Sticking and Picking in Pharmaceutical Tablet Compression: An IQ Consortium Review.
暂无分享,去创建一个
Mike Tobyn | Sayantan Chattoraj | Patrick David Daugherity | Todd McDermott | Angela Olsofsky | Wyatt J. Roth | M. Tobyn | S. Chattoraj | W. Roth | P. Daugherity | Todd McDermott | Angela Olsofsky
[1] Marcial Gonzalez,et al. A nonlocal contact formulation for confined granular systems , 2011, 1107.4607.
[2] M. Sherry Ku,et al. Use of the Biopharmaceutical Classification System in Early Drug Development , 2008, The AAPS Journal.
[3] Fernando Muzzio,et al. Enabling real time release testing by NIR prediction of dissolution of tablets made by continuous direct compression (CDC). , 2016, International journal of pharmaceutics.
[4] Feng Qian,et al. Formulation and process design for a solid dosage form containing a spray-dried amorphous dispersion of ibipinabant , 2013, Pharmaceutical development and technology.
[5] Krystan Reed,et al. Tablet sticking: Using a ‘compression toolbox’ to assess multiple tooling coatings options , 2015 .
[6] Naveen K. Bejugam,et al. Tablet formulation of an active pharmaceutical ingredient with a sticking and filming problem: direct compression and dry granulation evaluations , 2015, Drug development and industrial pharmacy.
[7] C. Leopold,et al. Novel aspects on the direct compaction of ibuprofen with special focus on sticking , 2017 .
[8] A. Narang,et al. Decoupling the contribution of dispersive and acid-base components of surface energy on the cohesion of pharmaceutical powders. , 2014, International journal of pharmaceutics.
[9] Michael Leane,et al. A proposal for a drug product Manufacturing Classification System (MCS) for oral solid dosage forms , 2015, Pharmaceutical development and technology.
[10] Wenli Zhang,et al. Novel application method of talcum powder to prevent sticking tendency and modify release of esomeprazole magnesium enteric-coated pellets , 2015, Pharmaceutical development and technology.
[11] V. Balaram. Recent advances in the determination of elemental impurities in pharmaceuticals – Status, challenges and moving frontiers , 2016 .
[12] Ajit S. Narang,et al. Molecular Basis of Crystal Morphology-Dependent Adhesion Behavior of Mefenamic Acid During Tableting , 2013, Pharmaceutical Research.
[13] Toshiyuki Niwa,et al. Influence of compression pressure and velocity on tablet sticking. , 2010, Chemical & pharmaceutical bulletin.
[14] Satu Lakio,et al. Single-step Coprocessing of Cohesive Powder via Mechanical Dry Coating for Direct Tablet Compression. , 2017, Journal of pharmaceutical sciences.
[15] Joseph Kushner. Utilizing quantitative certificate of analysis data to assess the amount of excipient lot-to-lot variability sampled during drug product development , 2013, Pharmaceutical development and technology.
[16] Mike Tobyn,et al. Multivariate analysis in the pharmaceutical industry: enabling process understanding and improvement in the PAT and QbD era , 2015, Pharmaceutical development and technology.
[17] Marianthi Ierapetritou,et al. Real time monitoring of powder blend bulk density for coupled feed-forward/feed-back control of a continuous direct compaction tablet manufacturing process. , 2015, International journal of pharmaceutics.
[18] P. Schmidt,et al. Influence of Compacted Hydrophobic and Hydrophilic Colloidal Silicon Dioxide on Tableting Properties of Pharmaceutical Excipients , 2005, Drug development and industrial pharmacy.
[19] Changquan Calvin Sun,et al. Mini review: Mechanisms to the loss of tabletability by dry granulation. , 2016, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[20] Caly Chien,et al. Effect of food on abiraterone pharmacokinetics: a review , 2017 .
[21] Preetanshu Pandey,et al. A quality by design approach to scale-up of high-shear wet granulation process , 2016, Drug development and industrial pharmacy.
