Synthesis and SAR of novel conformationally restricted oxazolidinones possessing gram-positive and fastidious gram-negative antibacterial activity. Part 2: Amino substitutions on heterocyclic D-ring system.
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[1] Ji-Young Kim,et al. Synthesis and SAR of novel conformationally-restricted oxazolidinones possessing gram-positive and fastidious gram-negative antibacterial activity. Part 1: Substituted pyrazoles. , 2007, Bioorganic & medicinal chemistry letters.
[2] S. Hagen,et al. Synthesis and structure-activity studies of novel benzocycloheptanone oxazolidinone antibacterial agents. , 2006, Bioorganic & medicinal chemistry letters.
[3] M. Wilcox. Update on linezolid: the first oxazolidinone antibiotic , 2005, Expert opinion on pharmacotherapy.
[4] D. Stevens,et al. A review of linezolid: the first oxazolidinone antibiotic , 2004, Expert review of anti-infective therapy.
[5] A. Nilius. Have the oxazolidinones lived up to their billing? Future perspectives for this antibacterial class. , 2003, Current opinion in investigational drugs.
[6] K. Marotti,et al. Staphylococcus aureus Cell Extract Transcription-Translation Assay: Firefly Luciferase Reporter System for Evaluating Protein Translation Inhibitors , 2001, Antimicrobial Agents and Chemotherapy.
[7] M. Schreier,et al. Pyrazole bioisosteres of leflunomide as B-cell immunosuppressants for xenotransplantation and chronic rejection: scope and limitations. , 1998, Journal of medicinal chemistry.
[8] P D Leeson,et al. 4-Heterocyclylpiperidines as selective high-affinity ligands at the human dopamine D4 receptor. , 1997, Journal of medicinal chemistry.
[9] W. Greenlee,et al. Renin inhibitors containing C-termini derived from mercaptoheterocycles. , 1992, Journal of medicinal chemistry.
[10] R. E. Valter,et al. Preparation of 3-dialkylamino-4-(3,5,6-trichloro-1,4-benzoquinon-2-yl)pyrazoles , 1992 .
[11] S. Rádl. Preparation of Some Pyrazole Derivatives by Extrusion of Elemental Sulfur from 1,3,4-Thiadiazines , 1992 .
[12] H. Oda,et al. 3-Alkylthio and 3-Aminopyrazolo [3,4-d] pyridazines.Ring Contraction of Pyridazino [4,5-e] [1,3,4] thiadiazines via Extrusion of Sulfur. , 1985 .
[13] G. Zubay,et al. In vitro synthesis of protein in microbial systems. , 1973, Annual review of genetics.