Eaton’s reagent-mediated metal-free and efficient synthesis of NH-sulfoximines

[1]  R. Vishwakarma,et al.  Metal-Free, Phosphonium Salt-Mediated Sulfoximination of Azine N-Oxides: Approach for the Synthesis of N-Azine Sulfoximines. , 2016, The Journal of organic chemistry.

[2]  L. Degennaro,et al.  Transfer of Electrophilic NH Using Convenient Sources of Ammonia: Direct Synthesis of NH Sulfoximines from Sulfoxides , 2016, Angewandte Chemie.

[3]  Dominique M. Roberge,et al.  Development of a Continuous Flow Sulfoxide Imidation Protocol Using Azide Sources under Superacidic Conditions , 2015 .

[4]  R. Luisi,et al.  Synthesis of Sulfoximine Carbamates by Rhodium-Catalyzed Nitrene Transfer of Carbamates to Sulfoxides. , 2015, The Journal of organic chemistry.

[5]  C. Bolm,et al.  Sulfur imidations: access to sulfimides and sulfoximines. , 2015, Chemical Society reviews.

[6]  Jason G. Kettle,et al.  General synthetic strategies towards N-alkyl sulfoximine building blocks for medicinal chemistry and the use of dimethylsulfoximine as a versatile precursor , 2014 .

[7]  N. Richards,et al.  Rhodium-catalyzed direct synthesis of unprotected NH-sulfoximines from sulfoxides. , 2014, Chemical communications.

[8]  C. Bolm,et al.  Light-induced ruthenium-catalyzed nitrene transfer reactions: a photochemical approach towards N-acyl sulfimides and sulfoximines. , 2014, Angewandte Chemie.

[9]  C. Bolm,et al.  Iron-catalyzed imidative kinetic resolution of racemic sulfoxides. , 2014, Chemistry.

[10]  U. Lücking Sulfoximines: a neglected opportunity in medicinal chemistry. , 2013, Angewandte Chemie.

[11]  Julia M. Schulze,et al.  The Lab Oddity Prevails: Discovery of Pan‐CDK Inhibitor (R)‐S‐Cyclopropyl‐S‐(4‐{[4‐{[(1R,2R)‐2‐hydroxy‐1‐methylpropyl]oxy}‐5‐(trifluoromethyl)pyrimidin‐2‐yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer , 2013, ChemMedChem.

[12]  C. Bolm,et al.  N‐Cyano Sulfoximines: COX Inhibition, Anticancer Activity, Cellular Toxicity, and Mutagenicity , 2013, ChemMedChem.

[13]  Jigar S. Patel,et al.  Synthesis and structure-activity relationship of potent, selective and orally active anthranilamide-based factor Xa inhibitors: application of weakly basic sulfoximine group as novel S4 binding element. , 2012, European journal of medicinal chemistry.

[14]  J. Marrot,et al.  Sulfilimines and Sulfoximines by Reaction of Nitriles with Perfluoroalkyl Sulfoxides , 2009 .

[15]  C. Bolm,et al.  Diphenylphosphanylsulfoximines as ligands in iridium-catalyzed asymmetric imine hydrogenations. , 2005, Angewandte Chemie.

[16]  C. Bolm,et al.  Highly modular synthesis of C1-symmetric aminosulfoximines and their use as ligands in copper-catalyzed asymmetric Mukaiyama-aldol reactions. , 2005, Chemistry.

[17]  A. White,et al.  Asymmetric decarboxylative Claisen rearrangement reactions of sulfoximine-substituted allylic tosylacetic esters. , 2005, The Journal of organic chemistry.

[18]  P. S. Kumar,et al.  Theoretical studies on the S–N interactions in sulfoximine , 2005 .

[19]  C. Bolm,et al.  Cu(OAc)2-catalyzed N-arylations of sulfoximines with aryl boronic acids. , 2005, Organic letters.

[20]  C. Bolm,et al.  C1-Symmetric Aminosulfoximines as Ligands in Copper-Catalyzed Carbonyl-Ene Reactions , 2005 .

[21]  T. Kensler,et al.  Potent, Selective and Low-Calcemic Inhibitors of CYP24 Hydroxylase: 24-Sulfoximine Analogues of the Hormone 1α,25-Dihydroxyvitamin D3 , 2004 .

[22]  C. Bolm,et al.  C(1)-symmetric sulfoximines as ligands in copper-catalyzed asymmetric Mukaiyama-type aldol reactions. , 2004, Angewandte Chemie.

[23]  C. Bolm,et al.  Synthetic and spectroscopic investigation of N-acylated sulfoximines. , 2004, Chemistry.

[24]  Parthasarathi Das,et al.  Asymmetric Synthesis of Cycloalkenyl and Alkenyloxiranes From Allylic Sulfoximines and Aldehydes and Application to Solid‐Phase Synthesis , 2004 .

[25]  C. Bolm,et al.  Rhodium-catalyzed imination of sulfoxides and sulfides: efficient preparation of N-unsubstituted sulfoximines and sulfilimines. , 2004, Organic letters.

[26]  C. Bolm,et al.  A new class of C1-symmetric monosulfoximine ligands for enantioselective hetero Diels-Alder reactions. , 2003, Chemical communications.

