Synthesis and selective cytotoxic activity of novel hybrid chalcones against prostate cancer cells.
暂无分享,去创建一个
S. Ramakrishna | R. Chandra | V. Lakshma Nayak | B. B. Gawali | M. Vishnuvardhan | C. Ashwini | M. Nagaraju | E. Gnana Deepthi
[1] V. Khedkar,et al. Synthesis, antitubercular evaluation and 3D-QSAR study of N-phenyl-3-(4-fluorophenyl)-4-substituted pyrazole derivatives. , 2012, Bioorganic & medicinal chemistry letters.
[2] N. Sahu,et al. Exploring pharmacological significance of chalcone scaffold: a review. , 2012, Current medicinal chemistry.
[3] Keduo Qian,et al. Structure-activity relationships of chalcone analogs as potential inhibitors of ADP- and collagen-induced platelet aggregation. , 2011, Bioorganic & medicinal chemistry.
[4] Lorenzo Caggiano,et al. Design, synthesis and antiproliferative activity of urocanic-chalcone hybrid derivatives , 2011 .
[5] Y. Na,et al. Chalcones as Novel Non-peptidic μ-Calpain Inhibitors , 2011 .
[6] Young Min Kim,et al. Characteristic of alkylated chalcones from Angelica keiskei on influenza virus neuraminidase inhibition. , 2011, Bioorganic & medicinal chemistry letters.
[7] W. Maltese,et al. A chalcone-related small molecule that induces methuosis, a novel form of non-apoptotic cell death, in glioblastoma cells , 2011, Molecular Cancer.
[8] Y. Asiri,et al. Design, synthesis, and biological evaluation of substituted hydrazone and pyrazole derivatives as selective COX-2 inhibitors: Molecular docking study. , 2011, Bioorganic & medicinal chemistry.
[9] Xue-Quan Wang,et al. Design, synthesis and cytotoxic activities of novel hybrid compounds between dihydrobenzofuran and imidazole. , 2011, Organic and biomolecular chemistry.
[10] P. Paré,et al. Estrogenic activity of chemical constituents from Tephrosia candida. , 2011, Journal of natural products.
[11] S. Riyadh. Enaminones as Building Blocks for the Synthesis of Substituted Pyrazoles with Antitumor and Antimicrobial Activities , 2011, Molecules.
[12] R. Roden,et al. α,β-Unsaturated carbonyl system of chalcone-based derivatives is responsible for broad inhibition of proteasomal activity and preferential killing of human papilloma virus (HPV) positive cervical cancer cells. , 2011, Journal of medicinal chemistry.
[13] W. Oh,et al. Chalcones as novel influenza A (H1N1) neuraminidase inhibitors from Glycyrrhiza inflata. , 2011, Bioorganic & medicinal chemistry letters.
[14] N. Suh,et al. Synthesis and biological evaluation of retinoid-chalcones as inhibitors of colon cancer cell growth. , 2010, Bioorganic & medicinal chemistry letters.
[15] S. Dulchavsky,et al. Growth inhibitory and apoptosis-inducing effects of xanthohumol, a prenylated chalone present in hops, in human prostate cancer cells. , 2010, Anticancer research.
[16] P. Reddanna,et al. Design, synthesis, and biological evaluation of prenylated chalcones as 5-LOX inhibitors. , 2010, Bioorganic & medicinal chemistry.
[17] R. F. Hartman,et al. Cell Cycle Arrest and Apoptosis Induction by an Anticancer Chalcone Epoxide , 2010, Archiv der Pharmazie.
[18] B. Insuasty,et al. Synthesis of novel pyrazolic analogues of chalcones and their 3-aryl-4-(3-aryl-4,5-dihydro-1H-pyrazol-5-yl)-1-phenyl-1H-pyrazole derivatives as potential antitumor agents. , 2010, Bioorganic & medicinal chemistry.
[19] Peng-Cheng Lv,et al. Synthesis and biological evaluation of pyrazole derivatives containing thiourea skeleton as anticancer agents. , 2010, Bioorganic & medicinal chemistry.
