Contemporary strategies for peptide macrocyclization.
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[1] A. Wheeler,et al. Synchronized synthesis of peptide-based macrocycles by digital microfluidics. , 2010, Angewandte Chemie.
[2] David J Craik,et al. Native chemical ligation applied to the synthesis and bioengineering of circular peptides and proteins. , 2010, Biopolymers.
[3] Jörg Rademann,et al. Cyclative cleavage through dipolar cycloaddition: polymer-bound azidopeptidylphosphoranes deliver locked cis-triazolylcyclopeptides as privileged protein binders. , 2010, Angewandte Chemie.
[4] K. Jolliffe,et al. Synthesis of all-L cyclic tetrapeptides using pseudoprolines as removable turn inducers. , 2010, Organic letters.
[5] D. Crich,et al. Cyclic peptide synthesis with thioacids. , 2010, Organic letters.
[6] K. Anseth,et al. On-resin peptide macrocyclization using thiol-ene click chemistry. , 2010, Chemical communications.
[7] R. Houghten,et al. Macrolactonization of peptide thioesters catalyzed by imidazole and its application in the synthesis of kahalalide B and analogues. , 2010, Organic letters.
[8] S. Danishefsky,et al. Total synthesis of cyclosporine: access to N-methylated peptides via isonitrile coupling reactions. , 2010, Journal of the American Chemical Society.
[9] Vishal Rai,et al. Macrocyclization of linear peptides enabled by amphoteric molecules. , 2010, Journal of the American Chemical Society.
[10] Jeremy C. Smith,et al. Hydrogen-Bond Driven Loop-Closure Kinetics in Unfolded Polypeptide Chains , 2010, PLoS Comput. Biol..
[11] M. Fujita,et al. Conformational preferences of short peptide fragments. , 2009, Angewandte Chemie.
[12] Austin B. Yongye,et al. Synthesis of cyclic peptides through direct aminolysis of peptide thioesters catalyzed by imidazole in aqueous organic solutions. , 2009, Journal of combinatorial chemistry.
[13] Austin B. Yongye,et al. Modeling of peptides containing D-amino acids: implications on cyclization , 2009, J. Comput. Aided Mol. Des..
[14] M Reza Ghadiri,et al. Probing the bioactive conformation of an archetypal natural product HDAC inhibitor with conformationally homogeneous triazole-modified cyclic tetrapeptides. , 2009, Angewandte Chemie.
[15] John M. Beierle,et al. Conformationally homogeneous heterocyclic pseudotetrapeptides as three-dimensional scaffolds for rational drug design: receptor-selective somatostatin analogues. , 2009, Angewandte Chemie.
[16] Jomana Elaridi,et al. Metathesis assisted synthesis of cyclic peptides. , 2009, Chemical communications.
[17] A. Fournier,et al. Applications of BOP reagent in solid phase synthesis. II: Solid phase side-chain to side-chain cyclizations using BOP reagent , 2009 .
[18] U. Schmidt,et al. Cyclotetrapeptides and cyclopentapeptides: occurrence and synthesis. , 2009, The journal of peptide research : official journal of the American Peptide Society.
[19] R. Sheppard,et al. Some 'difficult sequences' made easy. A study of interchain association in solid-phase peptide synthesis. , 2009, International journal of peptide and protein research.
[20] H. Kessler,et al. Cyclic hexapeptides derived from the human thymopoietin III. , 2009, International journal of peptide and protein research.
[21] K. Fan,et al. Cyclization of several linear penta- and heptapeptides with different metal ions studied by CD spectroscopy. , 2008, The journal of peptide research : official journal of the American Peptide Society.
[22] David R. Liu,et al. Translation of DNA into a library of 13,000 synthetic small-molecule macrocycles suitable for in vitro selection. , 2008, Journal of the American Chemical Society.
[23] D. Tai,et al. Molecularly imprinted cavities template the macrocyclization of tetrapeptides. , 2008, Chemical communications.
[24] P. Roller,et al. Recent Progress of Synthetic Studies to Peptide and Peptidomimetic Cyclization , 2008 .
[25] Daniel Fortin,et al. Efficient parallel synthesis of macrocyclic peptidomimetics. , 2008, Bioorganic & medicinal chemistry letters.
[26] Jean Martínez,et al. Synthesis of cyclic peptides via O–N-acyl migration , 2008 .
[27] C. Hackenberger,et al. Chemoselective peptide cyclization by traceless Staudinger ligation. , 2008, Angewandte Chemie.
[28] Stephen P. Hale,et al. The exploration of macrocycles for drug discovery — an underexploited structural class , 2008, Nature Reviews Drug Discovery.
