One pot synthesis using supported reagents system KSCN/SiO2–RNH3OAc/Al2O3: synthesis of 2-aminothiazoles and N-allylthioureas

[1]  T. Takido,et al.  One-Pot Synthesis of Benzo[b]thiophenes and Naphtho[2,1-b]thiophenes in the Presence of Acidic and Basic Supported Reagents , 2005 .

[2]  T. Takido,et al.  One-pot synthesis of N-allylthioureas using supported reagents , 2005 .

[3]  O. Repič,et al.  Reductive alkylation of thioureas: a highly practical synthesis of unsymmetrical N,N′-disubstituted thioureas , 2004 .

[4]  S. Lang,et al.  Thiourea inhibitors of herpes viruses. Part 2: N-Benzyl-N'-arylthiourea inhibitors of CMV. , 2004, Bioorganic & medicinal chemistry letters.

[5]  Jiyoun Lee,et al.  Analysis of structure-activity relationships with the N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea template for vanilloid receptor 1 antagonism. , 2004, Bioorganic & medicinal chemistry.

[6]  Y. Harigaya,et al.  A clay-mediated, regioselective synthesis of 2-(aryl/alkyl)amino-thiazolo[4,5-c]carbazoles , 2004 .

[7]  A. Katritzky,et al.  1-(Alkyl/arylthiocarbamoyl)benzotriazoles as stable isothiocyanate equivalents: synthesis of Di- and trisubstituted thioureas. , 2004, The Journal of organic chemistry.

[8]  T. Takido,et al.  One-pot synthesis of α-bromoesters and ketones from β-ketoesters and diketones using supported reagents system , 2004 .

[9]  M. Serrano-Wu,et al.  Regioselective Synthesis of 3-(Heteroaryl)-iminothiazolidin-4-ones , 2004 .

[10]  J. B. Christensen,et al.  Facile synthesis of aliphatic isothiocyanates and thioureas on solid phase using peptide coupling reagents , 2004 .

[11]  Wei Zhang,et al.  Fluorous electrophilic scavengers for solution-phase parallel synthesis , 2003 .

[12]  R. Maggi,et al.  MCM-41-TBD as a new, efficient, supported heterogeneous catalyst for the synthesis of thioureas , 2002 .

[13]  Tadashi Aoyama,et al.  One-pot synthesis of 2-aminothiazoles using supported reagents , 2002 .

[14]  J. Rudolph.  Facile Access to N-Thiazolyl α-Amino Acids from α-Bromo Ketones and α-Amino Acids , 2000 .

[15]  A. Loupy,et al.  Synthesis of 1-benzoyl-3-alkylthioureas by transamidation under microwave in dry media† , 2000 .

[16]  S. Samal,et al.  1-(Methyldithiocarbonyl)imidazole: a Useful Thiocarbonyl Transfer Reagent for Synthesis of Substituted Thioureas , 2000 .

[17]  T. Kurz,et al.  CVCLIZATION OF THIOCYANATO MALONATES WITH HYDROXYLAMINES TO 5-CARBOXYALKYL-4-OXO-THIAZOLI(DI)NES , 1999 .

[18]  A. Corradi,et al.  Condensation of thiourea derivatives with carbonyl compounds: one-pot synthesis of N-alkyl-1,3-thiazol-2-amines and of 3-alkyl-1,3-thiazolimines , 1999 .

[19]  M. Kodomari,et al.  One-Pot Synthesis Using Supported Reagents System: Conversion of β-Dicarbonyl Compounds to α-Thiocyano-β-dicarbonyl Compounds Using CuBr2/Al2O3-KSCN/SiO2 , 1998 .

[20]  I. Lagoja,et al.  Expedient Synthesis of N-Substituted 2-Aminothiazoles , 1998 .

[21]  J. Flygare,et al.  Solid-Phase Synthesis of 2-Aminothiazoles. , 1998, The Journal of organic chemistry.

[22]  A. W. Dean,et al.  A convenient procedure for the solution phase preparation of 2-aminothiazole combinatorial libraries , 1996 .

[23]  J M Morin,et al.  Phenethylthiazolethiourea (PETT) compounds, a new class of HIV-1 reverse transcriptase inhibitors. 1. Synthesis and basic structure-activity relationship studies of PETT analogs. , 1995, Journal of medicinal chemistry.

[24]  J. J. Parlow.  SIMULTANEOUS MULTISTEP SYNTHESIS USING POLYMERIC REAGENTS , 1995 .

[25]  M. Kodomari,et al.  Direct allylation of aromatic compounds with allylic chloride using the supported reagents system ZnCl2/SiO2–K2CO3/Al2O3 , 1995 .

[26]  H. Ishikawa,et al.  Synthesis and anti-pseudomonal activity of new 2-isocephems with a dihydroxypyridone moiety at C-7 , 1994 .

[27]  C. Garg,et al.  A Novel Thallium(III)‐Mediated Approach to 2‐Substituted Thiazoles from Enolizable Ketones. , 2010 .

[28]  A. Doherty,et al.  Structure-activity relationships of a series of 2-amino-4-thiazole-containing renin inhibitors. , 1992, Journal of medicinal chemistry.

[29]  H. Yamanaka,et al.  [Synthesis of 4,5-diarylthiazole derivatives as blood platelet aggregation inhibitors]. , 1990, Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan.

[30]  P. Young,et al.  3-[1-(2-Benzoxazolyl)hydrazino]propanenitrile derivatives: inhibitors of immune complex induced inflammation. , 1988, Journal of medicinal chemistry.

[31]  J. Clark,et al.  Inorganic-solid-supported potassium thiocyanate: study of reagent preparation and a convenient synthesis of tert-alkyl thiocyanates , 1987 .

[32]  K. D. Hargrave,et al.  N-(4-substituted-thiazolyl)oxamic acid derivatives, a new series of potent, orally active antiallergy agents. , 1983, Journal of medicinal chemistry.

[33]  M. Kodomari,et al.  A CONVENIENT SYNTHESIS OF ALKYL THIOCYANATES USING SILICA GEL SUPPORTED POTASSIUM THIOCYANATE , 1983 .

[34]  P. D. Maria,et al.  Tautomerism of aminothiazoles. pKBH+ Values of 2-aminothiazoles and of some model imines , 1982 .

[35]  P. D. Maria,et al.  Electrical effects in substituted thiazoles. pKa Values of some 5-substituted 2-aminothiazoles and 5-substituted 2-NN-dimethylaminothiazoles , 1980 .

[36]  Satyavan Sharma.  THIOPHOSGENE IN ORGANIC SYNTHESIS , 1978 .

[37]  E. Bergmann.  321. The rearrangement of thiocyanates into isothiocyanates , 1935 .