[22] A Sabir,et al. Formulation and process optimization to eliminate picking from market image tablets. , 2001, International journal of pharmaceutics.
[23] Vivek S. Dave,et al. Excipient variability and its impact on dosage form functionality. , 2015, Journal of pharmaceutical sciences.
[24] K. Morris,et al. Modeling of adhesion in tablet compression. II. Compaction studies using a compaction simulator and an instrumented tablet press. , 2004, Journal of pharmaceutical sciences.
[25] Gudrun A Fridgeirsdottir,et al. Support Tools in Formulation Development for Poorly Soluble Drugs. , 2016, Journal of pharmaceutical sciences.
[26] S. Byrn,et al. Stability of pharmaceutical salts in solid oral dosage forms , 2017, Drug development and industrial pharmacy.
[27] P. Schmidt,et al. Investigation of compacted hydrophilic and hydrophobic colloidal silicon dioxides as glidants for pharmaceutical excipients , 2004 .
[28] Maunu Toiviainen,et al. Continuous manufacturing of tablets with PROMIS-line - Introduction and case studies from continuous feeding, blending and tableting. , 2016, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.
[29] S. Srčič,et al. Application of instrumented nanoindentation in preformulation studies of pharmaceutical active ingredients and excipients , 2016, Acta pharmaceutica.
[30] John N. Staniforth. Use of Hydrogenated Vegetable Oil as a Tablet Lubricant , 1987 .
[31] C. Shang,et al. Modelling of the break force of tablets under diametrical compression. , 2013, International journal of pharmaceutics.
[32] Ben Forbes,et al. The influence of electrostatic properties on the punch sticking propensity of pharmaceutical blends , 2017 .
[33] H. Mangal,et al. Roll compaction/dry granulation: Suitability of different binders. , 2016, International journal of pharmaceutics.
[34] Fernando J. Muzzio,et al. Continuous Powder Mixing , 2015 .
[35] Fernando J. Muzzio,et al. Advanced Control of Continuous Pharmaceutical Tablet Manufacturing Processes , 2016 .
[36] P. Kleinebudde,et al. Effect of roll-compaction and milling conditions on granules and tablet properties. , 2016, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[37] S. Schumann,et al. The effects of chromium nitride ion bombardment treatment of tablet tooling on tablet adherence , 1992 .
[38] John F. Gamble,et al. Understanding the effect of API changes in pharmaceutical processing , 2017 .
[39] John N. Staniforth,et al. Aspects of Pharmaceutical Tribology , 1989 .
[40] D. F. Steele,et al. The mechanical properties of compacts of microcrystalline cellulose and silicified microcrystalline cellulose. , 2000, International journal of pharmaceutics.
[41] A. Narang,et al. Decoupling the Contribution of Surface Energy and Surface Area on the Cohesion of Pharmaceutical Powders , 2014, Pharmaceutical Research.
[42] Divyakant Desai,et al. Lubrication in tablet formulations. , 2010, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[43] Clive J Roberts,et al. Characterising the surface adhesive behavior of tablet tooling components by atomic force microscopy , 2011, Drug development and industrial pharmacy.
[44] Changquan Calvin Sun,et al. Mechanism and Kinetics of Punch Sticking of Pharmaceuticals. , 2017, Journal of pharmaceutical sciences.
[45] C. Sun,et al. Modulating Sticking Propensity of Pharmaceuticals Through Excipient Selection in a Direct Compression Tablet Formulation , 2018, Pharmaceutical Research.
[46] J. Kushner,et al. Scale-up model describing the impact of lubrication on tablet tensile strength. , 2010, International journal of pharmaceutics.
[47] P. Kleinebudde,et al. Roll compaction/dry granulation: Comparison between roll mill and oscillating granulator in dry granulation , 2012, Pharmaceutical development and technology.
