SYNTHESIS OF SOME NEW BENZOXAZINE DERIVATIVES OF BIOLOGICAL INTEREST

The synthesis of a number of biologically important imino-quinazolones has been achieved by the condensation of 3amino-2-aryl-4-quinazolone and aromatic aldehydes.

[1]  H. Ishida,et al.  The Effect of Polymerization Conditions on the Density and Tg of Bisphenol-A and Hexafluoroisopropylidene-Containing Polybenzoxazines , 2001 .

[2]  J. Plavec,et al.  A synthesis of alkyl 4-alkyl-2-hydroxy-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-2-carboxylates , 2001 .

[3]  B. Pfeiffer,et al.  Synthesis and in vitro evaluation of new 8-amino-1,4-benzoxazine derivatives as neuroprotective antioxidants. , 1999, Journal of medicinal chemistry.

[4]  K. Rissanen,et al.  Selective derivatisation of resorcarenes: 1. The regioselective formation of tetra-benzoxazine derivatives , 1997 .

[5]  J. Jang,et al.  Cure Studies of a Benzoxazine-Based Phenolic Resin by Isothermal Experiment , 1995 .

[6]  A. Kluge,et al.  Synthesis and antihypertensive activity of 4'-substituted spiro[4H-3,1-benzoxazine-4,4'-piperidin]-2(1H)-ones. , 1983, Journal of medicinal chemistry.

[7]  F. Labrie,et al.  Synthesis and central dopaminergic activities of (+/-)-hexahydro-7H-indolo[3,4-gh][1,4]benzoxazine derivatives [(+/-)-9-oxaergolines]. , 1983, Journal of medicinal chemistry.

[8]  L. Errede.  Acylanthranils. I. The pathway of quinazolone formation in the reaction of acylanthranils with anilines , 1976 .

[9]  M. D. Corbett,et al.  Syntheses of 4-acylamido-1,4-benzoxazine-2,3-diones and 4-(p-toluenesulfonamido)-1,4-benzoxazine-2,3-dione , 1972 .

[10]  B. Decroix,et al.  Intramolecular Addition of a Hydroxyl to an N-Acyliminium System. Application to the Synthesis of Isoindolo[2,1-a][3,1]benzoxazine and Isoindolo[1,2-c][2,4]benzoxazepine Derivatives , 2002 .

[11]  N. El-Din.  Synthesis and potential antibacterial activity of some 1,3-benzoxazin-4-one derivatives , 2000 .

[12]  U. Möllmann,et al.  Relationships Between the Chemical Structure of Substances and Their Antimycobacterial Activity Against Atypical Strains. Part 18. 3-Phenyl-2H-1,3-benzoxazine-2,4(3H)-diones and Isosteric 3-Phenylquinazoline-2,4(1H,3H)-diones , 1999 .