Facile reduction of aromatic nitro/azido functionality on solid support employing Al/NiCl2·6H2O and Al/NH4Cl: synthesis of pyrrolo[2,1-c][1,4]benzodiazepines
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[1] M. R. Pavia,et al. Multiple simultaneous synthesis of phenolic libraries , 1995, Molecular Diversity.
[2] A. Kamal,et al. Design, synthesis, and evaluation of new noncross-linking pyrrolobenzodiazepine dimers with efficient DNA binding ability and potent antitumor activity. , 2002, Journal of medicinal chemistry.
[3] A. Kamal,et al. Mild and efficient reduction of azides to amines: synthesis of fused [2,1-b]quinazolinones , 2002 .
[4] A. Kamal,et al. Simple and facile reduction of azides to amines: synthesis of DNA interactive pyrrolo[2,1-c][1,4]benzodiazepines , 2002 .
[5] A. Kamal,et al. Efficient solid-phase synthesis of DNA-interactive pyrrolo[2,1-c][1,4]benzodiazepine antitumour antibiotics☆ , 2002 .
[6] A. Kamal,et al. Recent developments in the design, synthesis and structure-activity relationship studies of pyrrolo[2,1-c][1,4]benzodiazepines as DNA-interactive antitumour antibiotics. , 2002, Current Medicinal Chemistry - Anti-Cancer Agents.
[7] A. Kamal,et al. Efficient reduction of aromatic nitro/azido groups on solid support employing indium: synthesis of pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones , 2001 .
[8] A. Kamal,et al. Solid-phase synthesis of pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones. , 2001, Bioorganic & medicinal chemistry letters.
[9] A. Kamal,et al. Reductive cyclization of ω-azido/nitrocarbonyl compounds by samarium iodide: a facile preparation of DNA-binding pyrrolo[2,1-c][1,4]benzodiazepine and its dimers☆ , 2000 .
[10] D. Tumelty,et al. The reduction of aromatic nitro groups on solid supports using sodium hydrosulfite (Na2S2O4) , 2000 .
[11] M. Gallop,et al. Solid-Phase Synthesis of 3,5-Disubstituted 2,3-Dihydro-1,5-benzothiazepin-4(5H)-ones , 1999 .
[12] D. Obrecht,et al. Solid-Phase Synthesis of 3H-Quinazolin-4-ones Based on an Aza Wittig-Mediated annulation Strategy , 1998 .
[13] M. Schwarz,et al. Solid-phase synthesis of substituted 1-phenyl-2-aminomethyl-benzimidazoles and 1-phenyl-2-thiomethyl-benzimidazoles , 1998 .
[14] R. W. Armstrong,et al. Solid support synthesis of polysubstituted tetrahydroquinolines via three-component condensation catalyzed by Yb(OTf)3 , 1998 .
[15] W. DeGrado,et al. Solid-Phase Synthesis of Benzopiperazinones , 1998 .
[16] G. Wei,et al. Solid phase synthesis of benzimidazolones , 1998 .
[17] R. Rivero,et al. Solid phase synthesis of 1-alkyl-2-alkylthio-5-carbamoylbenzimidazoles , 1998 .
[18] R. Rivero,et al. SOLID PHASE SYNTHESIS OF 3,4-DISUBSTITUTED-7-CARBAMOYL-1,2,3,4-TETRAHYDROQUINOXALIN-2-ONES , 1997 .
[19] R. Houghten,et al. The Current Status of Heterocyclic Combinatorial Libraries. , 1997, Chemical reviews.
[20] A. Kamal,et al. Synthesis of pyrrolo[2,1-c][1,4]benzodiazepine antibiotics: Oxidation of cyclic secondary amine with TPAP , 1997 .
[21] I. Hughes. Application of polymer-bound phosphonium salts as traceless supports for solid phase synthesis , 1996 .
[22] P. Schultz,et al. The Solid - Phase Synthesis of Oligoureas , 1996 .
[23] G. Wei,et al. Solid phase synthesis of benzimidazoles , 1996 .
[24] G. Jung,et al. Organic Chemistry on Solid Supports , 1996 .
[25] A. Kamal,et al. A new route for the synthesis of pyrrolo[2,1-c][1,4]benzodiazepine antibiotics via oxidation of cyclic secondary amine , 1996 .
[26] M. J. Gardner,et al. COMBINATORIAL SYNTHESIS : THE DESIGN OF COMPOUND LIBRARIES AND THEIR APPLICATION TO DRUG DISCOVERY , 1995 .
[27] D. Thurston,et al. SYNTHESIS OF DNA-INTERACTIVE PYRROLO2,1-C1,4BENZODIAZEPINES , 1994 .
[28] M. Waring,et al. Molecular Aspects of Anticancer Drug/DNA Interactions , 1993 .
[29] J. Lown,,et al. Molecular mechanism of binding of pyrrolo(1,4)benzodiazepine antitumour agents to deoxyribonucleic acid--anthramycin and tomaymycin. , 1979, Biochemical pharmacology.