[48] Bo Lang,et al. Hot-melt extrusion – basic principles and pharmaceutical applications , 2014, Drug development and industrial pharmacy.
[49] Richard L. Schild,et al. Application of imaging based tools for the characterisation of hollow spray dried amorphous dispersion particles. , 2014, International journal of pharmaceutics.
[50] Bozena Michniak-Kohn,et al. Mixing order of glidant and lubricant--influence on powder and tablet properties. , 2011, International journal of pharmaceutics.
[51] Matthew Roberts,et al. Effects of surface roughness and chrome plating of punch tips on the sticking tendencies of model ibuprofen formulations , 2003, The Journal of pharmacy and pharmacology.
[52] C. Ghoroi,et al. Influence of particle properties on powder bulk behaviour and processability. , 2017, International journal of pharmaceutics.
[53] Hisakazu Sunada,et al. Effect of water content on sticking during compression , 1997 .
[54] R. E. Gordon,et al. Utilization of differential scanning calorimetry in the compatibility screening of ibuprofen with the stearate lubricants and construction of phase diagrams , 1984 .
[55] I. Larson,et al. The role of physico-chemical and bulk characteristics of co-spray dried L-leucine and polyvinylpyrrolidone on glidant and binder properties in interactive mixtures. , 2015, International journal of pharmaceutics.
[56] M. S. Ku,et al. A biopharmaceutical classification-based Right-First-Time formulation approach to reduce human pharmacokinetic variability and project cycle time from First-In-Human to clinical Proof-Of-Concept , 2012, Pharmaceutical development and technology.
[57] K. El-Say,et al. COMPARATIVE STUDY AMONG DIFFERENT TECHNIQUES TO IMPROVE THE PHYSICAL AND TECHNICAL PROPERTIES PREVAILING TO COMPRESSION OF POORLY FLOWING AND HIGHLY COHESIVE DRUG , 2010 .
[58] David S. Jones,et al. Hot melt extrusion – processing solid solutions? , 2014, The Journal of pharmacy and pharmacology.
[59] R. Greenwood,et al. Application of external lubrication during the roller compaction of adhesive pharmaceutical formulations , 2013, Pharmaceutical development and technology.
[60] W. Stagner,et al. Application of multivariate methods to evaluate the functionality of bovine- and vegetable-derived magnesium stearate. , 2014, Journal of pharmaceutical sciences.
[61] William Early,et al. An evaluation of process parameters to improve coating efficiency of an active tablet film-coating process. , 2012, International journal of pharmaceutics.
[62] P. Kleinebudde,et al. Critical evaluation of root causes of the reduced compactability after roll compaction/dry granulation. , 2015, Journal of pharmaceutical sciences.
[63] R C Rowe,et al. Process control and scale-up of pharmaceutical wet granulation processes: a review. , 2001, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[64] J. Strong,et al. Scanning Electron Microscope Observations of Powder Sticking on Punches during a Limited Number (N < 5) of Compactions of Acetylsalicylic Acid , 2017, Pharmaceutical Research.
[65] D. F. Steele,et al. The Use of a Modified Resin for Studying the Internal Structure of Microcrystalline Cellulose Particles , 1998 .
[66] M. H. Rubinstein,et al. Structure-lubricity evaluation of magnesium stearate , 1988 .
[67] Stephen Edge,et al. Adsorption of an Amine Drug onto Microcrystalline Cellulose and Silicified Microcrystalline Cellulose Samples , 2003, Drug development and industrial pharmacy.
[68] K. Hapgood,et al. Investigation of the potential for direct compaction of a fine ibuprofen powder dry-coated with magnesium stearate , 2015, Drug development and industrial pharmacy.
[69] D. Lapham,et al. Gas adsorption on commercial magnesium stearate: Effects of degassing conditions on nitrogen BET surface area and isotherm characteristics. , 2017, International journal of pharmaceutics.
