Arylpiperazine derivatives of 3-propyl-beta-tetralonohydantoin as new 5-HT1A and 5-HT2A receptor ligands.
暂无分享,去创建一个
[1] L. Pardo,et al. Synthesis and structure-activity relationships of a new model of arylpiperazines. Study of the 5-HT(1a)/alpha(1)-adrenergic receptor affinity by classical hansch analysis, artificial neural networks, and computational simulation of ligand recognition. , 2001, Journal of medicinal chemistry.
[2] P. Grieco,et al. Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. , 2000, Bioorganic & medicinal chemistry.
[3] M. López-Rodríguez,et al. Synthesis and structure-activity relationships of a new model of arylpiperazines. 2. Three-dimensional quantitative structure-activity relationships of hydantoin-phenylpiperazine derivatives with affinity for 5-HT1A and alpha 1 receptors. A comparison of CoMFA models. , 1997, Journal of medicinal chemistry.
[4] B. Łozowicka,et al. The structure of 3[4-(4-phenylpiperazine)butyl]-5,5-diisopropylhydantion-new ligant of serotonin receptors. , 1997 .
[5] M. Pawłowski,et al. 3‐(ω‐Aminoalkyl)‐5,5‐dialkyl(or spirocycloalkyl‐1′,5‐)hydantoins as New 5‐HT1A and 5‐HT2A Receptor Ligands. , 1996 .
[6] I A Cliffe,et al. A pharmacological profile of the selective silent 5-HT1A receptor antagonist, WAY-100635. , 1995, European journal of pharmacology.
[7] H. Berendsen,et al. Depletion of brain serotonin differently affects behaviors induced by 5HT1A, 5HT1C, and 5HT2 receptor activation in rats. , 1991, Behavioral and neural biology.
[8] R. Glennon,et al. Do functional relationships exist between 5-HT1A and 5-HT2 receptors? , 1990, Pharmacology Biochemistry and Behavior.
[9] H. Berendsen,et al. Selective activation of 5HT1A receptors induces lower lip retraction in the rat , 1989, Pharmacology Biochemistry and Behavior.
[10] C. B. Davis,et al. Activity of aromatic substituted phenylpiperazines lacking affinity for dopamine binding sites in a preclinical test of antipsychotic efficacy. , 1989, Journal of medicinal chemistry.
[11] G. Goodwin,et al. The pharmacology of the hypothermic response in mice to 8-hydroxy-2-(DI-n-propylamino)tetralin (8-OH-DPAT) A model of presynaptic 5-HT1 function , 1985, Neuropharmacology.
[12] J. Springer,et al. Bioactive conformation of 1-arylpiperazines at central serotonin receptors. , 1985, Journal of medicinal chemistry.
[13] R. Fuller,et al. Structural relationships in the inhibition of [(3)H]serotonin binding to rat brain membranes in vitro by 1-phenyl-piperazines. , 1980, Biochemical Pharmacology.
[14] J. I. DeGraw,et al. Substituted 1,2,3,4-tetrahydro- -carbolines , 1967 .
[15] W. H. Burton,et al. Potential Growth Antagonists. I. Hydantoins and Disubstituted Glycines1,2 , 1960 .