[27]  C. Bolm,et al.  The stability of pseudopeptides bearing sulfoximines as chiral backbone modifying element towards proteinase K. , 2003, Bioorganic & medicinal chemistry letters.

[28]  Stefan Koep,et al.  Asymmetric synthesis of unsaturated, fused bicyclic proline analogues through amino alkylation of cyclic bis(allylsulfoximine)titanium complexes and migratory cyclization of delta-amino alkenyl aminosulfoxonium salts. , 2003, Journal of the American Chemical Society.

[29]  C. Barnes,et al.  Benzothiazines in synthesis. Formal syntheses of (+)-curcumene and (+)-curcuphenol , 2003 .

[30]  Xuechuan Hong,et al.  The Intramolecular, Stereoselective Addition of Sulfoximine Carbanions to α,β-Unsaturated Esters , 2003 .

[31]  C. Bolm,et al.  C2-symmetric bissulfoximines as ligands in copper-catalyzed enantioselective Diels-Alder reactions. , 2003, Organic letters.

[32]  C. Bolm,et al.  Turn formation initiated by a bissulfoximine motif: synthesis and structural investigation. , 2002, Organic letters.

[33]  C. Bolm,et al.  Highly enantioselective hetero-Diels-Alder reactions catalyzed by a C(2)-symmetric bis(sulfoximine) copper(II) complex. , 2001, Journal of the American Chemical Society.

[34]  C. Bolm,et al.  Synthesis of pseudopeptides with sulfoximines as chiral backbone modifying elements. , 2001, Chemistry.

[35]  M. Harmata,et al.  A One‐Pot, One‐Operation [3+3] Annulation Approach to Benzothiazines , 1999 .

[36]  H. Bailey L-S,R-buthionine sulfoximine: historical development and clinical issues. , 1998, Chemico-biological interactions.

[37]  Jochen R. Brandt,et al.  An efficient resolution of (±)-S-methyl-S-phenylsulfoximine with (+)-10-camphorsulfonic acid by the method of half-quantities , 1997 .

[38]  S. Claeson,et al.  Stereochemistry of the formation of endocyclic sulfoximides from o-carboxyphenyl sulfoxides , 1996 .

[39]  C. Bolm,et al.  Optically Active β-Hydroxy Sulfoximine/Nickel Complexes as Catalysts for the Enantioselective Conjugate Addition of Diethylzinc to Chalcones , 1992 .

[40]  W. L. Mock,et al.  Sulfoximine and sulfodiimine transition state analog inhibitors for carboxypeptidase A , 1989 .

[41]  G. Olah,et al.  Trimethylsilyl azide/triflic acid, a highly efficient electrophilic aromatic amination reagent , 1989 .

[42]  G. Olah Onium ions. 26. Aminodiazonium ions: preparation, proton, carbon-13, and nitrogen-15 NMR structural studies, and electrophilic amination of aromatics , 1983 .

[43]  M. Anderson,et al.  Inhibition of glutathione biosynthesis by prothionine sulfoximine (S-n-propyl homocysteine sulfoximine), a selective inhibitor of gamma-glutamylcysteine synthetase. , 1979, The Journal of biological chemistry.

[44]  N. Kunieda,et al.  OXYGEN EXCHANGE AND RACEMIZATION REACTIONS OF DIARYL SULFOXIDES IN SULFURIC ACID IN THE PRESENCE OF POTASSIUM CHLORIDE , 1977 .

[45]  Carl R. Johnson,et al.  Chemistry of sulfoxides and related compounds. XLIX. Synthesis of optically active sulfoximines from optically active sulfoxides , 1974 .

[46]  P. Eaton,et al.  Phosphorus pentoxide-methanesulfonic acid. Convenient alternative to polyphosphoric acid , 1973 .

[47]  Carl R. Johnson Utilization of sulfoximines and derivatives as reagents for organic synthesis , 1973 .

[48]  Carl R. Johnson,et al.  Chemistry of sulfoxides and related compounds. XLV. Asymmetric syntheses using optically active oxosulfonium alkylides , 1973 .

[49]  Y. Tamura,et al.  Synthesis and some properties of O-acyl-and O-nitrophenylhydroxylamines. , 1973, The Journal of organic chemistry.

[50]  Y. Tamura,et al.  A novel method for sulfilimines and sulfoximines , 1972 .

[51]  G. Satzinger,et al.  3‐Oxobenzo[d]isothia(IV)‐azole 1‐Oxides , 1971 .

[52]  Carl R. Johnson,et al.  Chemistry of sulfoxides and related compounds. XXVI. Preparation and synthetic applications of (dimethylamino)phenyloxosulfonium methylide , 1970 .

[53]  J. K. Whitehead,et al.  287. Preparation and properties of some aliphatic sulphoximines , 1952 .

[54]  E. McDermott,et al.  Action of nitrogen trichloride on certain proteins II. Synthesis of methionine sulphoximine and other sulphoximines , 1951, Proceedings of the Royal Society of London. Series B - Biological Sciences.

[55]  T. Moran,et al.  Action of Nitrogen Trichloride on Proteins : Progress in the Isolation of the Toxic Factor , 1949, Nature.