[70] T. Shinbrot,et al. Use of a static eliminator to improve powder flow. , 2009, International journal of pharmaceutics.
[71] K. Terada,et al. Imprinting on empty hard gelatin capsule shells containing titanium dioxide by application of the UV laser printing technique , 2014, Drug development and industrial pharmacy.
[72] J. Mitchell,et al. Effects of crystal habit on the sticking propensity of ibuprofen-A case study. , 2017, International journal of pharmaceutics.
[73] Ahmad Aljaberi,et al. Functional performance of silicified microcrystalline cellulose versus microcrystalline cellulose: a case study , 2009, Drug development and industrial pharmacy.
[74] C Vervaet,et al. Continuous direct compression as manufacturing platform for sustained release tablets. , 2017, International journal of pharmaceutics.
[75] P. Schmidt,et al. Investigation of the glidant properties of compacted colloidal silicon dioxide by angle of repose and X-ray photoelectron spectroscopy. , 2006, European journal of pharmaceutics and biopharmaceutics.
[76] Hong Wen,et al. Systematical approach of formulation and process development using roller compaction. , 2009, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[77] J. Polli,et al. Impact of Biopharmaceutics Classification System-based biowaivers. , 2010, Molecular pharmaceutics.
[78] Troy Shinbrot,et al. An observed correlation between flow and electrical properties of pharmaceutical blends , 2009 .
[79] Dolapo Olusanmi,et al. Measuring the sticking of mefenamic acid powders on stainless steel surface. , 2015, International journal of pharmaceutics.
[80] Changquan Calvin Sun. Dependence of ejection force on tableting speed—A compaction simulation study , 2015 .
[81] G. Finet,et al. Influence of the morphogranulometry and hydrophobicity of talc on its antisticking power in the production of tablets. , 2005, International journal of pharmaceutics.
[82] T. Laich,et al. Untersuchung schmiermittelabhängiger Kenngrössen an einer Exzentertablettenpresse ausgerüstet mit einem externen Schmiersystem , 1998 .
[83] C. Leopold,et al. A novel technique for the visualization of tablet punch surfaces: Characterization of surface modification, wear and sticking. , 2017, International journal of pharmaceutics.
[84] H. Takeuchi,et al. Prediction of effects of punch shapes on tableting failure by using a multi-functional single-punch tablet press , 2017, Asian journal of pharmaceutical sciences.
[85] Erin M. Hansuld,et al. A review of monitoring methods for pharmaceutical wet granulation. , 2014, International journal of pharmaceutics.
[86] Srimanta Sarkar,et al. Influence of the Punch Head Design on the Physical Quality of Tablets Produced in a Rotary Press. , 2017, Journal of pharmaceutical sciences.
[87] G. P. McCarthy,et al. Physicochemical comparison between microcrystalline cellulose and silicified microcrystalline cellulose , 1998 .
[88] Christel A. S. Bergström,et al. The Need for Restructuring the Disordered Science of Amorphous Drug Formulations , 2017, Pharmaceutical Research.
[89] Matthew Roberts,et al. Effect of punch tip geometry and embossment on the punch tip adherence of a model ibuprofen formulation , 2004, The Journal of pharmacy and pharmacology.
[90] A. Narang,et al. Effect of crystal habits on the surface energy and cohesion of crystalline powders. , 2014, International journal of pharmaceutics.
[91] John F. Gamble,et al. Monitoring process induced attrition of drug substance particles within formulated blends. , 2014, International journal of pharmaceutics.
[92] Fernando J. Muzzio,et al. Characterizing continuous powder mixing using residence time distribution , 2011 .
[93] P. Schmidt,et al. Mechanism of glidants: investigation of the effect of different colloidal silicon dioxide types on powder flow by atomic force and scanning electron microscopy. , 2004, Journal of pharmaceutical sciences.
[94] Koichi Wada,et al. Formulation design for poorly water-soluble drugs based on biopharmaceutics classification system: basic approaches and practical applications. , 2011, International journal of pharmaceutics.
