Discovery and Structure–Activity Relationships of Pyrrolone Antimalarials
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Ian H. Gilbert | Marcel Kaiser | David M. Shackleford | Susan A. Charman | Michael Campbell | I. Gilbert | S. Charman | M. Kaiser | Julia Morizzi | Dinakaran Murugesan | Kasiram Katneni | A. Hudson | Clive Yeates | Alka Mital | Alan Hudson | Julia Morizzi | Michael Campbell | K. Katneni | C. Yeates | Dinakaran Murugesan | A. Mital
[1] S. Croft,et al. Artemisone--a highly active antimalarial drug of the artemisinin class. , 2006, Angewandte Chemie.
[2] T. Kappe,et al. Benzimidazole condensed ring systems.4. New approaches to the synthesis of substituted pyrimido[1,6-a]-benzimidazole-1,3(2H,5H)-diones , 1989 .
[3] Tim Morris,et al. Physiological Parameters in Laboratory Animals and Humans , 1993, Pharmaceutical Research.
[4] P. Olliaro,et al. The Global Portfolio of New Antimalarial Medicines Under Development , 2009, Clinical pharmacology and therapeutics.
[5] Chris J Janse,et al. A Plasmodium berghei reference line that constitutively expresses GFP at a high level throughout the complete life cycle. , 2004, Molecular and biochemical parasitology.
[6] C. Bevan,et al. A high-throughput screening method for the determination of aqueous drug solubility using laser nephelometry in microtiter plates. , 2000, Analytical chemistry.
[7] G. Allen,et al. Behavior of 2-halo- and 2-trifluoromethyl-1,4-benzoquinones in the Nenitzescu indole synthesis , 1968 .
[8] M. Petzold,et al. Novel Polymorphisms in Plasmodium falciparum ABC Transporter Genes Are Associated with Major ACT Antimalarial Drug Resistance , 2011, PLoS ONE.
[9] G. Beale,et al. Susceptibility of Plasmodium falciparum to five drugs: an in vitro study of isolates mainly from Thailand. , 1983, Transactions of the Royal Society of Tropical Medicine and Hygiene.
[10] J. Vorkapić-Furač,et al. Sterically hindered N-aryl pyrroles: chromatographic separation of enantiomers and barriers to racemization , 1989 .
[11] A. Cowman,et al. Chemotherapy and drug resistance in malaria. , 1990, International journal for parasitology.
[12] Adam R Renslo,et al. Drug discovery and development for neglected parasitic diseases , 2006, Nature chemical biology.
[13] D. B. Martins,et al. Reactivity of chloroacetylated β-enamino compounds. Synthesis of heterocycles , 2002 .
[14] J. Richard,et al. Plasmodium Falciparum Malaria Parasite Cultures and Their Use in Immunology , 1990 .
[15] T. Kappe,et al. Benzimidazole condensed ring systems. 5. Studies on the Synthesis of Pyrimido[1,6-α]benzimidazole-1,3(2H,5H)-diones† , 1989 .
[16] M. Abraham,et al. Fast gradient HPLC method to determine compounds binding to human serum albumin. Relationships with octanol/water and immobilized artificial membrane lipophilicity. , 2003, Journal of pharmaceutical sciences.
[17] R. Obach,et al. Prediction of human clearance of twenty-nine drugs from hepatic microsomal intrinsic clearance data: An examination of in vitro half-life approach and nonspecific binding to microsomes. , 1999, Drug metabolism and disposition: the biological fate of chemicals.
[18] J. Haynes,et al. Quantitative assessment of antimalarial activity in vitro by a semiautomated microdilution technique , 1979, Antimicrobial Agents and Chemotherapy.