11] Maria Cristina Burla,et al. SIR97: a new tool for crystal structure determination and refinement , 1999 .
[12] E. Bures,et al. Regioselective Preparation of 2,4-, 3,4-, and 2,3,4-Substituted Furan Rings. 1. [1,4] O → C and [1,4] C → O Silyl Migrations of Silyl Ethers and Esters Attached to Furan and Thiophene Rings , 1997 .
[13] N. Kundu,et al. Palladium-catalyzed heteroannulation with acetylenic carbinols as synthons-synthesis of quinolines and 2,3-dihydro-4(1H)-quinolones , 1997 .
[14] R. Prager,et al. The chemistry of 5-oxodihydroisoxazoles .19. The synthesis and photolysis of N-thioacylisoxazol-5(2H)-ones , 1997 .
[15] Jang-Woo Kim,et al. Synthesis of 1-(dimethylsulfamoyl)-2- and 5-imidazolecarboxaldehydes. Rearrangement of 1-(dimethylsulfamoyl)-5-imidazole-carboxaldehyde to the 4-carboxaldehyde† , 1995 .
[16] J. Périchon,et al. DBU/DMSO promoted dehydrobromination of 1,1-dibromoolefins. A general synthesis of 1-bromoaromatic alkynes under mild conditions , 1994 .
[17] T. Fröhlich,et al. Synthesis of oligoribonucleotides containing isoguanosine , 1994 .
[18] D. Mathre,et al. Direct conversion of activated alcohols to azides using diphenyl phosphorazidate. A practical alternative to mitsunobu conditions , 1993 .
[19] D. Dess,et al. A useful 12-I-5 triacetoxyperiodinane (the Dess-Martin periodinane) for the selective oxidation of primary or secondary alcohols and a variety of related 12-I-5 species , 1991 .
[20] F. Diederich,et al. Solution-spray flash vacuum pyrolysis: a new method for the synthesis of linear poliynes with odd numbers of C.tplbond.C bonds from substituted 3,4-dialkynyl-3-cyclobutene-1,2-diones , 1991 .
[21] R. Friesen,et al. Hydroboration of C-arylglucals. Synthesis of the β-C-arylglucoside nucleus of chaetiacandin , 1990 .
[22] E. Bures,et al. The regiospecific formation and reactions of 4-lithio-2-(t-butyldimethylsilyl)- 3-(hydroxymethyl)furan: An approach to 3,4-disubstituted furans. , 1988 .
[23] E. Bures,et al. The 1,4 O→C silyl migrations of various 3-[(trialkylsilyl)-oxymethyl]-furans and -thiophenes , 1987 .
[24] A. Medici,et al. Palladium-Mediated Cross-Coupling Reactions Between Stannyl- and Bromothiazoles. Preparation of Thiazole Oligomers , 1987 .
[25] B. Chait,et al. Trypanothione: a novel bis(glutathionyl)spermidine cofactor for glutathione reductase in trypanosomatids. , 1985, Science.
[26] S. Nahm,et al. N-methoxy-n-methylamides as effective acylating agents , 1982 .
[27] E. Corey,et al. A synthetic method for formyl→ethynyl conversion (RCHO→RCCH or RCCR′) , 1972 .
[28] R. West,et al. Lithiation of trimethylsilyl compounds , 1968 .
[29] W. Shive,et al. SYNTHESIS OF INDOLE DERIVATIVES. 5-INDOLECARBOXYLIC ACID , 1955 .