[20] J. Heilmann,et al. Synthesis, cytotoxicity, anti-oxidative and anti-inflammatory activity of chalcones and influence of A-ring modifications on the pharmacological effect. , 2010, European journal of medicinal chemistry.
[21] So Ha Lee,et al. Design and synthesis of new potent anticancer pyrazoles with high FLT3 kinase inhibitory selectivity. , 2010, Bioorganic & medicinal chemistry.
[22] C. Khobragade,et al. Synthesis and biological evaluation of a novel series of pyrazole chalcones as anti-inflammatory, antioxidant and antimicrobial agents. , 2009, Bioorganic & medicinal chemistry.
[23] Y. Tzeng,et al. Synthesis and biological evaluation of 3',4',5'-trimethoxychalcone analogues as inhibitors of nitric oxide production and tumor cell proliferation. , 2009, Bioorganic & medicinal chemistry.
[24] B. Srinivasan,et al. Structure-activity relationship studies of chalcone leading to 3-hydroxy-4,3',4',5'-tetramethoxychalcone and its analogues as potent nuclear factor kappaB inhibitors and their anticancer activities. , 2009, Journal of medicinal chemistry.
[25] F. Souard,et al. A novel chalcone derivative which acts as a microtubule depolymerising agent and an inhibitor of P-gp and BCRP in in-vitro and in-vivo glioblastoma models , 2009, BMC Cancer.
[26] D. Hadjipavlou-Litina,et al. Chalcones in cancer: understanding their role in terms of QSAR. , 2009, Current medicinal chemistry.
[27] Shinji Ohta,et al. C-geranylated chalcones from the stems of Angelica keiskei with superoxide-scavenging activity. , 2008, Journal of natural products.
[28] B. Wasylyk,et al. Inhibition of the Ras-Net (Elk-3) pathway by a novel pyrazole that affects microtubules. , 2008, Cancer research.
[29] J. Gut,et al. Antimalarial prenylated chalcones from the twigs of Dorstenia barteri var. subtriangularis , 2007 .
[30] G. Pauli,et al. The pharmacognosy of Humulus lupulus L. (hops) with an emphasis on estrogenic properties. , 2006, Phytomedicine : international journal of phytotherapy and phytopharmacology.
[31] B. Ngadjui,et al. Antitrichomonal and antioxidant activities of Dorstenia barteri and Dorstenia convexa. , 2005, Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas.
[32] X. Wu,et al. Chalcones: an update on cytotoxic and chemoprotective properties. , 2005, Current medicinal chemistry.
[33] G. Folefoc,et al. Diprenylated chalcones and other constituents from the twigs of Dorstenia barteri var. subtriangularis. , 2004, Phytochemistry.
[34] F. Gozzo,et al. Regioselectivity in aromatic Claisen rearrangements. , 2003, The Journal of organic chemistry.
[35] R. Tapia,et al. Synthesis and antiprotozoal activity of naphthofuranquinones and naphthothiophenequinones containing a fused thiazole ring. , 2003, Bioorganic & medicinal chemistry.
[36] F. Belluti,et al. Synthesis and antitumor activity of new derivatives of xanthen-9-one-4-acetic acid. , 2002, Journal of medicinal chemistry.
[37] C. Di Giorgio,et al. 1,3-Diphenylpyrazoles: synthesis and antiparasitic activities of azomethine derivatives. , 2002, European journal of medicinal chemistry.
[38] J. Roseiro,et al. Flavonoids from Ulex airensis and Ulex europaeus ssp. europaeus. , 2002, Journal of natural products.
[39] S. Kouam,et al. Prenylated flavonoids from the aerial parts of Dorstenia mannii. , 2000, Phytochemistry.
[40] W. Ryan,et al. Automated parallel synthesis of chalcone-based screening libraries , 1998 .
[41] T. Maduskuie,et al. Hydroxyacetophenone-derived antagonists of the peptidoleukotrienes. , 1989, Journal of Medicinal Chemistry.
[42] T. Mosmann. Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays. , 1983, Journal of immunological methods.