One-pot synthesis of pyrido[2,3-d]pyrimidines via efficient three-component reaction in aqueous media
暂无分享,去创建一个
D. Shi | S. Ji | Xiang-Shan Wang | Jingwen Shi | L. Niu
[1] Q. Wang,et al. New potential inhibitors of cyclin-dependent kinase 4: design and synthesis of pyrido[2,3-d]pyrimidine derivatives under microwave irradiation. , 2006, Bioorganic & medicinal chemistry letters.
[2] D. Shi,et al. One-pot Synthesis of N-Hydroxylacridine Derivatives in Water , 2005 .
[3] D. Shi,et al. Three‐Component One‐Pot Synthesis of 1,4‐Dihydropyrano[2,3‐c]pyrazole Derivatives in Aqueous Media , 2004 .
[4] P. Bhuyan,et al. A novel three-component one-pot synthesis of pyrano[2,3-d]pyrimidines and pyrido[2,3-d]pyrimidines using microwave heating in the solid state , 2003 .
[5] C. Kappe,et al. High-throughput synthesis of N3-acylated dihydropyrimidines combining microwave-assisted synthesis and scavenging techniques. , 2003, Organic letters.
[6] U. Bora,et al. A novel microwave-mediated one-pot synthesis of indolizines via a three-component reaction. , 2003, Organic letters.
[7] J. Iqbal,et al. Cu(I)-catalyzed three component coupling protocol for the synthesis of quinoline derivatives , 2002 .
[8] T. Arrhenius,et al. A convenient solution and solid-phase synthesis of Δ5-2-oxopiperazines via N-acyliminium ions cyclization , 2002 .
[9] Yu Yuan,et al. Acid-free aza Diels-Alder reaction of Danishefsky's diene with imines. , 2002, Organic letters.
[10] R. Olsson,et al. A novel metal iodide promoted three-component synthesis of substituted pyrrolidines. , 2002, Organic letters.
[11] M. N. Nasr,et al. Pyrido [2, 3‐d]pyrimidines and Pyrimido[5′, 4′:5, 6]pyrido[2, 3‐d]pyrimidines as New Antiviral Agents: Synthesis and Biological Activity , 2002, Archiv der Pharmazie.
[12] J. Bower,et al. A new one-pot three-component condensation reaction for the synthesis of 2,3,4,6-tetrasubstituted pyridines. , 2002, Chemical communications.
[13] Dennis H. Evans,et al. One-step synthesis of substituted 6-amino-5-cyanospiro-4-(piperidine-4')- 2H,4H-dihydropyrazolo[3,4-b]pyrans. , 2002, Organic letters.
[14] B. List,et al. A Novel Proline‐Catalyzed Three‐Component Reaction of Ketones, Aldehydes, and Meldrum′s Acid. , 2001 .
[15] S. Carloni,et al. Clean synthesis in water. Part 2: Uncatalysed condensation reaction of Meldrum's acid and aldehydes , 2001 .
[16] V. Nair,et al. A novel synthesis of 2-aminopyrroles using a three-component reaction. , 2001, The Journal of organic chemistry.
[17] S. Queener,et al. Pneumocystis carinii and Toxoplasma gondii dihydrofolate reductase inhibitors and antitumor agents: synthesis and biological activities of 2,4-diamino-5-methyl-6-[(monosubstituted anilino)methyl] pyrido[2,3-d]pyrimidines. , 1999, Journal of medicinal chemistry.
[18] F. Bigi,et al. Montmorillonite KSF as an Inorganic, Water Stable, and Reusable Catalyst for the Knoevenagel Synthesis of Coumarin-3-carboxylic Acids. , 1999, The Journal of organic chemistry.
[19] J. S. Sandhu,et al. Studies on uracils: an efficient method for the synthesis of novel 1-allyl-6-(1′,2′,3′-triazolyl) analogues of HEPT , 1999 .
[20] A. Doherty,et al. Structure-activity relationships for a novel series of pyrido[2,3-d]pyrimidine tyrosine kinase inhibitors. , 1997, Journal of medicinal chemistry.
[21] R. Ballini,et al. CC bond fission via sulphones: A new ring cleavage of cyclic β-keto phenylsulphones , 1997 .
[22] R. Ballini,et al. The Michael reaction of nitroalkanes with conjugated enones in aqueous media , 1996 .
