A Deoxygenative [4+1] Annulation Involving N‐Acyldiazenes for an Efficient Synthesis of 2,2,5‐Trisubstituted 1,3,4‐Oxadiazole Derivatives

[1]  Ruifeng Li,et al.  Metal-free formal carbon-halogen bond insertion: facile syntheses of 3-halo 3,3'-disubstituted oxindoles and spirooxindole-γ-butyrolactones. , 2017, Chemical communications.

[2]  Kazuyuki Tokumaru,et al.  A convergent synthesis of 1,3,4-oxadiazoles from acyl hydrazides under semiaqueous conditions† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c7sc00195a Click here for additional data file. , 2017, Chemical science.

[3]  Jinyuan Jiang,et al.  P(NMe2)3-Mediated Aziridination of Imines with α-Ketoesters for Synthesis of Aziridine-2-carboxylates. , 2017, The Journal of organic chemistry.

[4]  B. Ashfeld,et al.  Phosphorus(III)-Mediated Stereoconvergent Formal [4+1]-Cycloannulation of 1,2-Dicarbonyls and o-Quinone Methides: A Multicomponent Assembly of 2,3-Dihydrobenzofurans. , 2016, Organic letters.

[5]  Ruifeng Li,et al.  Unusual Formal [1+4] Annulation through Tandem P(NMe2 )3 -Mediated Cyclopropanation/Base-Catalyzed Cyclopropane Rearrangement: Facile Syntheses of Cyclopentenimines and Cyclopentenones. , 2016, Chemistry.

[6]  Ruifeng Li,et al.  P(NMe2)3-mediated reductive [1+4] annulation of isatins with enones: a facile synthesis of spirooxindole-dihydrofurans. , 2015, Chemical communications.

[7]  B. Ashfeld,et al.  Stereochemical implications in the synthesis of 3,3′-spirocyclopropyl oxindoles from β-aryl/alkyl-substituted alkylidene oxindoles , 2015 .

[8]  Lei Wang,et al.  DMAP-Catalyzed [2 + 4] Cycloadditions of Allenoates with N-Acyldiazenes: Direct Method to 1,3,4-Oxadiazine Derivatives. , 2015, Organic letters.

[9]  A. Wu,et al.  Direct Annulation of Hydrazides to 1,3,4-Oxadiazoles via Oxidative C(CO)-C(Methyl) Bond Cleavage of Methyl Ketones. , 2015, Organic letters.

[10]  Qun Chen,et al.  One-Pot Synthesis of 2,5-Diaryl 1,3,4-Oxadiazoles via Di-tert-butyl Peroxide Promoted N-Acylation of Aryl Tetrazoles with Aldehydes. , 2015, The Journal of organic chemistry.

[11]  G. C. Fu,et al.  Use of a new spirophosphine to achieve catalytic enantioselective [4 + 1] annulations of amines with allenes to generate dihydropyrroles. , 2015, Journal of the American Chemical Society.

[12]  Y. Fujiwara,et al.  Biphenyl-derived phosphepines as chiral nucleophilic catalysts: enantioselective [4+1] annulations to form functionalized cyclopentenes. , 2014, Angewandte Chemie.

[13]  Ruifeng Li,et al.  Diastereoselective synthesis of functionalized spirocyclopropyl oxindoles via P(NMe2)3-mediated reductive cyclopropanation. , 2014, The Journal of organic chemistry.

[14]  Xiangying Tang,et al.  Phosphine-catalyzed annulations of 4,4-dicyano-2-methylenebut-3-enoates with maleimides and maleic anhydride. , 2014, Angewandte Chemie.

[15]  M. Shi,et al.  Phosphine-catalyzed asymmetric [4+1] annulation of activated α,β-unsaturated ketones with Morita-Baylis-Hillman carbonates: enantioselective synthesis of spirooxindoles containing two adjacent quaternary stereocenters. , 2014, Chemical communications.

[16]  Fei Wang,et al.  Asymmetric NHC-catalyzed aza-Diels-Alder reactions: highly enantioselective route to α-amino acid derivatives and DFT calculations. , 2014, Organic letters.

[17]  J. Kwiatkowski,et al.  Asymmetric synthesis of spiropyrazolones through phosphine-catalyzed [4+1] annulation. , 2014, Angewandte Chemie.

[18]  Bin Xu,et al.  Pd-catalyzed oxidative annulation of hydrazides with isocyanides: synthesis of 2-amino-1,3,4-oxadiazoles. , 2014, Organic letters.

[19]  Zhengjie He,et al.  Phosphane-catalyzed [4+1] annulation between nitroalkenes and Morita-Baylis-Hillman carbonates: facile synthesis of isoxazoline N-oxides by phosphorus ylides. , 2014, Chemistry, an Asian journal.

[20]  H. Waldmann,et al.  Catalytic Enantioselective 1,3-Dipolar Cycloadditions of Azomethine Ylides for Biology-Oriented Synthesis , 2014, Accounts of chemical research.

[21]  K. Patel,et al.  Review of Synthesis of 1,3,4-Oxadiazole Derivatives , 2014 .

