Preclinical evaluation of new and highly potent analogues of octreotide for predictive imaging and targeted radiotherapy.
暂无分享,去创建一个
Martin A Walter | M. Walter | J. Reubi | Véronique Eltschinger | H. Maecke | Jean Claude Reubi | Mihaela Ginj | Helmut R Maecke | Jianhua Chen | Veronique Eltschinger | M. Ginj | Jianhua Chen
[1] J. Stewart. Solid Phase Peptide Synthesis , 1984 .
[2] E. P. Krenning,et al. Somatostatin receptor scintigraphy with [111In-DTPA-d-Phe1]- and [123I-Tyr3]-octreotide: the Rotterdam experience with more than 1000 patients , 1993, European Journal of Nuclear Medicine.
[3] E. Krenning,et al. Somatostatin receptors in human cancer: Incidence, characteristics, functional correlates and clinical implications , 1992, The Journal of Steroid Biochemistry and Molecular Biology.
[4] L. Travaini,et al. Biokinetics and dosimetry in patients administered with 111In-DOTA-Tyr3-Octreotide: Implications for internal radiotherapy with 90Y-DOTATOC , 2000 .
[5] S. Lamberts,et al. Somatostatin receptor subtypes in human thymoma and inhibition of cell proliferation by octreotide in vitro. , 2000, The Journal of clinical endocrinology and metabolism.
[6] J. Edwardson,et al. Fates of endocytosed somatostatin sst2 receptors and associated agonists. , 1998, The Biochemical journal.
[7] J. Laissue,et al. Immunohistochemical localization of somatostatin receptors sst2A in human tumors. , 1998, The American journal of pathology.
[8] A. Schally,et al. Human ovarian cancers express somatostatin receptors. , 2000, The Journal of clinical endocrinology and metabolism.
[9] G. Capellá,et al. Loss of sst2 somatostatin receptor gene expression in human pancreatic and colorectal cancer. , 1996, Cancer research.
[10] D. Hoyer,et al. Differential expression of five somatostatin receptor subtypes, SSTR1-5, in the CNS and peripheral tissue. , 1994, Digestion.
[11] J. Reubi,et al. Concomitant expression of several peptide receptors in neuroendocrine tumours: molecular basis for in vivo multireceptor tumour targeting , 2003, European Journal of Nuclear Medicine and Molecular Imaging.
[12] G. Meno-Tetang,et al. SOM230: a novel somatostatin peptidomimetic with broad somatotropin release inhibiting factor (SRIF) receptor binding and a unique antisecretory profile. , 2002, European journal of endocrinology.
[13] J. Schmitt,et al. Frequent expression of immunoreactive somatostatin receptors in cervical and endometrial cancer. , 2003, Gynecologic oncology.
[14] L. Gordon,et al. Randomized controlled trial of yttrium-90-labeled ibritumomab tiuxetan radioimmunotherapy versus rituximab immunotherapy for patients with relapsed or refractory low-grade, follicular, or transformed B-cell non-Hodgkin's lymphoma. , 2002, Journal of clinical oncology : official journal of the American Society of Clinical Oncology.
[15] C. Waldherr,et al. The clinical value of [90Y-DOTA]-D-Phe1-Tyr3-octreotide (90Y-DOTATOC) in the treatment of neuroendocrine tumours: a clinical phase II study. , 2001, Annals of oncology : official journal of the European Society for Medical Oncology.
[16] J. Lewis,et al. Comparison of four 64Cu-labeled somatostatin analogues in vitro and in a tumor-bearing rat model: evaluation of new derivatives for positron emission tomography imaging and targeted radiotherapy. , 1999, Journal of medicinal chemistry.
[17] T. Visser,et al. Yttrium-90 and indium-111 labelling, receptor binding and biodistribution of [DOTA0,d-Phe1,Tyr3]octreotide, a promising somatostatin analogue for radionuclide therapy , 1997, European Journal of Nuclear Medicine.
