Catalyst‐Free and One‐Pot Procedure for Fast Formation of α‐Ketoamides Using α‐Oxocarboxylic Acids and Amines at Room Temperature

[1]  Kuan Zhang,et al.  Correction: nBu4NI-Mediated oxidation of methyl ketones to α-ketoamides: using ammonium, primary and secondary amine-salt as an amine moiety. , 2017, Organic & biomolecular chemistry.

[2]  Yiping Chen,et al.  Solvent-free one-pot oxidation of ethylarenes for the preparation of α-ketoamides under mild conditions , 2017 .

[3]  Shiuh-Tzung Liu,et al.  One pot synthesis of α-ketoamides from ethylarenes and amines: a metal free difunctionalization strategy. , 2016, Organic & biomolecular chemistry.

[4]  N. Zhu,et al.  Copper-TEMPO-catalyzed synthesis of α-ketoamides via tandem sp(3)C-H aerobic oxidation and amination of phenethyl alcohol derivatives. , 2016, Organic & biomolecular chemistry.

[5]  M. Aga,et al.  SeO2 mediated efficient synthesis of amides and α-ketoamides of secondary amines with wide substrate scope , 2016 .

[6]  N. Shankaraiah,et al.  Microwave-assisted direct oxidative synthesis of α-ketoamides from aryl methyl ketones and amines by a water soluble Cu(I)-complex , 2016 .

[7]  Qingwen Li,et al.  A two-step continuous synthesis of α-ketoamides and α-amino ketones from 2° benzylic alcohols using hydrogen peroxide as an economic and benign oxidant , 2016 .

[8]  G. Sekar,et al.  Metal free synthesis of α-keto amides from 2-hydroxy acetophenones through domino alcohol oxidation–oxidative amidation reaction , 2015 .

[9]  Bikram Singh,et al.  Selective C–Si Bond Formation through C–H Functionalization , 2015 .

[10]  G. Sekar,et al.  Metal free one-pot synthesis of α-ketoamides from terminal alkenes , 2015 .

[11]  B. A. Shah,et al.  Copper(II)‐Triflate‐Catalyzed Oxidative Amidation of Terminal Alkynes: A General Approach to α‐Ketoamides , 2015 .

[12]  B. A. Shah,et al.  Iodine‐Promoted Oxidative Amidation of Terminal Alkenes – Synthesis of α‐Ketoamides, Benzothiazoles, and Quinazolines , 2015 .

[13]  G. Sekar,et al.  Copper-Catalyzed One-Pot Synthesis of α-Ketoamides from 1-Arylethanols , 2015 .

[14]  G. Sekar,et al.  Iron‐TEMPO‐Catalyzed Domino Aerobic Alcohol Oxidation/Oxidative Cross‐Dehydrogenative Coupling for the Synthesis of α‐Keto Amides , 2014 .

[15]  N. Iranpoor,et al.  Direct Nickel‐Catalyzed Amination of Phenols via CO Bond Activation using 2,4,6‐Trichloro‐1,3,5‐triazine (TCT) as Reagent , 2014 .

[16]  B. A. Shah,et al.  A general metal free approach to α-ketoamides via oxidative amidation-diketonization of terminal alkynes. , 2014, Chemical communications.

[17]  P. Sun,et al.  The syntheses of α-ketoamides via(n)Bu4NI-catalyzed multiple sp(3)C-H bond oxidation of ethylarenes and sequential coupling with dialkylformamides. , 2014, Organic & biomolecular chemistry.

[18]  R. Vishwakarma,et al.  Metal-free oxidative amidation of 2-oxoaldehydes: a facile access to α-ketoamides. , 2014, Organic letters.

[19]  Hua Wang,et al.  Copper-catalyzed oxidative condensation of α-oxocarboxylic acids with formamides: synthesis of α-ketoamides. , 2013, Organic & biomolecular chemistry.

[20]  Lei Wang,et al.  Silver-catalyzed amidation of benzoylformic acids with tertiary amines via selective carbon-nitrogen bond cleavage. , 2013, Organic & biomolecular chemistry.

[21]  Lei Wang,et al.  Cu(II)-catalyzed decarboxylative acylation of acyl C-H of formamides with α-oxocarboxylic acids leading to α-ketoamides. , 2013, Chemical communications.

[22]  M. Shiro,et al.  Study on 1,3,5-triazine chemistry in dehydrocondensation: gauche effect on the generation of active triazinylammonium species. , 2012, Chemistry.

[23]  K. R. Prabhu,et al.  NIS-catalyzed reactions: amidation of acetophenones and oxidative amination of propiophenones. , 2012, Chemistry.

[24]  Huayou Hu,et al.  Coupling of methyl ketones and primary or secondary amines leading to α-ketoamides. , 2012, The Journal of organic chemistry.