[29] Douglas A. Horton,et al. Cyclic tetrapeptides via the ring contraction strategy: chemical techniques useful for their identification. , 2008, Organic & biomolecular chemistry.
[30] H. Kessler,et al. Conformational preference and potential templates of N-methylated cyclic pentaalanine peptides. , 2008, Chemistry.
[31] Michael G Thomas,et al. Nonribosomal peptide synthetases involved in the production of medically relevant natural products. , 2008, Molecular pharmaceutics.
[32] H. Murakami,et al. Reprogramming the translation initiation for the synthesis of physiologically stable cyclic peptides. , 2008, ACS chemical biology.
[33] C. K. Andrade,et al. Design and synthesis of cyclic RGD pentapeptoids by consecutive Ugi reactions. , 2008, Organic letters.
[34] R. Raines,et al. Protein prosthesis: 1,5-disubstituted[1,2,3]triazoles as cis-peptide bond surrogates. , 2007, Journal of the American Chemical Society.
[35] R. Lokey,et al. Click chemistry as a macrocyclization tool in the solid-phase synthesis of small cyclic peptides. , 2007, Organic letters.
[36] D. Speijer,et al. 1,2,3-Triazoles as peptide bond isosteres: synthesis and biological evaluation of cyclotetrapeptide mimics. , 2007, Organic & biomolecular chemistry.
[37] Theodore V. Tselios,et al. Cyclic Peptides in Disease , 2007 .
[38] H. Kessler,et al. N-methylated cyclic pentaalanine peptides as template structures. , 2006, Journal of the American Chemical Society.
[39] S. Joo,et al. High-throughput sequence determination of cyclic peptide library members by partial Edman degradation/mass spectrometry. , 2006, Journal of the American Chemical Society.
[40] Vasso Apostolopoulos,et al. Round and round we go: cyclic peptides in disease. , 2006, Current medicinal chemistry.
[41] Kang Chen,et al. Evaluation of biologically relevant short alpha-helices stabilized by a main-chain hydrogen-bond surrogate. , 2006, Journal of the American Chemical Society.
[42] Ian D. Williams,et al. Ruthenium-catalyzed cycloaddition of alkynes and organic azides. , 2006, Journal of the American Chemical Society.
[43] J. Reek,et al. Carbosilane dendrimeric carbodiimides: site isolation as a lactamization tool. , 2006, The Journal of organic chemistry.
[44] J. V. van Maarseveen,et al. Click chemistry as a route to cyclic tetrapeptide analogues: synthesis of cyclo-[Pro-Val-psi(triazole)-Pro-Tyr]. , 2006, Organic letters.
[45] J. Campagne,et al. Macrolactonizations in the total synthesis of natural products. , 2006, Chemical reviews.
[46] C. Montalbetti,et al. Amide bond formation and peptide coupling , 2005 .
[47] M. Ghadiri,et al. Efficient route to C2 symmetric heterocyclic backbone modified cyclic peptides. , 2005, Organic letters.
[48] Jieping Zhu,et al. Conformation-directed macrocyclization reactions , 2005 .
[49] M. Finn,et al. Head-to-tail peptide cyclodimerization by copper-catalyzed azide-alkyne cycloaddition. , 2005, Angewandte Chemie.
[50] D. Fairlie,et al. Proteases universally recognize beta strands in their active sites. , 2005, Chemical reviews.
[51] Nishanth Marthandan,et al. Photolithographic synthesis of cyclic peptide arrays using a differential deprotection strategy. , 2005, Chemical communications.
[52] K. Jolliffe,et al. Pseudoprolines as removable turn inducers: tools for the cyclization of small peptides. , 2004, The Journal of organic chemistry.
[53] Paramjit S. Arora,et al. A highly stable short α-helix constrained by a main-chain hydrogen-bond surrogate , 2004 .
[54] S. Korsmeyer,et al. Activation of Apoptosis in Vivo by a Hydrocarbon-Stapled BH3 Helix , 2004, Science.
[55] N. Sewald,et al. An improved method for the solution cyclization of peptides under pseudo-high dilution conditions. , 2004, Journal of biotechnology.
[56] Judit Tulla-Puche,et al. On-resin native chemical ligation for cyclic peptide synthesis. , 2004, The Journal of organic chemistry.
[57] M. Chelli,et al. On‐resin head‐to‐tail cyclization of cyclotetrapeptides: optimization of crucial parameters , 2004, Journal of peptide science : an official publication of the European Peptide Society.
[58] G. Tian,et al. Studies on the Synthetic Methodology of Head to Tail Cyclization of Linear Peptides , 2003, Letters in Peptide Science.
