A simple, novel and convenient method for the synthesis of 1-aminophosphinic acids: synthesis of a novel C2-symmetric phosphinic acid pseudodipeptide

[1]  T. Yamagishi,et al.  Diastereoselective synthesis of alpha,beta'-disubstituted aminomethyl(2-carboxyethyl)phosphinates as phosphinyl dipeptide isosteres. , 2008, Organic letters.

[2]  B. Kaboudin,et al.  First resolution of ( R , R )- and ( S , S )-bis(1-hydroxyphenylmethyl)phosphinic acids via diastereomeric salt formation with enantiopure 1-phenylethylamines , 2008 .

[3]  A. Krężel,et al.  Conformational investigations of bis(α-aminoalkyl)phosphinic acids and studies of the stability of their complexes with Cu(II) , 2008 .

[4]  B. Kaboudin,et al.  β-Cyclodextrin as an efficient catalyst for the one-pot synthesis of 1-aminophosphonic esters in water , 2007 .

[5]  T. Yamagishi,et al.  Diastereoselective Synthesis of Novel α-Amino-α′-hydroxyphosphinates by Hydrophosphinylation of α-Amino-H-phosphinates to Aldehydes , 2007 .

[6]  T. Yamagishi,et al.  Diastereoselective addition of α-substituted α-amino-H-phosphinates to imines using Yb(OTf)3 as an efficient Lewis acid catalyst , 2007 .

[7]  Asit K Chakraborti,et al.  An extremely efficient three-component reaction of aldehydes/ketones, amines, and phosphites (Kabachnik-Fields reaction) for the synthesis of alpha-aminophosphonates catalyzed by magnesium perchlorate. , 2007, The Journal of organic chemistry.

[8]  B. Kaboudin,et al.  A new, efficient, and simple method for the one-pot synthesis of alpha-acetoxyphosphonates from aldehydes under solvent-free conditions. , 2006, Bioorganic & medicinal chemistry letters.

[9]  T. Yamagishi,et al.  Diastereoselective alkylation of iminomethylenephosphinates possessing an asymmetric center at the phosphorus atom , 2006 .

[10]  B. Kaboudin,et al.  A Novel Method for the Synthesis of Bis(1-diethoxyphosphorylalkyl)amines from Diimines , 2006 .

[11]  B. Kaboudin,et al.  A novel method for the separation of bis(alpha-hydroxyalkyl)phosphinic acid diastereoisomers via formation of novel cyclic phosphinic acids. , 2006, The Journal of organic chemistry.

[12]  B. Kaboudin,et al.  TMSCl-promoted addition of diethyl phosphite to an imine for the synthesis of bis [1-diethoxyphosphorylalkyl] amines , 2006 .

[13]  Fatemeh Farjadian,et al.  Synthesis of phosphorothioates using thiophosphate salts , 2006, Beilstein journal of organic chemistry.

[14]  B. Kaboudin,et al.  The first separation and stereochemical determination of bis(α-hydroxyalkyl) phosphinic acids diastereoisomers , 2005 .

[15]  H. Cristau,et al.  Diastereoselective addition of 2H-2-oxo-1,4,2-oxazaphosphinanes to aldehydes and imines. , 2005, The Journal of organic chemistry.

[16]  B. Kaboudin,et al.  A simple and convenient procedure for the synthesis of 1-aminophosphonates from aromatic aldehydes , 2005 .

[17]  F. Saadati,et al.  Alumina-Ammonium Acetate as an Efficient Reagent for the One-Pot Synthesis of cis-2,4,5-Triarylimidazolines from Aromatic Aldehydes , 2005 .

[18]  C. Stevens,et al.  Synthetic methods for azaheterocyclic phosphonates and their biological activity. , 2004, Chemical reviews.

[19]  F. Saadati,et al.  Studies on the synthesis of 1-aminoalkylphosphonates from aldehydes using silica-supported ammonium hydrogen carbonate , 2004 .

[20]  B. Kaboudin,et al.  CONVENIENT SYNTHESIS OF 1-AMINOALKYLPHOSPHONATES UNDER SOLVENT-FREE CONDITIONS , 2004 .

