Mukaiyama’s reagent promoted C–N bond formation: a new method to synthesize 3-alkylquinazolin-4-ones

[1]  T. Mansour,et al.  Oxidative palladium catalysis in S(N)Ar reactions leading to heteroaryl ethers from pyridotriazol-1-yloxy heterocycles with aryl boronic acids. , 2009, Journal of the American Chemical Society.

[2]  Michael G. Yang,et al.  Synthesis of 3-substituted-4(3H)-quinazolinones via HATU-mediated coupling of 4-hydroxyquinazolines with amines. , 2009, Organic letters.

[3]  L. Meijer,et al.  Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: synthesis, biological evaluation and molecular modeling studies. , 2008, European journal of medicinal chemistry.

[4]  T. Mansour,et al.  The scope and mechanism of phosphonium-mediated S(N)Ar reactions in heterocyclic amides and ureas. , 2007, The Journal of organic chemistry.

[5]  N. Argade,et al.  The Chemistry of Recently Isolated Naturally Occurring Quinazolinone Alkaloids , 2006 .

[6]  L. Meijer,et al.  Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3. , 2006, Bioorganic & medicinal chemistry letters.

[7]  B. Song,et al.  Synthesis and antifungal bioactivities of 3-alkylquinazolin- 4-one derivatives. , 2006, Molecules.

[8]  B. Jean-Claude,et al.  The combi-targeting concept: synthesis of stable nitrosoureas designed to inhibit the epidermal growth factor receptor (EGFR). , 2006, Journal of medicinal chemistry.

[9]  T. Mansour,et al.  An efficient direct amination of cyclic amides and cyclic ureas. , 2006, Organic letters.

[10]  C. Montalbetti,et al.  Amide bond formation and peptide coupling , 2005 .

[11]  R. Nilakantan,et al.  2-(Quinazolin-4-ylamino)-[1,4]benzoquinones as covalent-binding, irreversible inhibitors of the kinase domain of vascular endothelial growth factor receptor-2. , 2005, Journal of medicinal chemistry.

[12]  P. Guiry,et al.  Synthesis of Quinazolinones and Quinazolines , 2005 .

[13]  R. Comis,et al.  The current situation: erlotinib (Tarceva) and gefitinib (Iressa) in non-small cell lung cancer. , 2005, The oncologist.

[14]  Galith Abourbeh,et al.  High-affinity epidermal growth factor receptor (EGFR) irreversible inhibitors with diminished chemical reactivities as positron emission tomography (PET)-imaging agent candidates of EGFR overexpressing tumors. , 2005, Journal of medicinal chemistry.

[15]  Q. Zeng,et al.  Antimalarial Activities and Therapeutic Properties of Febrifugine Analogs , 2005, Antimicrobial Agents and Chemotherapy.

[16]  W. Su,et al.  Pd2(dba)3/P(i-BuNCH2CH2)3N-catalyzed Stille cross-coupling of aryl chlorides. , 2004, Organic letters.

[17]  A. Mahamoud,et al.  SYNTHESIS OF NEW QUINAZOLINE DERIVATIVES , 2004 .

[18]  J. Bergman,et al.  Recent Developments in the Field of Quinazoline Chemistry , 2003 .

[19]  Alper,et al.  Palladium-catalyzed cyclocarbonylation of o-iodoanilines with heterocumulenes: regioselective preparation of 4(3H)-quinazolinone derivatives , 2000, The Journal of organic chemistry.

[20]  L. Kuyper,et al.  Synthesis of 1,3-diamino-7,8,9,10-tetrahydropyrido[3,2-f]-quinazolines. Inhibitors of Candida albicans dihydrofolate reductase as potential antifungal agents , 1997 .

[21]  E. B. Skibo,et al.  Rational design of quinazoline-based irreversible inhibitors of human erythrocyte purine nucleoside phosphorylase. , 1991, Biochemistry.

[22]  G. Gunaherath,et al.  Natural Product Chemistry, 125. Synthesis of Quinazolinones Related to the Structure Proposed for Echinozoli-none , 1989 .

[23]  P. Chaudhuri.  Echinozolinone, an alkaloid from Echinops echinatus , 1987 .

[24]  N. Iwasawa,et al.  A CONVENIENT METHOD FOR THE CONSTRUCTION OF β-LACTAM COMPOUNDS FROM β-AMINO ACIDS USING 2-CHLORO-1-METHYLPYRIDINIUM IODIDE AS CONDENSING REAGENT , 1984 .

[25]  T. Mukaiyama.  New Synthetic Reactions Based on the Onium Salts of Aza‐Arenes [New synthetic methods (29)] , 1979 .

[26]  K. Saigo,et al.  A facile synthesis of carboxamides by using 1-methyl-2-halopyridinium iodides as coupling reagents. , 1975 .

[27]  H. Jackson,et al.  Chemosterilization of Schistosoma mansoni , 1968, Nature.

[28]  J. Mead,et al.  An alkaloid with high antimalarial activity from Dichroa febrifuga. , 1947, Journal of the American Chemical Society.