Discovery and optimization of novel constrained pyrrolopyridone BET family inhibitors.
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Ana L. Aguirre | A. Bogdan | Justin D Dietrich | P. Kovar | Chang H. Park | D. Albert | Dachun Liu | Xiaoyu Lin | G. Rajaraman | J. Marjanovic | G. Sheppard | C. Hutchins | Yujia Dai | W. Kati | Rongqi Wang | Le Wang | M. Bui | J. Pratt | T. Magoc | D. Wilcox | Leiming Li | R. Mantei | Xiaoli Huang | K. McDaniel | Yu Shen | S. Fidanze | J. Holms | Lisa A. Hasvold