Synthesis and Structure−Activity Relationships of a Novel Series of 2,3,5,6,7,9-Hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-Dioxide KATP Channel Openers: Discovery of (−)-(9S)-9-(3-Bromo-4-fluorophenyl)-2,3,5,6,7,9- hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-Dioxide (A-278637), a Potent KATP Open
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J. Sullivan | R. Henry | J. Brioni | M. Gopalakrishnan | R. Tang | Henry Q. Zhang | P. Kym | M. Kort | R. Gregg | M. Brune | S. Buckner | A. Daza | M. Holladay | Ivan Milicic | Michael C. Fitzgerald | M. Coghlan | I. Drizin | W. Carroll | K. Whiteaker | R. Altenbach | H. Bai | T. Fey | S. Turner | Linda L. King | Yiyuan Chen | L. Yi | Christopher Cassidy