Synthesis and anti-Trypanosoma cruzi activity of new 3-phenylthio-nor-β-lapachone derivatives.
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J. Cavaleiro | V. Ferreira | F. D. da Silva | A. C. Bombaça | K. Salomão | S. D. de Castro | D. D. da Rocha | M. Cardoso
[1] J. Urbina. Recent Clinical Trials for the Etiological Treatment of Chronic Chagas Disease: Advances, Challenges and Perspectives , 2015, The Journal of eukaryotic microbiology.
[2] F. C. D. Silva,et al. Synthesis of fused chromene-1,4-naphthoquinones via ring-closing metathesis and Knoevenagel-electrocyclization under acid catalysis and microwave irradiation , 2014 .
[3] V. Ferreira,et al. Synthesis and anti-Trypanosoma cruzi activity of naphthoquinone-containing triazoles: electrochemical studies on the effects of the quinoidal moiety. , 2013, Bioorganic & medicinal chemistry.
[4] M. Lamberti,et al. Synergistic enhancement of antitumor effect of β-Lapachone by photodynamic induction of quinone oxidoreductase (NQO1). , 2013, Phytomedicine : international journal of phytotherapy and phytopharmacology.
[5] Melissa C. Srougi,et al. Catalase Abrogates β-Lapachone–Induced PARP1 Hyperactivation–Directed Programmed Necrosis in NQO1-Positive Breast Cancers , 2013, Molecular Cancer Therapeutics.
[6] M. Neves,et al. Gas phase reactions of ß-substituted hetero-Diels–Alder adducts of meso-tetraphenylporphyrin using tandem mass spectrometry , 2013 .
[7] F. Frézard,et al. Potent naphthoquinones against antimony-sensitive and -resistant Leishmania parasites: synthesis of novel α- and nor-α-lapachone-based 1,2,3-triazoles by copper-catalyzed azide-alkyne cycloaddition. , 2013, European journal of medicinal chemistry.
[8] V. Ferreira,et al. Novel 1H-1,2,3-, 2H-1,2,3-, 1H-1,2,4- and 4H-1,2,4-triazole derivatives: a patent review (2008 – 2011) , 2013, Expert opinion on therapeutic patents.
[9] P. Gaur,et al. Addition of thiols to o-quinone methide: new 2-hydroxy-3-phenylsulfanylmethyl[1,4]naphthoquinones and their activity against the human malaria parasite Plasmodium falciparum (3D7). , 2013, European journal of medicinal chemistry.
[10] L. V. Lotufo,et al. A new approach for the synthesis of 3-substituted cytotoxic nor-β-lapachones , 2013 .
[11] A. S. de Araujo,et al. On the search for potential anti-Trypanosoma cruzi drugs: synthesis and biological evaluation of 2-hydroxy-3-methylamino and 1,2,3-triazolic naphthoquinoidal compounds obtained by click chemistry reactions. , 2012, European journal of medicinal chemistry.
[12] A. Rassi,et al. American Trypanosomiasis (Chagas Disease). , 2019, Infectious disease clinics of North America.
[13] D. Ross,et al. NAD(P)H:quinone oxidoreductase 1 (NQO1) in the sensitivity and resistance to antitumor quinones. , 2012, Biochemical pharmacology.
[14] A. Cho,et al. The chemical biology of naphthoquinones and its environmental implications. , 2012, Annual review of pharmacology and toxicology.
[15] V. Pore,et al. Click chemistry: 1,2,3-triazoles as pharmacophores. , 2011, Chemistry, an Asian journal.
[16] F. C. D. Silva,et al. Synthesis of New o-Quinone Methides from β-LapachoneAnalogues , 2011 .
[17] Â. Pinto,et al. Synthesis and anti-Trypanosoma cruzi activity of β-lapachone analogues. , 2011, European journal of medicinal chemistry.
[18] M. N. Soeiro,et al. Screening of Potential anti-Trypanosoma cruzi Candidates: In Vitro and In Vivo Studies , 2011, The open medicinal chemistry journal.
[19] V. Ferreira,et al. Strategies for the synthesis of bioactive pyran naphthoquinones. , 2010, Organic & biomolecular chemistry.
[20] C. Bern,et al. Chagas disease in Spain, the United States and other non-endemic countries. , 2010, Acta tropica.
[21] Z. Yadón,et al. Chagas disease: a Latin American health problem becoming a world health problem. , 2010, Acta tropica.
[22] C. Kaiser,et al. Synthesis, biological activity, and molecular modeling studies of 1H-1,2,3-triazole derivatives of carbohydrates as alpha-glucosidases inhibitors. , 2010, Journal of medicinal chemistry.
[23] Â. Pinto,et al. Synthesis of α‐ and β‐Pyran Naphthoquinones as a New Class of Antitubercular Agents , 2010, Archiv der Pharmazie.
[24] V. Ferreira,et al. ß-Lapachone: Medicinal chemistry significance and structural modifications , 2010 .
[25] M. D. Vargas,et al. Theoretical studies of the tautomerism in 3-(2-R-Phenylhydrazono)-naphthalene- 1,2,4-triones: synthesis of copper(II) complexes and studies of antibacterial and antitumor activities , 2010 .
[26] Solange Lisboa de Castro,et al. The Trypanocidal Activity of Naphthoquinones: A Review , 2009, Molecules.
[27] M. Heinrich,et al. Red Lapacho (Tabebuia impetiginosa)--a global ethnopharmacological commodity? , 2009, Journal of ethnopharmacology.
[28] C. Kaiser,et al. Synthesis of α- and β-lapachone derivatives from hetero diels-alder trapping of alkyl and aryl o-quinone methides , 2009 .
[29] V. Ferreira,et al. Cytotoxic, Trypanocidal Activities and Physicochemical Parameters of nor-β-Lapachone-based 1,2,3-Triazoles , 2009 .
[30] V. Ferreira,et al. Naphthoquinoidal [1,2,3]-triazole, a new structural moiety active against Trypanosoma cruzi. , 2008, European journal of medicinal chemistry.
[31] C. K. Andrade,et al. Synthesis and anti-Trypanosoma cruzi activity of derivatives from nor-lapachones and lapachones. , 2008, Bioorganic & medicinal chemistry.
[32] D. V. Berdyshev,et al. Chemistry of naphthazarin derivatives 13. Conformational analysis of 3-(alk-1-enyl)-2-hydroxy-1,4-naphthoquinones by quantum chemistry methods , 2006 .
[33] D. Boothman,et al. New tricks for old drugs: the anticarcinogenic potential of DNA repair inhibitors , 2006, Journal of Molecular Histology.
[34] F. Emery,et al. Studies on the trypanocidal activity of semi-synthetic pyran[b-4,3]naphtho[1,2-d]imidazoles from beta-lapachone. , 2004, European journal of medicinal chemistry.
[35] R. Munday. Activation and detoxification of naphthoquinones by NAD(P)H: quinone oxidoreductase. , 2004, Methods in enzymology.
[36] W. de Souza,et al. Interaction of Trypanosoma cruzi with heart muscle cells: ultrastructural and cytochemical analysis of endocytic vacuole formation and effect upon myogenesis in vitro. , 1986, European journal of cell biology.