[21]  P. Wieczorek,et al.  Herbicidal activity of phosphonic, phosphinic, and phosphonous acid analogues of phenylglycine and phenylalanine , 1995, Journal of Plant Growth Regulation.

[22]  J. Lewkowski.  The semiempirical study on the addition of the chiral ammonium hypophosphite to an aldehyde , 2004 .

[23]  B. Kaboudin,et al.  Silica-Supported Ammonium Hydrogen Carbonate as an Efficient Reagent for One-Pot Synthesis of 1-Aminophosphonates from Aldehydes , 2003 .

[24]  J. Lewkowski.  The unusual stereochemical behaviour of ferrocenecarboxaldehyde in reaction with chiral alkylammonium hypophosphite , 2003 .

[25]  B. Kaboudin,et al.  Microwave-assisted synthesis of α-aminophosphinic acids from hypophosphorus acid salts under solvent free conditions , 2003 .

[26]  N. Zefirov,et al.  Regioselective synthesis of cis- and trans-2,4,5-triarylimidazolines and 2,4,5-triarylimidazoles from available reagents , 2003 .

[27]  T. Yamagishi,et al.  Diastereoselective synthesis of β-substituted α-hydroxyphosphinates through hydrophosphinylation of α-heteroatom-substituted aldehydes , 2003 .

[28]  B. Kaboudin.  A convenient synthesis of 1-aminophosphonates from 1-hydroxyphosphonates , 2003 .

[29]  B. Kaboudin.  A simple and new method for the synthesis of thiophosphates , 2002 .

[30]  B. Kaboudin.  Novel Methods for the Synthesis of Phosphonate Esters on the Solid Surface , 2002 .

[31]  A. Mazur,et al.  Enantioselective synthesis of phosphinyl peptidomimetics via an asymmetric Michael reaction of phosphinic acids with acrylate derivatives , 2002 .

[32]  R. Nazari,et al.  Microwave-assisted synthesis of 1-aminoalkyl phosphonates under solvent-free conditions , 2001 .

[33]  B. Kaboudin.  Surface-Mediated Solid Phase Reactions: A Simple and New Method for the Synthesis of α-Aminophosphonates under Solvent-Free Conditions , 2001 .

[34]  S. Chandrasekhar,et al.  Three component coupling catalyzed by TaCl5–SiO2: synthesis of α-amino phosphonates , 2001 .

[35]  V. Dive,et al.  Convenient synthesis and diversification of dehydroalaninyl phosphinic peptide analogues. , 2001, Organic Letters.

[36]  R. Nazari,et al.  A CONVENIENT AND MILD PROCEDURE FOR THE PREPARATION OF α-KETO PHOSPHONATES OF 1-HYDROXYPHOSPHONATES UNDER SOLVENT-FREE CONDITIONS USING MICROWAVE , 2001 .

[37]  T. Ishikawa,et al.  Modified guanidines as chiral superbases: the first example of asymmetric silylation of secondary alcohols , 2001 .

[38]  J. Jiráček,et al.  Phosphinic acid compounds in biochemistry, biology and medicine. , 2000, Current medicinal chemistry.

[39]  G. Baziard-Mouysset,et al.  New One-Step Synthesis of 2-Aryl-1H-Imidazoles: Dehydrogenation of 2-Aryl-Δ2-Imidazolines with Dimethylsulfoxide , 2000 .

[40]  Shuj Kobayashi,et al.  Facile synthesis of α-amino phosphonates in water using a Lewis acid–surfactant-combined catalyst , 2000 .

[41]  B. Ranu,et al.  General Procedure for the Synthesis of α-Amino Phosphonates from Aldehydes and Ketones Using Indium(III) Chloride as a Catalyst , 1999 .

[42]  E. Corey,et al.  Enantioselective synthesis of alpha-amino nitriles from N-benzhydryl imines and HCN with a chiral bicyclic guanidine as catalyst. , 1999, Organic letters.

[43]  R. Somanathan,et al.  Synthesis of racemic cis and trans 2,4,5-tripyridylimidazolines , 1998 .

