Direct synthesis of oxazolidin-2-ones from tert-butyl allylcarbamate via halo-induced cyclisation
暂无分享,去创建一个
[1] D. S. Reddy,et al. Design, Synthesis, and Identification of Silicon Incorporated Oxazolidinone Antibiotics with Improved Brain Exposure. , 2015, ACS medicinal chemistry letters.
[2] L. Goracci,et al. New potent antibacterials against Gram-positive multiresistant pathogens: effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles. , 2014, Bioorganic & medicinal chemistry.
[3] C. Frost,et al. Copper-catalyzed one-pot synthesis of N-aryl oxazolidinones from amino alcohol carbamates. , 2014, Organic letters.
[4] M. White,et al. N-Boc Amines to Oxazolidinones via Pd(II)/Bis-sulfoxide/Brønsted Acid Co-Catalyzed Allylic C–H Oxidation , 2014, Journal of the American Chemical Society.
[5] Artur M. S. Silva,et al. Synthesis and Transformation of Halochromones , 2014 .
[6] L. Goracci,et al. New linezolid-like 1,2,4-oxadiazoles active against Gram-positive multiresistant pathogens. , 2013, European journal of medicinal chemistry.
[7] Hao Xu,et al. Iron(II)-catalyzed intramolecular aminohydroxylation of olefins with functionalized hydroxylamines. , 2013, Journal of the American Chemical Society.
[8] Á. Molnár. Efficient, selective, and recyclable palladium catalysts in carbon-carbon coupling reactions. , 2011, Chemical reviews.
[9] M. Sukwattanasinitt,et al. Novel synthetic route to 1,4-dihydropyridines from β-amino acrylates by using titanium(IV) chloride under facile conditions , 2010 .
[10] G. Madhusudhan,et al. Stereoselective synthesis of novel (R)- and (S)-5-azidomethyl-2-oxazolidinones from (S)-epichlorohydrin: a key precursor for the oxazolidinone class of antibacterial agents ☆ , 2008 .
[11] Jeffrey C. Culhane,et al. Synthesis of novel oxazolidinone antimicrobial agents. , 2008, Bioorganic & medicinal chemistry.
[12] Akbar Ali,et al. Design and synthesis of HIV-1 protease inhibitors incorporating oxazolidinones as P2/P2' ligands in pseudosymmetric dipeptide isosteres. , 2007, Journal of medicinal chemistry.
[13] Kevin D. Revell,et al. Synthesis of 2-oxazolidinones from beta-lactams: stereospecific total synthesis of (-)-cytoxazone and all of its stereoisomers. , 2007, Organic letters.
[14] J. Adrio,et al. Gold-catalyzed synthesis of alkylidene 2-oxazolidinones and 1,3-oxazin-2-ones. , 2006, The Journal of organic chemistry.
[15] Yoichi M. A. Yamada,et al. Total synthesis and structural elucidation of azaspiracid-1. Final assignment and total synthesis of the correct structure of azaspiracid-1. , 2006, Journal of the American Chemical Society.
[16] P. G. Hultin,et al. Practical Synthesis of Fluorous Oxazolidinone Chiral Auxiliaries from α-Amino Acids , 2005 .
[17] S. Hirono,et al. Convenient synthesis of oxazolidinones by the use of halomethyloxirane, primary amine, and carbonate salt. , 2005, The Journal of organic chemistry.
[18] K. Wheeler,et al. 5-Endo-dig electrophilic cyclization of 1,4-disubstituted but-3-yn-1-ones: regiocontrolled synthesis of 2,5-disubstituted 3-bromo- and 3-iodofurans. , 2005, Organic letters.
[19] S. Jockusch,et al. Stereocontrol within confined spaces: enantioselective photooxidation of enecarbamates inside zeolite supercages. , 2004, Journal of the American Chemical Society.
[20] A. Zakarian,et al. A convergent total synthesis of hemibrevetoxin B. , 2003, Journal of the American Chemical Society.
[21] B. Mallesham,et al. Highly efficient CuI-catalyzed coupling of aryl bromides with oxazolidinones using Buchwald's protocol: a short route to linezolid and toloxatone. , 2003, Organic letters.
[22] M. Carducci,et al. Asymmetric halo aldol reaction (AHA). , 2003, Organic letters.
[23] N. Turro,et al. Highly diastereoselective dioxetane formation in the photooxygenation of enecarbamates with an oxazolidinone chiral auxiliary: steric control in the [2 + 2] cycloaddition of singlet oxygen through conformational alignment. , 2002, Journal of the American Chemical Society.
[24] E. Hu,et al. An aldol-based approach to the asymmetric synthesis of L-callipeltose, the deoxyamino sugar of L-callipeltoside A. , 2001, Organic letters.
[25] S. J. Brickner,et al. Oxazolidinone Antibacterial Agents. An Enantioselective Synthesis of the [6,5,5] Tricyclic Fused Oxazolidinone Ring System and Application to the Synthesis of a Rigid DuP 721 Analogue. , 1996, The Journal of organic chemistry.
[26] D. Ager,et al. 1,2-Amino Alcohols and Their Heterocyclic Derivatives as Chiral Auxiliaries in Asymmetric Synthesis. , 1996, Chemical reviews.
[27] S. J. Brickner,et al. Synthesis and antibacterial activity of U-100592 and U-100766, two oxazolidinone antibacterial agents for the potential treatment of multidrug-resistant gram-positive bacterial infections. , 1996, Journal of medicinal chemistry.
[28] J. Wouters,et al. A reversible monoamine oxidase inhibitor, toloxatone: structural and electronic properties , 1992 .
[29] D. Brittelli,et al. Antibacterials. synthesis and structure-activity studies of 3-aryl-2-oxooxazolidines. 4. Multiply-substituted aryl derivatives. , 1992, Journal of medicinal chemistry.
[30] M. A. Wuonola,et al. Chiral synthesis of DuP 721, a new antibacterial agent , 1989 .
[31] Joel Morris,et al. The total synthesis of the polyether antibiotic X-206 , 1988 .
[32] M. A. Wuonola,et al. Oxazolidinones, a new class of synthetic antibacterial agents: in vitro and in vivo activities of DuP 105 and DuP 721 , 1987, Antimicrobial Agents and Chemotherapy.
[33] W. Hehre,et al. Modeling chemical reactivity. 7. The effect of a change in rate-limiting step on the stereoselectivity of electrophilic addition to allylic alcohols and related chiral alkenes , 1987 .
[34] P. Barr,et al. Nucleic acid related compounds. 38. Smooth and high-yield iodination and chlorination at C-5 of uracil bases and p-toluyl-protected nucleosides , 1982 .
[35] D. Evans,et al. Enantioselective aldol condensations. 2. Erythro-selective chiral aldol condensations via boron enolates , 1981 .