Structure-based design and pharmacokinetic optimization of covalent allosteric inhibitors of the mutant GTPase KRASG12C.
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Doyle J Cassar | J. Breed | D. Ogg | Lyman J. L. Feron | S. Lamont | Michael Tonge | A. Chakraborty | R. Carbajo | S. Cosulich | G. Robb | E. Gleave | C. Phillips | S. Bagal | I. Cumming | M. S. Bodnarchuk | P. Kemmitt | S. Ross | F. W. Goldberg | J. Kettle | S. Bickerton | M. Davies | A. Eatherton | L. Evans | Shaun M. Fillery | S. Harlfinger | Lyndsey L. Hanson | M. Howard | R. Howells | A. Jackson | J. Kingston | H. Lewis | Songlei Li | Libin Liu | R. Polanski | David M Robinson | James W. Smith | R. Whiteley | Junsheng Yang | Longfei Zhang | Xiliang Zhao | Frederick W. Goldberg | Christopher Phillips | Lyndsey Hanson | R. J. Carbajo | F. Goldberg | Emma S. Gleave | Scott G. Lamont | Junsheng Yang | Stephanie Harlfinger | S. Cosulich | M. Bodnarchuk | Sue Bickerton | Jason Breed | Atanu Chakraborty | Michael Davies | Laura Evans | Shaun Fillery | Martin Howard | Jennifer K. Kingston | Songlei Li | Derek Ogg | David M Robinson | Sarah J Ross | James Smith | Xiliang Zhao