[95] A. Kara,et al. An application for zirconia as a pharmaceutical die set , 2004 .
[96] Changquan Calvin Sun,et al. Systematic evaluation of common lubricants for optimal use in tablet formulation , 2018, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.
[97] C. Sun,et al. Ribbon thickness influences fine generation during dry granulation. , 2017, International journal of pharmaceutics.
[98] Alexander Krok,et al. Numerical investigation into the influence of the punch shape on the mechanical behavior of pharmaceutical powders during compaction , 2014 .
[99] T. Shinbrot,et al. AFM study of hydrophilicity on acetaminophen crystals. , 2012, International journal of pharmaceutics.
[100] P. Kleinebudde,et al. Evaluation of lubrication methods: How to generate a comparable lubrication for dry granules and powder material for tableting processes , 2014 .
[101] P. Schmidt,et al. Preparation and optimization of l-leucine as lubricant for effervescent tablet formulations , 1995 .
[102] Manabu Ito,et al. Development of new shaped punch to predict scale-up issue in tableting process. , 2014, Journal of pharmaceutical sciences.
[103] H. Ishihara,et al. Studies on the mechanism of printing film-coated tablets containing titanium dioxide in the film by using UV laser irradiation , 2009, Drug development and industrial pharmacy.
[104] P. Schmidt,et al. Optimization of an effervescent tablet formulation containing spray dried L-leucine and polyethylene glycol 6000 as lubricants using a central composite design. , 1998, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[105] I. Larson,et al. Effect of the deformability of guest particles on the tensile strength of tablets from interactive mixtures. , 2016, International journal of pharmaceutics.
[106] Changquan Calvin Sun. Materials science tetrahedron--a useful tool for pharmaceutical research and development. , 2009, Journal of pharmaceutical sciences.
[107] G. Bolhuis,et al. BONDING CHARACTERISTICS BY SCANNING ELECTRON-MICROSCOPY OF POWDERS MIXED WITH MAGNESIUM STEARATE , 1978 .
[108] Changquan Calvin Sun,et al. Powder properties and compaction parameters that influence punch sticking propensity of pharmaceuticals. , 2017, International journal of pharmaceutics.
[109] M. Ghadiri,et al. Tribo-electrification of active pharmaceutical ingredients and excipients , 2012 .
[111] M. Davies,et al. Scanning probe microscopy in the field of drug delivery. , 2007, Advanced drug delivery reviews.
[112] T De Beer,et al. Identifying overarching excipient properties towards an in-depth understanding of process and product performance for continuous twin-screw wet granulation. , 2017, International journal of pharmaceutics.
[113] I. Larson,et al. Relationship between surface concentration of L-leucine and bulk powder properties in spray dried formulations. , 2015, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[114] M. Rutland,et al. AFM Colloidal Probe Measurements Implicate Capillary Condensation in Punch-Particle Surface Interactions during Tableting. , 2017, Langmuir : the ACS journal of surfaces and colloids.
[115] M. H. Rubinstein,et al. Tablet lubricants I. Theory and modes of action , 1981 .
[116] C. Leopold,et al. Evaluation of the suitability of various lubricants for direct compaction of sorbitol tablet formulations. , 2013 .
[117] J. Kushner,et al. A quality-by-design study for an immediate-release tablet platform: examining the relative impact of active pharmaceutical ingredient properties, processing methods, and excipient variability on drug product quality attributes. , 2014, Journal of pharmaceutical sciences.
[118] P. Leterme,et al. Relation between structural characteristics of talc and its properties as an antisticking agent in the production of tablets. , 2003, European Journal of Pharmaceutical Sciences.
[119] Mohammad Hassan Khalid,et al. Effect of roll compaction on granule size distribution of microcrystalline cellulose–mannitol mixtures: computational intelligence modeling and parametric analysis , 2017, Drug design, development and therapy.