[59] Y. Ye,et al. Studies on the synthetic methodology of head to tail cyclization of linear peptides , 2003, Letters in Peptide Science.
[60] J. Davies. The cyclization of peptides and depsipeptides , 2003, Journal of peptide science : an official publication of the European Peptide Society.
[61] M Reza Ghadiri,et al. A heterocyclic peptide nanotube. , 2003, Journal of the American Chemical Society.
[62] Douglas A. Horton,et al. Difficult macrocyclizations: new strategies for synthesizing highly strained cyclic tetrapeptides. , 2003, Organic letters.
[63] H. Schoemaker,et al. A pincer auxiliary to force difficult lactamisations. , 2003, Organic & biomolecular chemistry.
[64] U. Kazmaier,et al. Via Ugi reactions to conformationally fixed cyclic peptides. , 2003, Chemical communications.
[65] C. Schmuck,et al. Highly stable self-assembly in water: ion pair driven dimerization of a guanidiniocarbonyl pyrrole carboxylate zwitterion. , 2003, Journal of the American Chemical Society.
[66] Lu Th,et al. A New Tri-Orthogonal Strategy for Peptide Cyclization , 2002 .
[67] Michael D. Burkart,et al. Biomimetic synthesis and optimization of cyclic peptide antibiotics , 2002, Nature.
[68] Luke G Green,et al. A stepwise huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes. , 2002, Angewandte Chemie.
[69] N. Sewald,et al. Peptides: Chemistry and Biology , 2002 .
[70] Morten Meldal,et al. Peptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(i)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides. , 2002, The Journal of organic chemistry.
[71] J. Taunton,et al. Kinetic control of proline amide rotamers: total synthesis of trans,trans- and cis,cis-ceratospongamide. , 2002, Journal of the American Chemical Society.
[72] P. Dawson,et al. Design and Synthesis of a Protein Catenane , 2001 .
[73] P. Dawson,et al. Design and Synthesis of a Protein Catenane This work was supported by The Skaggs Institute for Chemical Biology, The Sloan Foundation, and NIH-GM570132 (PED). We thank Dr. Songpong Deechongkit for assistance with the analytical ultracentrifuge and CD measurements. , 2001, Angewandte Chemie.
[74] P. Dawson,et al. Synthesis of peptides and proteins without cysteine residues by native chemical ligation combined with desulfurization. , 2001, Journal of the American Chemical Society.
[75] F. Robey. Selective and facile cyclization of N-chloroacetylated peptides from the C4 domain of HIV Gp120 in LiCl/DMF solvent systems. , 2000, The journal of peptide research : official journal of the American Peptide Society.
[76] G. Verdine,et al. An All-Hydrocarbon Cross-Linking System for Enhancing the Helicity and Metabolic Stability of Peptides , 2000 .
[77] W. Meutermans,et al. Synthesis of Difficult Cyclic Peptides by Inclusion of a Novel Photolabile Auxiliary in a Ring Contraction Strategy , 1999 .
[78] M. Mutter,et al. Pseudo-prolines in cyclic peptides: Conformational stabilisation of cyclo[Pro-Thr(ψMe,Mepro)-Pro] , 1999 .
[79] J. Tam,et al. THIA ZIP REACTION FOR SYNTHESIS OF LARGE CYCLIC PEPTIDES : MECHANISMS AND APPLICATIONS , 1999 .
[80] J. Tam,et al. Lactone and Lactam Library Synthesis by Silver Ion-Assisted Orthogonal Cyclization of Unprotected Peptides† , 1999 .
[81] John A. Robinson,et al. Structural Mimicry of Canonical Conformations in Antibody Hypervariable Loops Using Cyclic Peptides Containing a Heterochiral Diproline Template , 1999 .
[82] Helen E Blackwell,et al. Highly Efficient Synthesis of Covalently Cross-Linked Peptide Helices by Ring-Closing Metathesis. , 1998, Angewandte Chemie.
[83] S. Kent,et al. A novel method to synthesize cyclic peptides , 1998 .
[84] Garland R. Marshall,et al. Conformational Analysis of Reverse-Turn Constraints by N-Methylation and N-Hydroxylation of Amide Bonds in Peptides and Non-Peptide Mimetics , 1998 .
[85] H. Nöth,et al. Facile Synthesis of Cyclic Tetrapeptides from Nonactivated Peptide Esters on Metal Centers. , 1998, Angewandte Chemie.
[86] A. Chamberlin,et al. Chemical Synthesis of Natural Product Peptides: Coupling Methods for the Incorporation of Noncoded Amino Acids into Peptides. , 1997, Chemical reviews.
[87] J. Tam,et al. Metal ion-assisted peptide cyclization , 1997 .
