Structure of the δ-opioid receptor bound to naltrindole
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Aashish Manglik | Brian K. Kobilka | Andrew C. Kruse | Sébastien Granier | William I. Weis | A. Kruse | T. S. Kobilka | Foon Sun Thian | W. Weis | B. Kobilka | A. Manglik | S. Granier | Tong Sun Kobilka
[1] L. Pardo,et al. Crystal structure of the μ-opioid receptor bound to a morphinan antagonist , 2012, Nature.
[2] Bryan L. Roth,et al. Structure of the human kappa opioid receptor in complex with JDTic , 2012, Nature.
[3] A. Kruse,et al. Structure of the human M2 muscarinic acetylcholine receptor bound to an antagonist , 2011, Nature.
[4] R. Stevens,et al. Structure of the human k-opioid receptor in complex with JDTic , 2012 .
[5] K. Befort,et al. The delta opioid receptor: an evolving target for the treatment of brain disorders. , 2011, Trends in pharmacological sciences.
[6] Randy J. Read,et al. Acta Crystallographica Section D Biological , 2003 .
[7] Vincent B. Chen,et al. Correspondence e-mail: , 2000 .
[8] Arthur Christopoulos,et al. A Novel Mechanism of G Protein-coupled Receptor Functional Selectivity , 2008, Journal of Biological Chemistry.
[9] Gebhard F. X. Schertler,et al. Structure of a β1-adrenergic G-protein-coupled receptor , 2008, Nature.
[10] Randy J. Read,et al. Phaser crystallographic software , 2007, Journal of applied crystallography.
[11] B. Delateur,et al. Restoration of Function , 2007, Journal of burn care & research : official publication of the American Burn Association.
[12] Kevin Cowtan,et al. research papers Acta Crystallographica Section D Biological , 2005 .
[13] M. Eguchi. Recent advances in selective opioid receptor agonists and antagonists , 2004, Medicinal research reviews.
[14] W. Delano. The PyMOL Molecular Graphics System , 2002 .
[15] D. Ferguson,et al. Investigation of the selectivity of oxymorphone- and naltrexone-derived ligands via site-directed mutagenesis of opioid receptors: exploring the "address" recognition locus. , 2001, Journal of medicinal chemistry.
[16] H. Akil,et al. Selectivity of mu-opioid receptor determined by interfacial residues near third extracellular loop. , 2000, European journal of pharmacology.
[17] B. O'dowd,et al. Oligomerization of mu- and delta-opioid receptors. Generation of novel functional properties. , 2000, The Journal of biological chemistry.
[18] F. Monsma,et al. Creating a functional opioid alkaloid binding site in the orphanin FQ receptor through site-directed mutagenesis. , 1998, Molecular pharmacology.
[19] J. Dodge,et al. Structure/activity relationships , 1998 .
[20] C. Wahlestedt,et al. Novel “Restoration of Function” Mutagenesis Strategy to Identify Amino Acids of the δ-Opioid Receptor Involved in Ligand Binding* , 1997, The Journal of Biological Chemistry.
[21] Z. Otwinowski,et al. Processing of X-ray diffraction data collected in oscillation mode. , 1997, Methods in enzymology.
[22] C. Chen,et al. Differential binding domains of peptide and non-peptide ligands in the cloned rat kappa opioid receptor. , 1994, The Journal of biological chemistry.
[23] G Vassart,et al. ORL1, a novel member of the opioid receptor family , 1994, FEBS letters.
[24] P. Portoghese,et al. Application of the message-address concept in the design of highly potent and selective non-peptide delta opioid receptor antagonists. , 1988, Journal of medicinal chemistry.
[25] A. Lipkowski,et al. Peptides as receptor selectivity modulators of opiate pharmacophores. , 1986, Journal of medicinal chemistry.
[26] A Goldstein,et al. Specific receptor for the opioid peptide dynorphin: structure--activity relationships. , 1981, Proceedings of the National Academy of Sciences of the United States of America.
[27] D. L. Larson,et al. A novel opioid receptor site directed alkylating agent with irreversible narcotic antagonistic and reversible agonistic activities. , 1980, Journal of medicinal chemistry.
[28] W. A. Sexton,et al. STRUCTURE—ACTIVITY RELATIONSHIPS , 1958, The Journal of pharmacy and pharmacology.