NS-49, a novel α1a-adrenoceptor-selective agonist characterization using recombinant human α1-adrenoceptors

[1]  R. Graham,et al.  alpha 1-adrenergic receptor subtypes. Molecular structure, function, and signaling. , 1996, Circulation research.

[2]  G. Tsujimoto,et al.  Selectivity of the imidazoline α‐adrenoceptor agonists (oxymetazoline and cirazoline) for human cloned α1‐adrenoceptor subtypes , 1995 .

[3]  R. Graham,et al.  Cloning, expression, and tissue distribution of the rat homolog of the bovine alpha 1C-adrenergic receptor provide evidence for its classification as the alpha 1A subtype. , 1994, Molecular pharmacology.

[4]  K. Minneman,et al.  Selectivity of agonists for cloned alpha 1-adrenergic receptor subtypes. , 1994, Molecular pharmacology.

[5]  T. Branchek,et al.  The rat homologue of the bovine alpha 1c-adrenergic receptor shows the pharmacological properties of the classical alpha 1A subtype. , 1994, Molecular pharmacology.

[6]  G. Tsujimoto,et al.  The pharmacological profile of cloned and stably expressed α1B-adrenoceptor in CHO cells , 1994 .

[7]  T. Branchek,et al.  The alpha 1-adrenergic receptor that mediates smooth muscle contraction in human prostate has the pharmacological properties of the cloned human alpha 1c subtype. , 1994, Molecular pharmacology.

[8]  K. Minneman,et al.  Alpha 1-adrenergic receptor subtypes. , 1994, Annual review of pharmacology and toxicology.

[9]  G. Tsujimoto,et al.  Cloning, functional expression and tissue distribution of human cDNA for the alpha 1C-adrenergic receptor. , 1993, Biochemical and biophysical research communications.

[10]  J. Lomasney,et al.  Pharmacologic characterization of cloned alpha 1-adrenoceptor subtypes: selective antagonists suggest the existence of a fourth subtype. , 1992, European journal of pharmacology.

[11]  R. Graham,et al.  Solution-phase library screening for the identification of rare clones: isolation of an alpha 1D-adrenergic receptor cDNA. , 1991, Molecular pharmacology.

[12]  M. Caron,et al.  Molecular cloning and expression of the cDNA for the alpha 1A-adrenergic receptor. The gene for which is located on human chromosome 5. , 1991, The Journal of biological chemistry.

[13]  G. Tsujimoto,et al.  Two pharmacologically distinct alpha 1-adrenoceptor subtypes in the contraction of rabbit aorta: each subtype couples with a different Ca2+ signalling mechanism and plays a different physiological role. , 1990, Molecular pharmacology.

[14]  M. Caron,et al.  Molecular cloning and expression of the cDNA for a novel alpha 1-adrenergic receptor subtype. , 1990, The Journal of biological chemistry.

[15]  G. Tsujimoto,et al.  Characterization of α1-adrenergic receptor subtypes linked to iodide efflux in rat FRTL cells , 1990 .

[16]  G. Tsujimoto,et al.  Glycogen phosphorylase activation by two different alpha 1-adrenergic receptor subtypes: methoxamine selectively stimulates a putative alpha 1-adrenergic receptor subtype (alpha 1a) that couples with Ca2+ influx. , 1989, Molecular pharmacology.

[17]  M. Caron,et al.  Molecular cloning and expression of the cDNA for the hamster alpha 1-adrenergic receptor. , 1988, Proceedings of the National Academy of Sciences of the United States of America.

[18]  M. Endoh,et al.  Further characterization of the myocardial alpha-adrenoceptors mediating positive inotropic effects in the rabbit myocardium. , 1988, European journal of pharmacology.

[19]  K. Minneman Alpha 1-adrenergic receptor subtypes, inositol phosphates, and sources of cell Ca2+. , 1988, Pharmacological reviews.

[20]  P. Abel,et al.  Heterogeneity of alpha 1-adrenergic receptors revealed by chlorethylclonidine. , 1987, Molecular pharmacology.

[21]  P. Insel,et al.  Alpha 1-adrenergic receptor-linked guanine nucleotide-binding protein in muscle and kidney epithelial cells. , 1987, Molecular pharmacology.

[22]  P. Abel,et al.  α1Adrenoceptor subtypes linked to different mechanisms for increasing intracellular Ca2+ in smooth muscle , 1987, Nature.

[23]  P. Abel,et al.  Alpha-1 adrenergic receptor binding and contraction of rat caudal artery. , 1986, The Journal of pharmacology and experimental therapeutics.

[24]  K. Honda,et al.  Alpha-1 adrenoceptor antagonist effects of the optical isomers of YM-12617 in rabbit lower urinary tract and prostate. , 1986, The Journal of pharmacology and experimental therapeutics.

[25]  I. Creese,et al.  Characterization of alpha 1-adrenergic receptor subtypes in rat brain: a reevaluation of [3H]WB4104 and [3H]prazosin binding. , 1986, Molecular pharmacology.

[26]  R. Tsien,et al.  A new generation of Ca2+ indicators with greatly improved fluorescence properties. , 1985, The Journal of biological chemistry.

[27]  R. Ruffolo IMPORTANT CONCEPTS OF RECEPTOR THEORY , 1982 .

[28]  D Rodbard,et al.  Ligand: a versatile computerized approach for characterization of ligand-binding systems. , 1980, Analytical biochemistry.