[44]  钱长涛,et al.  One-pot synthesis of α-amino phosphonates from aldehydes using lanthanide triflate as a catalyst , 1998 .

[45]  E. Corey,et al.  A simplified synthesis of (±)-1,2-diphenyl-1,2-diaminoethane (1) from benzaldehyde and ammonia. Revision of the structures of the long-known intermediates “hydrobenzamide” and “amarine” , 1997 .

[46]  W. Chan,et al.  Multiple solid phase synthesis of (RS)-1-aminophosphinic acids , 1996 .

[47]  B. Walker,et al.  A highly convenient route to optically pure α-aminophosphonic acids , 1995 .

[48]  V. Dive,et al.  SYNTHESIS OF 1-(N-BENZYLOXYCARBONYLAMINO)-5-(N-TERBUTYLOXYCARBONYLAMINO)PENTYLPHOSPHINIC ACID , 1994 .

[49]  R. Dommisse,et al.  A novel synthetic route to 1-aminoalkylphosphinic acids , 1994 .

[50]  M. Port,et al.  A practical synthesis of α-aminophosphonic acids. , 1992 .

[51]  Paweł Kafarski,et al.  BIOLOGICAL ACTIVITY OF AMINOPHOSPHONIC ACIDS , 1991 .

[52]  G. Hägele,et al.  SYNTHESIS OF AMINOBENZYLPHOSPHONOUS ACIDS VIA DIRECT AMIDOALKYLATION OF HYPOPHOSPHOROUS ACID , 1990 .

[53]  E. Corey,et al.  Versatile chiral reagent for the highly enantioselective synthesis of either anti or syn ester aldols , 1990 .

[54]  E. Corey,et al.  Practical enantioselective Diels-Alder and aldol reactions using a new chiral controller system , 1989 .

[55]  J. Wood,et al.  Renin inhibitors. Synthesis of transition-state analogue inhibitors containing phosphorus acid derivatives at the scissile bond. , 1989, Journal of medicinal chemistry.

[56]  E. Corey,et al.  Enantioselective synthesis of the C(18) - C(35) segment of immunosuppressant FK-506 using efficient new methodology , 1989 .

[57]  M. Oba,et al.  Formation of N,N'-disubstituted methanediamine derivatives from hexamethyldisilazane and aldehydes via stepwise reactions , 1988 .

[58]  P. Bartlett,et al.  Phosphorus amino acid analogues as inhibitors of leucine aminopeptidase. , 1987, Journal of medicinal chemistry.

[59]  K. Saigo,et al.  Improved optical resolution of (.+-.)-1,2-diphenylethylenediamine. , 1986 .

[60]  C. Hassall,et al.  Synthesis and structure-activity relationships of antibacterial phosphonopeptides incorporating (1-aminoethyl)phosphonic acid and (aminomethyl)phosphonic acid. , 1986, Journal of medicinal chemistry.

[61]  P. Lea,et al.  ORGANIC PHOSPHORUS COMPOUNDS 761 SYNTHESIS AND PROPERTIES OF PHOSPHINOTHRICIN DERIVATIVES , 1983 .

[62]  R. Engel.  Phosphonates as analogues of natural phosphates , 1977 .

[63]  Martin Grayson,et al.  Topics in Phosphorus Chemistry , 1977 .

[64]  R. Gancarz,et al.  A Useful Method for the Preparation of 1-Aminoalkanephosphonic Acids , 1977 .

[65]  D. Seyferth,et al.  Reactions of dimethylphosphono-substituted diazoalkanes. (MeO)2P(O)CR transfer to olefins and 1,3-dipolar additions of (MeO)2P(O)C(N2)R , 1971 .

[66]  J. Barycki,et al.  Simple synthesis of 2-aminoethylphosphonic acid and related compounds , 1970 .

[67]  A. Guttmann,et al.  Synthesis and Antibacterial Activity of Some New Aminophosphinic Acids1 , 1961 .

[68]  H. Schmidt.  Über eine neue Gruppe von organischen Phosphorverbindungen , 1948 .