CYP1A-mediated metabolism of the Janus kinase-3 inhibitor 4-(4'-hydroxyphenyl)-amino-6,7-dimethoxyquinazoline: structural basis for inactivation by regioselective O-demethylation.
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F. Uckun | E. Sudbeck | C. Mao | R. Malaviya | Hao Chen | Jason C. Thoen | Chun-Lin Chen | Xing-Ping Liu