[23] A. Vasudevan,et al. 2,4-diamino-5-deaza-6-substituted pyrido[2,3-d]pyrimidine antifolates as potent and selective nonclassical inhibitors of dihydrofolate reductases. , 1996, Journal of medicinal chemistry.
[24] C. Monneret,et al. Synthesis of deoxy analogs of HEPT involving a palladium (0) catalyzed coupling , 1994 .
[25] Chao-Jun Li. Organic reactions in aqueous media - with a focus on carbon-carbon bond formation , 1993 .
[26] H. Mitsuya,et al. Molecular targets for AIDS therapy. , 1990, Science.
[27] J. S. Sandhu,et al. Studies on uracils. 10. A facile one-pot synthesis of pyrido[2,3-d]- and pyrazolo[3,4-d]pyrimidines , 1990 .
[28] J. S. Sandhu,et al. Studies of pyrimidine-2,4-diones: synthesis of novel condensed pyrido[2,3-d]pyrimidines via intramolecular cycloadditions , 1988 .
[29] J. S. Sandhu,et al. Studies on Pyrimidine-Annelated Heterocycles; 8.1 Intramolecular Cycloaddition of Thiophene and Nitrile Oxide or Nitrone Groups Bonded to 1,3-Dimethyluracils , 1988 .
[30] R. T. Walker,et al. Synthesis and antiviral properties of (E)-5-(2-bromovinyl)-2'-deoxycytidine-related compounds. , 1988, Journal of medicinal chemistry.
[31] E. De Clercq,et al. Specific phosphorylation of 5-ethyl-2'-deoxyuridine by herpes simplex virus-infected cells and incorporation into viral DNA. , 1987, The Journal of biological chemistry.
[32] E. De Clercq,et al. 2'-Fluorinated arabinonucleosides of 5-(2-haloalkyl)uracil: synthesis and antiviral activity. , 1987, Journal of medicinal chemistry.
[33] J Desmyter,et al. Both 2',3'-dideoxythymidine and its 2',3'-unsaturated derivative (2',3'-dideoxythymidinene) are potent and selective inhibitors of human immunodeficiency virus replication in vitro. , 1987, Biochemical and biophysical research communications.
[34] E. Clercq. Chemotherapeutic approaches to the treatment of the acquired immune deficiency syndrome (AIDS). , 1986 .
[35] J. Burchenal,et al. Synthesis and biological activities of 5-deaza analogues of aminopterin and folic acid. , 1986, Journal of Medicinal Chemistry.
[36] E. Declercq. Potential of bromovinyldeoxyuridine in anticancer chemotherapy. , 1986 .
[37] Y. Kitade,et al. Pyrimidines. 17. Novel pyrimidine to pyridine transformation reaction. One-step synthesis of pyrido[2,3-d]pyrimidines , 1981 .
[38] R. Breslow,et al. REVERSING THE SELECTIVITY OF CYCLODEXTRIN BISIMIDAZOLE RIBONUCLEASE MIMICS BY CHANGING THE CATALYST GEOMETRY , 1980 .
[39] Tadashi. Sasaki,et al. Search for a simpler synthetic model system for intramolecular 1,3-dipolar cycloaddition to the 5,6-double bond of a pyrimidine nucleoside , 1980 .
[40] F. Yoneda,et al. A NEW RING TRANSFORMATION OF ISOXAZOLO[3,4-d]PYRIMIDINES INTO PYRIMIDO[4,5-d]PYRIMIDINES , 1979 .
[41] R. T. Walker,et al. The synthesis of the potent anti-herpes virus agent, E-5(2-bromovinyl)-2′-deoxyuridine and related compounds , 1979 .
[42] 丸本 龍二,et al. Kondensierte Pyrimidine. III. Synthese von Isoxazolo [3,4-d] pyrimidinen , 1977 .
[43] T. Bradshaw,et al. 5-Substituted pyrimidine nucleosides and nucleotides , 1977 .
[44] G. Anderson,et al. Pyrido(2,3-d)pyrimidines. IV. Synthetic studies leading to various oxopyrido(2,3-d)pyrimidines. , 1976, The Journal of organic chemistry.
[45] A. D. Broom,et al. Studies on the acylation of some 6-aminouracil derivatives. , 1972, The Journal of organic chemistry.
[46] A. Strecker. Ueber die künstliche Bildung der Milchsäure und einen neuen, dem Glycocoll homologen Körper; , 1850 .