Discovery, structure-activity relationships, pharmacokinetics, and efficacy of glucokinase activator (2R)-3-cyclopentyl-2-(4-methanesulfonylphenyl)-N-thiazol-2-yl-propionamide (RO0281675).
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A. Railkar | J. Grippo | F. Matschinsky | P. Mahaney | J. Grimsby | L. Qi | R. Kester | J. Tengi | R. Sarabu | G. Holland | K. Guertin | W. L. Corbett | M. Dvorozniak | N. Haynes | F. T. Bizzarro | Darryl W Hilliard | Cheryl L Spence | F. Bizzarro