[18] R. Lefkowitz,et al. Signalling: Seven-transmembrane receptors , 2002, Nature Reviews Molecular Cell Biology.
[19] A. Schally,et al. RAPID COMMUNICATION: Human Ovarian Cancers Express Somatostatin Receptors , 2000 .
[20] P. Smith-Jones,et al. The somatostatin receptor-targeted radiotherapeutic [90Y-DOTA-dPhe1,Tyr3]octreotide (90Y-SMT 487) eradicates experimental rat pancreatic CA 20948 tumours , 1998, European Journal of Nuclear Medicine.
[21] Eva Forssell-Aronsson,et al. and Somatostatin Receptor Subtypes in Thyroid Tumors , 2000 .
[22] J. Reubi,et al. A new peptidic somatostatin agonist with high affinity to all five somatostatin receptors. , 2002, European journal of pharmacology.
[23] S. Schulz,et al. Differential β-Arrestin Trafficking and Endosomal Sorting of Somatostatin Receptor Subtypes* , 2004, Journal of Biological Chemistry.
[24] S. Melmed,et al. Expression of three somatostatin receptor subtypes in pituitary adenomas: evidence for preferential SSTR5 expression in the mammosomatotroph lineage. , 1994, The Journal of clinical endocrinology and metabolism.
[25] M. Hennig,et al. Radiometal‐Labelled Macrocyclic Chelator‐Derivatised Somatostatin Analogue with Superb Tumour‐Targeting Properties and Potential for Receptor‐Mediated Internal Radiotherapy , 1999 .
[26] B. Bernard,et al. DOTA-NOC, a high-affinity ligand of somatostatin receptor subtypes 2, 3 and 5 for labelling with various radiometals , 2003, European Journal of Nuclear Medicine and Molecular Imaging.
[27] T. O'Dorisio,et al. Radiolabeled peptides in diagnosis and tumor imaging: clinical overview. , 2002, Seminars in nuclear medicine.
[28] E P Krenning,et al. Comparison of (111)In-labeled somatostatin analogues for tumor scintigraphy and radionuclide therapy. , 1998, Cancer research.
[29] G. Mengod,et al. Expression and localization of somatostatin receptor SSTR1, SSTR2, and SSTR3 messenger RNAs in primary human tumors using in situ hybridization. , 1994, Cancer research.
[30] Y. Menda,et al. Evaluating the clinical effectiveness of 90Y-SMT 487 in patients with neuroendocrine tumors. , 2003, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[31] R. Sheppard,et al. Solid phase peptide synthesis : a practical approach , 1989 .
[32] Mu Wang,et al. Subcellular localization of radiolabeled somatostatin analogues: implications for targeted radiotherapy of cancer. , 2003, Cancer research.
[33] J. Laissue,et al. Somatostatin receptor sst1–sst5 expression in normal and neoplastic human tissues using receptor autoradiography with subtype-selective ligands , 2001, European Journal of Nuclear Medicine.
[34] E. Krenning,et al. [177Lu-DOTA0,Tyr3]octreotate: comparison with [111In-DTPA0]octreotide in patients , 2001, European Journal of Nuclear Medicine.
[35] J. Reubi,et al. Affinity profiles for human somatostatin receptor subtypes SST1–SST5 of somatostatin radiotracers selected for scintigraphic and radiotherapeutic use , 2000, European Journal of Nuclear Medicine.
[36] J. Mueller‐Brand,et al. Yttrium-90-labelled somatostatin-analogue for cancer treatment , 1998, The Lancet.
[37] I. Sobhani,et al. Detection of neuroendocrine tumors: 99mTc-P829 scintigraphy compared with 111In-pentetreotide scintigraphy. , 2002, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[38] M. Papotti,et al. Expression of somatostatin receptor types 2, 3 and 5 in biopsies and surgical specimens of human lung tumours , 2001, Virchows Archiv.