Novel oxybispyridylboronic acids: synthesis and study of their reactivity in Suzuki-type cross-coupling reactions
暂无分享,去创建一个
[1] Aurélien Lesnard,et al. Synthesis of novel halo-oxybispyridines, new building blocks in cholinergic medicinal chemistry , 2006 .
[2] T. Liljefors,et al. Neuronal nicotinic acetylcholine receptors: structural revelations, target identifications, and therapeutic inspirations. , 2005, Journal of medicinal chemistry.
[3] A. Batsanov,et al. 2-Ethoxy-3-pyridylboronic acid: a versatile reagent for the synthesis of highly-functionalised 3-aryl/heteroaryl-pyridines via Suzuki cross-coupling reactions , 2005 .
[4] M. Parmentier,et al. Pyridino-directed lithiation of anisylpyridines: new access to functional pyridylphenols , 2005 .
[5] A. Batsanov,et al. Palladium-catalyzed cross-coupling reactions of pyridylboronic acids with heteroaryl halides bearing a primary amine group: synthesis of highly substituted bipyridines and pyrazinopyridines. , 2005, The Journal of organic chemistry.
[6] S. Rault,et al. Efficient synthesis of halohydroxypyridines by hydroxydeboronation , 2005 .
[7] M. Dart,et al. Design of ligands for the nicotinic acetylcholine receptors: the quest for selectivity. , 2004, Current topics in medicinal chemistry.
[8] Jana Sopkova-de Oliveira Santos,et al. Synthesis of novel halopyridinylboronic acids and esters. Part 4: Halopyridin-2-yl-boronic acids and esters are stable, crystalline partners for classical Suzuki cross-coupling☆ , 2003 .
[9] S. Rault,et al. 2-bromo-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine, a new unexpected bifunctional building block for combinatorial chemistry. , 2003, Acta crystallographica. Section C, Crystal structure communications.
[10] M. Romanelli,et al. Cholinergic nicotinic receptors: Competitive ligands, allosteric modulators, and their potential applications , 2003, Medicinal research reviews.
[11] Y. Fort,et al. First regioselective ortho-lithiation induced by a 2-chloropyridyl group complexation. , 2003, The Journal of organic chemistry.
[12] S. Rault,et al. 2-(6-bromopyridin-3-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane and (6-bromopyridin-3-yl)boronic acid, new bifunctional building blocks for combinatorial chemistry. , 2003, Acta crystallographica. Section C, Crystal structure communications.
[13] S. Rault,et al. Synthesis of novel halopyridinylboronic acids and esters. Part 2: 2,4, or 5-Halopyridin-3-yl-boronic acids and esters , 2002 .
[14] C. B. Davis,et al. Synthesis and structure-activity relationship of novel pyridyl ethers for the nicotinic acetylcholine receptor. , 2000, Bioorganic & medicinal chemistry letters.
[15] Akira Suzuki,et al. Recent advances in the cross-coupling reactions of organoboron derivatives with organic electrophiles, 1995–1998 , 1999 .
[16] D. Donnelly-roberts,et al. ABT-594 [(R)-5-(2-azetidinylmethoxy)-2-chloropyridine]: a novel, orally effective analgesic acting via neuronal nicotinic acetylcholine receptors: I. In vitro characterization. , 1998, The Journal of pharmacology and experimental therapeutics.
[17] D. Donnelly-roberts,et al. Identification and initial structure-activity relationships of (R)-5-(2-azetidinylmethoxy)-2-chloropyridine (ABT-594), a potent, orally active, non-opiate analgesic agent acting via neuronal nicotinic acetylcholine receptors. , 1998, Journal of medicinal chemistry.
[18] Norio Miyaura,et al. Palladium-Catalyzed Cross-Coupling Reactions of Organoboron Compounds , 1995 .