[22]  Andrew D. Smith,et al.  Asymmetric NHC-catalyzed redox α-amination of α-aroyloxyaldehydes. , 2013, Organic letters.

[23]  B. Kalluraya,et al.  Synthesis, characterization and molecular docking studies of some new 1,3,4-oxadiazolines bearing 6-methylpyridine moiety for antimicrobial property. , 2013, European journal of medicinal chemistry.

[24]  H. Lang,et al.  (Multi)ferrocenyl Five-Membered Heterocycles: Excellent Connecting Units for Electron Transfer Studies , 2013 .

[25]  Chihaya Adachi,et al.  Oxadiazole- and triazole-based highly-efficient thermally activated delayed fluorescence emitters for organic light-emitting diodes , 2013 .

[26]  A. T. Radosevich,et al.  Reductive homocondensation of benzylidene- and alkylidenepyruvate esters by a P(NMe2)3-mediated tandem reaction. , 2013, Organic letters.

[27]  J. Barbosa-Filho,et al.  Synthetic Approaches and Pharmacological Activity of 1,3,4-Oxadiazoles: A Review of the Literature from 2000–2012 , 2012, Molecules.

[28]  M. Shi,et al.  Phosphine-catalyzed asymmetric [4+1] annulation of Morita-Baylis-Hillman carbonates with dicyano-2-methylenebut-3-enoates. , 2012, Chemical communications.

[29]  Kerly F. M. Pasqualoto,et al.  Synthesis, molecular modeling and preliminary biological evaluation of a set of 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazole as potential antibacterial, anti-Trypanosoma cruzi and antifungal agents. , 2011, Bioorganic & medicinal chemistry.

[30]  M. Shi,et al.  Chemoselective Reduction of Isatin-Derived Electron-Deficient Alkenes Using Alkylphosphanes as Reduction Reagents , 2011 .

[31]  Zhengjie He,et al.  Phosphine-catalyzed [4 + 1] annulation between α,β-unsaturated imines and allylic carbonates: synthesis of 2-pyrrolines. , 2011, The Journal of organic chemistry.

[32]  K. Mikami,et al.  Palladium-Catalyzed Enantioselective Ene and Aldol Reactions with Isatins, Keto Esters, and Diketones: Reliable Approach to Chiral Tertiary Alcohols , 2011 .

[33]  You Huang,et al.  Phosphine-catalyzed domino reaction: highly stereoselective synthesis of trans-2,3-dihydrobenzofurans from salicyl N-thiophosphinyl imines and allylic carbonates. , 2010, Organic letters.

[34]  Junliang Zhang,et al.  An unexpected phosphine-catalyzed regio- and diastereoselective [4+1] annulation reaction of modified allylic compounds with activated enones. , 2010, Chemistry, an Asian journal.

[35]  Xiaofeng Tong,et al.  2-(Acetoxymethyl)buta-2,3-dienoate, a versatile 1,4-biselectrophile for phosphine-catalyzed (4 + n) annulations with 1,n-Bisnucleophiles (n = 1, 2). , 2010, Journal of the American Chemical Society.

[36]  Zhenming Liu,et al.  Efficient synthesis of a series of novel fructose-based 3-acetyl-5-alkyl-2,3-dihydro-1,3,4-oxadiazole derivatives and studies of the reaction mechanism , 2009 .

[37]  X. Qian,et al.  1,3,4-Oxadiazoline derivatives as novel potential inhibitors targeting chitin biosynthesis: design, synthesis and biological evaluation. , 2009, Bioorganic & medicinal chemistry letters.

[38]  Pan‐Lin Shao,et al.  [4+2] cycloaddition of ketenes with N-benzoyldiazenes catalyzed by N-heterocyclic carbenes. , 2009, Angewandte Chemie.

[39]  X. Qian,et al.  1,3,4-Oxadiazole-3(2H)-carboxamide derivatives as potential novel class of monoamine oxidase (MAO) inhibitors: synthesis, evaluation, and role of urea moiety. , 2008, Bioorganic & medicinal chemistry.

[40]  V. Ratovelomanana-Vidal,et al.  CeCl3.7H2O: an effective additive in Ru-catalyzed enantioselective hydrogenation of aromatic alpha-ketoesters. , 2008, The Journal of organic chemistry.

[41]  K. Scheidt,et al.  Direct amination of homoenolates catalyzed by N-heterocyclic carbenes. , 2008, Journal of the American Chemical Society.

[42]  Yan Pan,et al.  GLB prevents tumor metastasis of Lewis lung carcinoma by inhibiting tumor adhesion actions , 2005, Acta Pharmacologica Sinica.

[43]  Tetsuo Tsutsui,et al.  Blue light‐emitting organic electroluminescent devices , 1990 .

[44]  K. Yamamoto,et al.  In vitro sensitivity of mycoplasmas isolated from various animals and sewage to antibiotics and nitrofurans. , 1971, The Journal of antibiotics.

[45]  平尾 一郎 5-[2-(5-ニトロ-2-フリル)-1-(2-フリル)ビニル]-2-アミノ-1,3,4-オキサジアゾールの合成粘 , 1967 .