Labeling and preliminary in vivo evaluation of the 5-HT(7) receptor selective agonist [(11)C]E-55888.

[1]  G. Knudsen,et al.  (11)C-labeling and preliminary evaluation of vortioxetine as a PET radioligand. , 2014, Bioorganic & medicinal chemistry letters.

[2]  T. Billard,et al.  Molecular imaging of the serotonin 5-HT7 receptors: from autoradiography to positron emission tomography , 2014, Reviews in the neurosciences.

[3]  G. Knudsen,et al.  Synthesis, radiolabeling and in vivo evaluation of [(11)C](R)-1-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT(7) receptor. , 2014, European journal of medicinal chemistry.

[4]  G. Knudsen,et al.  Anti-PSMA labeled liposomes loaded with Actinium-225 for potential antivascular alpha-radiotherapy , 2014 .

[5]  Anders Ettrup,et al.  Design, synthesis, radiolabeling and in vivo evaluation of potential positron emission tomography (PET) radioligands for brain imaging of the 5-HT₇ receptor. , 2014, Bioorganic & medicinal chemistry.

[6]  L. Chen,et al.  Design and selection parameters to accelerate the discovery of novel central nervous system positron emission tomography (PET) ligands and their application in the development of a novel phosphodiesterase 2A PET ligand. , 2013, Journal of medicinal chemistry.

[7]  G. Knudsen,et al.  Palladium-mediated conversion of para-aminoarylboronic esters into para-aminoaryl-11C-methanes , 2013 .

[8]  G. Knudsen,et al.  Synthesis and in vitro evaluation of oxindole derivatives as potential radioligands for 5-HT(7) receptor imaging with PET. , 2012, ACS chemical neuroscience.

[9]  G. Knudsen,et al.  Synthesis and evaluation of [¹¹C]Cimbi-806 as a potential PET ligand for 5-HT₇ receptor imaging. , 2012, Bioorganic & medicinal chemistry.

[10]  D. Le Bars,et al.  Synthesis and biological evaluation of potential 5-HT(7) receptor PET radiotracers. , 2011, European journal of medicinal chemistry.

[11]  Gitte M Knudsen,et al.  Measuring Endogenous 5-HT Release by Emission Tomography: Promises and Pitfalls , 2010, Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism.

[12]  N. Gillings A restricted access material for rapid analysis of [(11)C]-labeled radiopharmaceuticals and their metabolites in plasma. , 2009, Nuclear medicine and biology.

[13]  P. Hedlund The 5-HT7 receptor and disorders of the nervous system: an overview , 2009, Psychopharmacology.

[14]  D. Zamanillo,et al.  5-HT7 receptor activation inhibits mechanical hypersensitivity secondary to capsaicin sensitization in mice , 2009, PAIN.

[15]  S. Henriksen,et al.  5-HT7 Receptor Inhibition and Inactivation Induce Antidepressantlike Behavior and Sleep Pattern , 2005, Biological Psychiatry.

[16]  P. Whiting,et al.  Genetic knockout and pharmacological blockade studies of the 5-HT7 receptor suggest therapeutic potential in depression , 2005, Neuropharmacology.

[17]  P D Leeson,et al.  Effect of plasma protein binding on in vivo activity and brain penetration of glycine/NMDA receptor antagonists. , 1997, Journal of medicinal chemistry.