Mechanisms of P-gp inhibition and effects on membrane fluidity of a new rifampicin derivative, 1,8-dibenzoyl-rifampicin.
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F. Carvalho | C. Nunes | S. Reis | F. Remião | V. Vilas-Boas | M. Bastos | Renata Silva | L. Ferreira | Cátia Vieira
[1] F. Carvalho,et al. Doxorubicin decreases paraquat accumulation and toxicity in Caco-2 cells. , 2013, Toxicology letters.
[2] J. Schellens,et al. Restricted brain penetration of the tyrosine kinase inhibitor erlotinib due to the drug transporters P-gp and BCRP , 2012, Investigational New Drugs.
[3] M. de Lourdes Bastos,et al. P‐glycoprotein activity in human Caucasian male lymphocytes does not follow its increased expression during aging , 2011, Cytometry. Part A : the journal of the International Society for Analytical Cytology.
[4] M. X. Fernandes,et al. New Uses for Old Drugs: Pharmacophore‐Based Screening for the Discovery of P‐Glycoprotein Inhibitors , 2011, Chemical biology & drug design.
[5] Donald W. Miller,et al. Assessment of P-glycoprotein Activity in the Blood-Brain Barrier (BBB) Using Near Infrared Fluorescence (NIRF) Imaging Techniques , 2011, Pharmaceutical Research.
[6] G. Levin,et al. Induction of drug efflux protein expression by venlafaxine but not desvenlafaxine , 2011, Biopharmaceutics & drug disposition.
[7] F. Carvalho,et al. In vitro study of P-glycoprotein induction as an antidotal pathway to prevent cytotoxicity in Caco-2 cells , 2011, Archives of Toxicology.
[8] S. Apte. Selecting surfactants for the maximum inhibition of the activity of the multidrug resistance efflux pump transporter, P-glycoprotein: conceptual development. , 2010 .
[9] J. Duarte,et al. Effect of chronic ethanol exposure on the hepatotoxicity of ecstasy in mice: an ex vivo study. , 2008, Toxicology in vitro : an international journal published in association with BIBRA.
[10] C. Hirayama,et al. Constitutive Overexpression of P-glycoprotein, Rather than Breast Cancer Resistance Protein or Organic Cation Transporter 1, Contributes to Acquisition of Imatinib-Resistance in K562 Cells , 2008, Pharmaceutical Research.
[11] J. Duarte,et al. P-glycoprotein induction: an antidotal pathway for paraquat-induced lung toxicity. , 2006, Free radical biology & medicine.
[12] M. Pirmohamed,et al. Induction of P-glycoprotein in lymphocytes by carbamazepine and rifampicin: the role of nuclear hormone response elements. , 2006, British journal of clinical pharmacology.
[13] P. Couraud,et al. Rat Brain Endothelial Cell Lines for the Study of Blood–Brain Barrier Permeability and Transport Functions , 2005, Cellular and Molecular Neurobiology.
[14] S. Reis,et al. Influence of some anti-inflammatory drugs in membrane fluidity studied by fluorescence anisotropy measurementsPresented at the 17th Conference of the European Colloid & Interface Science Society, Firenze, Italy, September 21?26, 2003 , 2004 .
[15] C. Dey,et al. P-glycoprotein inhibitors and their screening: a perspective from bioavailability enhancement. , 2003, Pharmacological research.
[16] D. Begley,et al. Lipids in blood-brain barrier models in vitro I: Thin-layer chromatography and high-performance liquid chromatography for the analysis of lipid classes and long-chain polyunsaturated fatty acids , 2002, In Vitro Cellular & Developmental Biology - Animal.
[17] R. Kim. Drugs as P-glycoprotein substrates, inhibitors, and inducers , 2002, Drug metabolism reviews.
[18] Maria do Céu Costa,et al. NMR studies of some rifamycins , 2001 .
[19] H K Kroemer,et al. The role of intestinal P-glycoprotein in the interaction of digoxin and rifampin. , 1999, The Journal of clinical investigation.
[20] V. Ling,et al. Effect of quercetin on Hoechst 33342 transport by purified and reconstituted P-glycoprotein. , 1997, Biochemical pharmacology.
[21] A. Schinkel,et al. P-glycoprotein in the blood-brain barrier of mice influences the brain penetration and pharmacological activity of many drugs. , 1996, The Journal of clinical investigation.
[22] B. Sankaran,et al. P-glycoprotein Is Stably Inhibited by Vanadate-induced Trapping of Nucleotide at a Single Catalytic Site (*) , 1995, The Journal of Biological Chemistry.
[23] Y. Assaraf,et al. Potentiation of anticancer-drug cytotoxicity by multidrug-resistance chemosensitizers involves alterations in membrane fluidity leading to increased membrane permeability. , 1995, European journal of biochemistry.
[24] A. Strosberg,et al. Regulation of gamma‐glutamyl transpeptidase and alkaline phosphatase activities in immortalized rat brain microvessel endothelial cells , 1994, Journal of cellular physiology.
[25] D. Lasič,et al. Liposomes: From Physics to Applications , 1993 .
[26] M. Melamed,et al. Expression of the multidrug resistance gene product (P-glycoprotein) in human normal and tumor tissues. , 1990, The journal of histochemistry and cytochemistry : official journal of the Histochemistry Society.
[27] S. Gupta,et al. Cyclosporin A reverses vincristine and daunorubicin resistance in acute lymphatic leukemia in vitro. , 1986, The Journal of clinical investigation.
[28] T. Tsuruo,et al. Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil. , 1981, Cancer research.
[29] W. D. Mcelroy,et al. Kinetics of the firefly luciferase catalyzed reactions. , 1974, Biochemistry.
[30] Oliver H. Lowry,et al. Protein measurement with the Folin phenol reagent. , 1951, The Journal of biological chemistry.
[31] I. Tucker,et al. Mechanistic studies of the effect of bile salts on rhodamine 123 uptake into RBE4 cells. , 2012, Molecular pharmaceutics.
[32] P. Pávek,et al. Expression and function of p-glycoprotein in normal tissues: effect on pharmacokinetics. , 2010, Methods in molecular biology.
[33] A. Hilgeroth,et al. Impact of Novel MDR Modulators on Human Cancer Cells: Reversal Activities and Induction Studies , 2008, Pharmaceutical Research.
[34] V. Knick,et al. P-Glycoprotein mediated resistance to 5′-nor-anhydro-vinblastine (Navelbine®) , 2007, Investigational New Drugs.
[35] G. Decorti,et al. Induction of proteins involved in multidrug resistance (P-glycoprotein, MRP1, MRP2, LRP) and of CYP 3A4 by rifampicin in LLC-PK1 cells. , 2004, European journal of pharmacology.
[36] T. Grogan,et al. P-glycoprotein expression in malignant lymphoma and reversal of clinical drug resistance with chemotherapy plus high-dose verapamil. , 1991, Journal of clinical oncology : official journal of the American Society of Clinical Oncology.
[37] J. Lakowicz. Principles of fluorescence spectroscopy , 1983 .