[88] James P. Tam,et al. Synthesis and Application of Unprotected Cyclic Peptides as Building Blocks for Peptide Dendrimers , 1997 .
[89] D. Fairlie,et al. Conformational Control by Thiazole and Oxazoline Rings in Cyclic Octapeptides of Marine Origin. Novel Macrocyclic Chair and Boat Conformations. , 1997 .
[90] D. Ryan,et al. PSEUDO-PROLINES AS A MOLECULAR HINGE : REVERSIBLE INDUCTION OF CIS AMIDE BONDS INTO PEPTIDE BACKBONES , 1997 .
[91] Michael Bienert,et al. Cyclization of all-L-Pentapeptides by Means of 1-Hydroxy-7-azabenzotriazole-Derived Uronium and Phosphonium Reagents. , 1996, The Journal of organic chemistry.
[92] D. Fairlie,et al. Conformational control by thiazole and oxazoline rings in cyclic octapeptides of marine origin. Novel macrocyclic chair and boat conformations , 1996 .
[93] J. Tam,et al. Cyclic Peptides from Linear Unprotected Peptide Precursors through Thiazolidine Formation , 1996 .
[94] Scott J. Miller,et al. Application of Ring-Closing Metathesis to the Synthesis of Rigidified Amino Acids and Peptides , 1996 .
[95] M. Mutter,et al. Pseudo-Prolines as a Solubilizing, Structure-Disrupting Protection Technique in Peptide Synthesis , 1996 .
[96] Horst Kessler,et al. Cyclic RGD Peptides Containing β-Turn Mimetics , 1996 .
[97] S. Akabori,et al. Biomimetic Synthesis of Gramicidin S. Direct Formation of the Antibiotic from Pentapeptide Active Esters Having No Protecting Group on the Side Chain of the Orn Residue. , 1994 .
[98] D. Hudson,et al. A novel, convenient, three-dimensional orthogonal strategy for solid-phase synthesis of cyclic peptides , 1993 .
[99] D. Siri,et al. Prediction of the best linear precursor in the synthesis of cyclotetrapeptides by molecular mechanic calculations , 1992 .
[100] R. W. Hoffmann,et al. Flexible Molecules with Defined Shape—Conformational Design , 1992 .
[101] D. Seebach,et al. Solubilization of Peptides in Non‐polar Organic Solvents by the Addition of Inorganic Salts: Facts and Implications , 1989 .
[102] C. Li,et al. New segment-coupling method for peptide synthesis in aqueous solution: application to synthesis of human [Gly17]-beta-endorphin. , 1981, Proceedings of the National Academy of Sciences of the United States of America.
[103] D. Veber,et al. Practical synthesis of cyclic peptides, with an example of dependence of cyclization yield upon linear sequence , 1979 .
[104] S. Hentges,et al. A Vanadium Carbonyl Trihydride, H3V(CO)3diars , 1977 .
[105] M. Rothe,et al. Synthesis of Cyclotri‐L‐prolyl, a Cyclotripeptide Having a Nine‐Membered Ring , 1965 .
[106] G. F. Gause,et al. Gramicidin S and its use in the Treatment of Infected Wounds , 1944, Nature.
[107] S. Ingemann,et al. Improved Auxiliary for the Synthesis of Medium-Sized Bis(lactams) , 2008 .
[108] Valentina Aureggi. 1,3-Dipolar cycloadditions , 2007 .
[109] P. Merino. 1,3-Dipolar Cycloadditions , 2004 .
[110] J. Pelletier,et al. A new tri-orthogonal strategy for peptide cyclization. , 2002, Organic letters.
[111] T. Muir,et al. Chemoselective backbone cyclization of unprotected peptides , 1997 .
[112] T. Muir,et al. Synthesis of proteins by native chemical ligation. , 1994, Science.
[113] T. Y. Tsang. Mechanisms and Applications , 1989 .
[114] J. Smith,et al. Reverse turns in peptides and proteins. , 1980, CRC critical reviews in biochemistry.
[115] K. Kopple,et al. Reverse Turns in Peptides and Protein , 1980 .
[116] S. Mazur,et al. Chemistry of polymer-bound o-benzyne. Frequency of encounter between substituents on crosslinked polystyrenes , 1979 .
[117] J. Rebek,et al. Organic chemistry on the solid phase. Site-site interactions on functionalized polystyrene , 1977 .
[118] K. Lübke,et al. THE SYNTHESIS OF CYCLIC PEPTIDES , 1965 .
[119] R. Sheppard,et al. Peptides—XIII : Effects of configuration on dielectric increments and cyclization of some simple peptides , 1963 .