Templated scaffolds of cis- and trans-tetrahydrofuran γ-amino acids: γ-azido-β-hydroxy-tetrahydrofuran-2-carboxylates from pentono-δ-lactones
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[1] O. Ichihara,et al. Synthesis of all diastereomeric methyl 2,5-anhydro-3-deoxy-hexonates: precursors to C-2-deoxynucleosides and THF-templated γ- and δ-amino acids , 2003 .
[2] D. Seebach,et al. On the Biodegradation of β‐Peptides , 2002 .
[3] D. Seebach,et al. Cellular Uptake Studies with β‐Peptides , 2002 .
[4] B. Jaun,et al. γ2‐, γ3‐, and γ2,3,4‐Amino Acids, Coupling to γ‐Hexapeptides: CD Spectra, NMR Solution and X‐ray Crystal Structures of γ‐Peptides , 2002 .
[5] D. Hoyer,et al. Linear, Peptidase-Resistantβ2/β3-Di- andα/β3-Tetrapeptide Derivatives with Nanomolar Affinities to a Human Somatostatin Receptor, Preliminary Communication , 2001 .
[6] S. Gellman,et al. Toward beta-peptide tertiary structure: self-association of an amphiphilic 14-helix in aqueous solution. , 2001, Organic letters.
[7] S. Gellman,et al. Parallel sheet secondary structure in gamma-peptides. , 2001, Journal of the American Chemical Society.
[8] D. Seebach,et al. Synthesis of cyclo-β-tripeptides and their biological in vitro evaluation as antiproliferatives against the growth of human cancer cell lines , 2001 .
[9] W. DeGrado,et al. beta-Peptides: from structure to function. , 2001, Chemical reviews.
[10] D. Seebach,et al. Design, Synthesis, NMR-Solution and X-Ray Crystal Structure ofN-Acyl-γ-dipeptide Amides That Form aβII′-Type Turn , 2001 .
[11] D. Hoyer,et al. Peptide folding induces high and selective affinity of a linear and small beta-peptide to the human somatostatin receptor 4. , 2001, Journal of medicinal chemistry.
[12] T. Claridge,et al. cis - and trans -3-Azido-oxetane-2-carboxylate scaffolds: hexamers of oxetane cis -β-amino acids , 2001 .
[13] C. Toniolo,et al. First Rigid Peptide Foldamers with an Alternating Cis−Trans Amide Sequence. An Oligomeric Building Block for the Construction of New Helices, Large-Ring Cyclic Correlates, and Nanotubes , 2001 .
[14] D. Seebach,et al. The Outstanding Biological Stability of β‐ and γ‐Peptides toward Proteolytic Enzymes: An In Vitro Investigation with Fifteen Peptidases , 2001 .
[15] D. Seebach,et al. Synthesis and CD Spectra in MeCN, MeOH, and H2O ofγ-Oligopeptides with Hydroxy Groups on the Backbone, Preliminary Communication , 2001 .
[16] B. Jaun,et al. Preparation and determination of X-ray-crystal and NMR-solution structures of γ2,3,4-peptides , 2001 .
[17] S. Gellman,et al. 12-Helix Formation in Aqueous Solution with Short β-Peptides Containing Pyrrolidine-Based Residues , 2000 .
[18] S. Gellman,et al. Antibiotics: Non-haemolytic β-amino-acid oligomers , 2000, Nature.
[19] D. Hoyer,et al. The cyclo-β-tetrapeptide (β-HPhe-β-HThr-β-HLys-β-HTrp): synthesis, NMR structure in methanol solution, and affinity for human somatostatin receptors , 2000 .
[20] H. Hauser,et al. β‐Peptides as Inhibitors of Small‐Intestinal Cholesterol and Fat Absorption , 1999 .
[21] S. Hanessian,et al. Synthesis and folding preferences of γ-amino acid oligopeptides: stereochemical control in the formation of a reverse turn and a helix , 1999 .
[22] D. Hoyer,et al. Synthesis and Biological Evaluation of a Cyclo-β-tetrapeptide as a Somatostatin Analogue. , 1999, Angewandte Chemie.
[23] R. Aplin,et al. An octameric carbopeptoid; secondary structure in octameric and tetrameric 5-aminomethyl-tetrahydrofuran-2-carboxylates , 1999 .
[24] S. Durell,et al. Formation of Short, Stable Helices in Aqueous Solution by β-Amino Acid Hexamers , 1999 .
[25] M. Moloney,et al. Novel peptidomimetic structures: enantioselective synthesis of conformationally constrained lysine, ornithine and alanine analogues from pyroglutamic acid , 1999 .
[26] S. Michnick,et al. Design of Secondary Structures in Unnatural Peptides: Stable Helical γ-Tetra-, Hexa-, and Octapeptides and Consequences of α-Substitution , 1998 .
[27] Samuel H. Gellman,et al. Foldamers: A Manifesto , 1998 .
[28] B. Jaun,et al. γ‐Peptides Forming More Stable Secondary Structures than α‐Peptides: Synthesis and helical NMR‐solution structure of the γ‐hexapeptide analog of H‐(Val‐Ala‐Leu)2‐OH , 1998 .
[29] M. Sansom,et al. Secondary structure in oligomers of carbohydrate amino acids , 1998 .
[30] N. Chandler,et al. N-α-benzoyl-cis-4-amino-L-proline: A γ-turn mimetic , 1996 .
[31] C. Bichard,et al. Acid-catalysed transformation of α-trifluoromethanesulfonates of γ- and δ-lactones into 2,5-disubstituted homochiral tetrahydrofurans , 1993 .
[32] F. Gasparini,et al. Total, asymmetric synthesis of (1r-1-c-(6′-amino-7′h-purin-8′-yl)-1,4-anhydro-3-azido-2,3-dideoxy-d-erythro-pentitol. , 1992 .
[33] C. Toniolo,et al. Structural characterization of the .beta.-bend ribbon spiral: crystallographic analysis of two long (L-Pro-Aib)n sequential peptides , 1992 .
[34] C. Bichard,et al. The ring contraction of δ-lactones with leaving group α-substituents : a strategy for the synthesis of 2,5-disubstituted highly functionalised homochiral tetrahydrofurans , 1992 .
[35] D. Osguthorpe,et al. Design of a natural cis peptide bond motif to form type VI β-turn mimetic , 1992 .
[36] Paul W Smith,et al. Synthesis of (2R,3S,4R)-3,4-dihydroxyproline from D-ribonolactone; an approach to the synthesis of polyfunctionalised D-amino acids from sugar lactones. X-Ray molecular structures of 2-azido-3,4-O-(R)-benzylidene-2-deoxy-D-ribono-1,5-lactone, 2-azido-2-deoxy-D-ribono-1,4-lactone, and (2R,3S,3R)-3,4- , 1987 .
[37] R. Allan,et al. Synthesis of analogues of GABA. XII. cis- and trans-4-Aminotetrahydrofuran-2-carboxylic acid , 1984 .