[25]  L. Zhang,et al.  Copper-catalyzed aerobic oxidative cross-dehydrogenative coupling of amine and α-carbonyl aldehyde: a practical and efficient approach to α-ketoamides with wide substrate scope. , 2012, Organic letters.

[26]  Feng-Tian Du,et al.  Copper-catalyzed direct oxidative synthesis of α-ketoamides from aryl methyl ketones, amines, and molecular oxygen , 2012 .

[27]  L. Zhang,et al.  Copper-catalyzed aerobic oxidative coupling of aryl acetaldehydes with anilines leading to α-ketoamides. , 2011, Angewandte Chemie.

[28]  De‐Xian Wang,et al.  Highly efficient and expedient synthesis of 5-hydroxy-1H-pyrrol-2-(5H)-ones from FeCl3-catalyzed tandem intramolecular enaminic addition of tertiary enamides to ketones and 1,3-hydroxy rearrangement. , 2010, Organic letters.

[29]  J. Sivaguru,et al.  Photochemical type II reaction of atropchiral benzoylformamides to point chiral oxazolidin-4-ones. Axial chiral memory leading to enantiomeric resolution of photoproducts. , 2010, Chemical communications.

[30]  Q. Zhang,et al.  Ag-containing all-carbon 1,3-dipoles: generation and formal cycloaddition for furo[3,2-b]-beta/gamma-lactams. , 2010, Chemical communications.

[31]  Ning Jiao,et al.  Dioxygen activation under ambient conditions: Cu-catalyzed oxidative amidation-diketonization of terminal alkynes leading to alpha-ketoamides. , 2010, Journal of the American Chemical Society.

[32]  De‐Xian Wang,et al.  Cr(III)(salen)Cl catalyzed enantioselective intramolecular addition of tertiary enamides to ketones: a general access to enantioenriched 1H-pyrrol-2(3H)-one derivatives bearing a hydroxylated quaternary carbon atom. , 2009, Journal of the American Chemical Society.

[33]  H. Gronemeyer,et al.  Retinoid receptor subtype-selective modulators through synthetic modifications of RARgamma agonists. , 2009, Bioorganic & medicinal chemistry.

[34]  M. Kanai,et al.  Enantioselective synthesis of SM-130686 based on the development of asymmetric Cu(I)F catalysis to access 2-oxindoles containing a tetrasubstituted carbon. , 2009, Journal of the American Chemical Society.

[35]  R. Bates,et al.  Synthesis of (-)-MonomorineI , 2009 .

[36]  D. A. Klumpp,et al.  Superacid-promoted reactions of alpha-ketoamides and related systems. , 2008, The Journal of organic chemistry.

[37]  G. Błotny Recent applications of 2,4,6-trichloro-1,3,5-triazine and its derivatives in organic synthesis , 2006 .

[38]  Wei Zhang,et al.  Fluorous 2,4-Dichloro-1,3,5-triazine (F-DCT) as Amide Coupling Agent. , 2006, QSAR & combinatorial science.

[39]  J. S. Carey,et al.  Analysis of the reactions used for the preparation of drug candidate molecules. , 2006, Organic & biomolecular chemistry.

[40]  M. Gu,et al.  Design, synthesis, and biological evaluation of isoquinoline-1,3,4-trione derivatives as potent caspase-3 inhibitors. , 2006, Journal of medicinal chemistry.

[41]  G. Signore,et al.  Organometallic alkylation of 2-chloro-4,6-dimethoxy-1,3,5-triazine: a study , 2005 .

[42]  R. Singh,et al.  One-Pot Route to New α,α-Difluoroamides and α-Ketoamides , 2003 .

[43]  D. Cunningham,et al.  alpha-Keto amides as precursors to heterocycles--generation and cycloaddition reactions of piperazin-5-one nitrones. , 2003, Organic & biomolecular chemistry.

[44]  B. Patrick,et al.  Control of Enantioselectivity in the Photochemical Conversion of α-Oxoamides into β-Lactam Derivatives , 2002 .

[45]  B. Kolesińska,et al.  A novel generation of coupling reagents. Enantiodifferentiating coupling reagents prepared in situ from 2-chloro-4,6-dimethoxy-1,3,5-triazine (CDMT) and chiral tertiary amines. , 2001, The Journal of organic chemistry.

[46]  G. Giacomelli,et al.  An easy and convenient synthesis of Weinreb amides and hydroxamates. , 2001, The Journal of organic chemistry.

[47]  M. Taddei,et al.  Solid-Supported Chloro[1,3,5]triazine. A Versatile New Synthetic Auxiliary for the Synthesis of Amide Libraries , 1999 .

[48]  A. Chamberlin,et al.  Chemical Synthesis of Natural Product Peptides: Coupling Methods for the Incorporation of Noncoded Amino Acids into Peptides. , 1997, Chemical reviews.

[49]  Takakazu Yamamoto,et al.  Catalytic double carbonylation of organohalogen compounds promoted by palladium complexes , 1983 .