论文信息 - Effective Synthesis of a Carbon-linked Diazirinyl Fatty Acid Derivative via Reduction of the Carbonyl Group to Methylene with Triethylsilane and Trifluoroacetic Acid

Effective Synthesis of a Carbon-linked Diazirinyl Fatty Acid Derivative via Reduction of the Carbonyl Group to Methylene with Triethylsilane and Trifluoroacetic Acid

Friedel-Crafts acylation of the aryldiazirine with ω-ester-α-acyl halide and successive reduction of the carbonyl group to methylene with triethylsilane and trifluoroacetic acid gave diazirinylated fatty acids.

M. Hashimoto | Y. Hatanaka | K. Nabeta

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