[120] Niklas Sandler,et al. Pneumatic dry granulation: potential to improve roller compaction technology in drug manufacture , 2011, Expert opinion on drug delivery.
[121] Thomas De Beer,et al. Process Analytical Technology for continuous manufacturing of solid-dosage forms , 2015 .
[122] John F. Gamble,et al. Monitoring and end-point prediction of a small scale wet granulation process using acoustic emission , 2009, Pharmaceutical development and technology.
[123] T Flanagan,et al. Biopharmaceutical aspects and implications of excipient variability in drug product performance , 2017, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[124] R. Kelly,et al. Salt disproportionation: A material science perspective. , 2017, International journal of pharmaceutics.
[125] I. C. Sinka,et al. Break force and tensile strength relationships for curved faced tablets subject to diametrical compression. , 2013, International journal of pharmaceutics.
[126] Gordon L. Amidon,et al. Prediction of Solubility and Permeability Class Membership: Provisional BCS Classification of the World’s Top Oral Drugs , 2009, The AAPS Journal.
[127] Ratnesh Lal,et al. Multidimensional atomic force microscopy for drug discovery: a versatile tool for defining targets, designing therapeutics and monitoring their efficacy. , 2010, Life sciences.
[128] M Krumme,et al. The influence of engravings on the sticking of tablets. Investigations with an instrumented upper punch. , 1999, Pharmaceutical development and technology.
[129] John W. Jones,et al. Determination of process variables affecting drug particle attrition within multi-component blends during powder feed transmission , 2017, Pharmaceutical development and technology.
[130] P. Leterme,et al. Study of talcs as antisticking agents in the production of tablets. , 2002, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.
[131] Sandeep Kumar,et al. Application of a hot-melt granulation process to enhance fenofibrate solid dose manufacturing , 2016, Drug development and industrial pharmacy.
[132] Ahmad Almaya,et al. A Demonstration of Mixing Robustness in a Direct Compression Continuous Manufacturing Process. , 2017, Journal of pharmaceutical sciences.
[133] F. Neville,et al. Colloidal Silica Particle Synthesis and Future Industrial Manufacturing Pathways: A Review , 2016 .
[134] M. Roberts,et al. Effect of lubricant type and concentration on the punch tip adherence of model ibuprofen formulations , 2004, The Journal of pharmacy and pharmacology.
[135] A. Narang,et al. Effect of milling temperatures on surface area, surface energy and cohesion of pharmaceutical powders. , 2015, International journal of pharmaceutics.
[136] K. Danjo,et al. Effect of Temperature on the Sticking of Low Melting Point Materials , 1993 .
[137] Joseph P. Neilly,et al. A material sparing method for quantitatively measuring tablet sticking , 2011 .
[138] T. Andersson,et al. Preformulation investigation and challenges; salt formation, salt disproportionation and hepatic recirculation , 2017, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.
[139] Jinjiang Li,et al. Lubricants in Pharmaceutical Solid Dosage Forms , 2014 .
[140] C. Leopold,et al. A comparative study on the sticking tendency of ibuprofen and ibuprofen sodium dihydrate to differently coated tablet punches , 2018, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[141] K. Pathak,et al. Pharmaceutical product development technologies based on the biopharmaceutical classification system. , 2009, Die Pharmazie.
[142] C. Leopold,et al. Investigation of the tableting behavior of Ibuprofen DC 85 W , 2018, Drug development and industrial pharmacy.
[143] M. Tobyn,et al. The use of colloid probe microscopy to predict aerosolization performance in dry powder inhalers: AFM and in vitro correlation. , 2006, Journal of pharmaceutical sciences.
[144] W. Abdelwahed,et al. DESIGHN AND EVALUATION OF A NEW FORMULATIONS OF ENALAPRIL MALEATE 20 MG TABLET IN A TIME EFFICIENT AND ON A LARGE INDUSTRIAL SCALE , 2014 .