Discovery of 1-[2-(1-methyl-1H-pyrazol-5-yl)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]-3-(pyridin-4-ylmethyl)urea as a potent NAMPT (nicotinamide phosphoribosyltransferase) activator with attenuated CYP inhibition.
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E. Sergienko | M. Yokoyama | S. Gardell | Tsuyoshi Nakamura | A. Pinkerton | Ken Sakurai | T. Tsuji | Jun Tanaka | Daigo Asano | Y. Sogawa | K. Terayama | E. H. Sessions | Mayuko Akiu | Mika Yokoyama