An Efficient Biginelli One-Pot Synthesis of New Benzoxazole-Substituted Dihydropyrimidinones and Thiones Catalysed by Alumina-Supported Trifluoromethane Sulfonic Acid Under Solvent Free Conditions

[1]  B. Sain,et al.  Alumina supported MoO3: An efficient and reusable heterogeneous catalyst for synthesis of 3,4-dihydropyridine-2(1H)-ones under solvent free conditions , 2008 .

[2]  Murugulla Adharvana Chari,et al.  Silica gel / NaHSO4 : an efficient and recyclable heterogeneous catalyst for high yield synthesis of 1, 5-benzodiazepine derivatives under microwave irradiation , 2007 .

[3]  Rajive Gupta,et al.  Covalently anchored sulfonic acid onto silica as an efficient and recoverable interphase catalyst for the synthesis of 3,4-dihydropyrimidinones/thiones , 2007 .

[4]  J. Bazureau,et al.  A new approach to N-3 functionalized 3,4-dihydropyrimidine-2(1H)-ones with 1,2,4-oxadiazole group as amide isostere via ionic liquid-phase technology , 2007 .

[5]  Jian-Rong Jin,et al.  HBF4-catalyzed Biginelli reaction: One-pot synthesis of dihydropyrimidin-2(1H)-ones under solvent-free conditions , 2007 .

[6]  A. Shaabani,et al.  Tangstophosphoric acid (H3PW12O40): An efficient and eco-friendly catalyst for the one-pot synthesis of dihydropyrimidin-2(1H)-ones , 2006 .

[7]  K. Mukkanti,et al.  Silica gel/FeCl3: An efficient and recyclable heterogenous catalyst for one step synthesis of 4(3H)-quinazolinones under solvent free conditions , 2006 .

[8]  Murugulla Adharvana Chari,et al.  Silicagel supported sodium hydrogensulfate as a heterogenous catalyst for high yield synthesis of 3,4-dihydropyrimidin-2 (1H)-ones , 2004 .

[9]  T. Ramalingam,et al.  Microwave-Assisted Efficient synthesis of Dihydro Pyrimidines: Improved High Yielding Protocol for the Biginelli Reaction , 2000 .

[10]  I. Yalcin,et al.  Synthesis and antimicrobial activity of some novel 2,5- and/or 6-substituted benzoxazole and benzimidazole derivatives. , 1999, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

[11]  A. Shutalev,et al.  A New Convenient Synthesis of 5-Acyl-1,2,3,4-tetrahydropyrimidine-2-thiones/ones , 1998 .

[12]  G. Breton Selective Monoacetylation of Unsymmetrical Diols Catalyzed by Silica Gel-Supported Sodium Hydrogen Sulfate , 1997 .

[13]  S. I. Hommeltoft,et al.  Role of Ester Intermediates in Isobutane Alkylation and Its Consequence for the Choice of Catalyst System , 1997 .

[14]  C. Kappe,et al.  Conformational analysis of 4-aryl-dihydropyrimidine calcium channel modulators. A comparison of ab initio, semiempirical and X-ray crystallographic studies , 1997 .

[15]  Jinsheng Chen,et al.  Synthesis of the tricyclic portions of batzelladines A, B and D. Revision of the stereochemistry of batzelladines A and D , 1996 .

[16]  P. Wipf,et al.  A SOLID PHASE PROTOCOL OF THE BIGINELLI DIHYDROPYRIMIDINE SYNTHESIS SUITABLE FOR COMBINATORIAL CHEMISTRY , 1995 .

[17]  M. F. Bean,et al.  Novel Alkaloids from the Sponge Batzella sp.: Inhibitors of HIV gp120-Human CD4 Binding , 1995 .

[18]  C. Kappe 100 years of the biginelli dihydropyrimidine synthesis , 1993 .

[19]  B. Snider,et al.  Biomimetic synthesis of (.+-.)-crambines A, B, C1, and C2. Revision of the structure of crambines B and C1 , 1993 .

[20]  S. Moreland,et al.  Dihydropyrimidine calcium channel blockers. 4. Basic 3-substituted-4-aryl-1,4-dihydropyrimidine-5-carboxylic acid esters. Potent antihypertensive agents. , 1992, Journal of medicinal chemistry.

[21]  A Hedberg,et al.  Dihydropyrimidine calcium channel blockers. 3. 3-Carbamoyl-4-aryl-1,2,3,4-tetrahydro-6-methyl-5-pyrimidinecarboxylic acid esters as orally effective antihypertensive agents. , 1991, Journal of medicinal chemistry.

[22]  G. Rovnyak,et al.  Substituted 1,4-dihydropyrimidines. 3. Synthesis of selectively functionalized 2-hetero-1,4-dihydropyrimidines , 1989 .

[23]  T. Nishiguchi,et al.  Dehydration of alcohols catalysed by metallic sulphates supported on silica gel , 1989 .

[24]  K. Atwal,et al.  Synthesis of substituted 1,2,3,4-tetrahydro-6-methyl-2-oxo-5-pyrimidinecarboxylic acid esters: the Biginelli condensation revisited , 1987 .

[25]  M. Malley,et al.  Synthesis of substituted 1,2,3,4-tetrahydro-6-methyl-2-thioxo-5-pyrimidinecarboxylic acid esters , 1987 .

[26]  O. Cox,et al.  Synthesis and biological activity of benzothiazolo- and benzoxazolo[3,2-a]quinolinium salts. , 1982, Journal of medicinal chemistry.

[27]  K. Folkers,et al.  Hydrogenation of Cyclic Ureides under Elevated Temperatures and Pressures. I.1 2-Keto-1,2,3,4-tetrahydropyrimidines , 1934 .

[28]  H. Harwood,et al.  RESEARCHES ON PYRIMIDINES. CXXX. SYNTHESIS OF 2-KETO-1,2,3,4-TETRAHYDROPYRIMIDINES , 1932 .