Miconazole, a New Broad‐spectrum Antimycotic, in the Treatment of Vaginal Candidosis
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Introduction Miconazole" is a synthetic I-phenethyl-imidazole (Fig. 1) possessing highly potent and broad-spectrum antifungal and antibacterial activity (1,2). In vitro, i t is a t least as effective as tolnaftate against dermatophytes, as effective as nystatin against yeasts, and as effective as sodium-benzyl-penicillin against gram-positive bacilli and cocci (2). I t is ineffective against gram-negative bacteria. In the clinic, miconazole has proved effective in the topical treatment of chronic tinea pedis and onychomycosis (3, 4); and it is not absorbed when administered topically or iiitravaginally (5). This paper reports the first trial of the new compound against vaginal candidosis.""
[1] J. V. van Cutsem,et al. Treatment of long-term tinea pedis with miconazole. Double-blind clinical evaluation. , 1970, Archives of dermatology.
[2] J. Heeres,et al. The preparation and antimycotic properties of derivatives of 1-phenethylimidazole. , 1969, Journal of medicinal chemistry.