Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics
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Steven H. Liang | N. Vasdev | Benjamin H. Rotstein | Nickeisha A Stephenson | Nickeisha A. Stephenson
[1] Steven H. Liang,et al. Alternative approaches for PET radiotracer development in Alzheimer's disease: imaging beyond plaque. , 2014, Journal of labelled compounds & radiopharmaceuticals.
[2] M. Yusubov,et al. Applications of iodonium salts and iodonium ylides as precursors for nucleophilic fluorination in Positron Emission Tomography , 2013 .
[3] V. Pike,et al. No-carrier-added [18F]fluoroarenes from the radiofluorination of diaryl sulfoxides. , 2013, Chemical communications.
[4] M. Carroll,et al. Evaluation of tetraethylammonium bicarbonate as a phase-transfer agent in the formation of [18F]fluoroarenes , 2012 .
[5] Eunsung Lee,et al. Nickel-mediated oxidative fluorination for PET with aqueous [18F] fluoride. , 2012, Journal of the American Chemical Society.
[6] V. Pike,et al. Single-step Radiosyntheses of '18F-Labeled Click Synthons' from Azide-functionalized Diaryliodonium Salts. , 2012, European journal of organic chemistry.
[7] J. Passchier,et al. Metal-free oxidative fluorination of phenols with [18F]fluoride. , 2012, Angewandte Chemie.
[8] J. Gelovani,et al. Synthesis and preliminary evaluation of [18F]-labeled 2-oxoquinoline derivatives for PET imaging of cannabinoid CB2 receptor. , 2012, Nuclear medicine and biology.
[9] S. Ametamey,et al. 18F‐Radiolabeling of Aromatic Compounds Using Triarylsulfonium Salts , 2012 .
[10] Jimin Park,et al. Facile aromatic radiofluorination of [18F]flumazenil from diaryliodonium salts with evaluation of their stability and selectivity. , 2011, Organic & biomolecular chemistry.
[11] B. Feringa,et al. Strain-promoted copper-free "click" chemistry for 18F radiolabeling of bombesin. , 2011, Angewandte Chemie.
[12] Eunsung Lee,et al. A Fluoride-Derived Electrophilic Late-Stage Fluorination Reagent for PET Imaging , 2011, Science.
[13] Viktor V. Zhdankin,et al. Iodonium salts in organic synthesis , 2011 .
[14] G. Griffiths,et al. A first synthesis of 18F‐radiolabeled lapatinib: a potential tracer for positron emission tomographic imaging of ErbB1/ErbB2 tyrosine kinase activity , 2011 .
[15] Linlin Qin,et al. Unprecedented directing group ability of cyclophanes in arene fluorinations with diaryliodonium salts. , 2011, Organic letters.
[16] C. Mamat,et al. Cross‐Coupling Reactions as Valuable Tool for the Preparation of PET Radiotracers , 2011 .
[17] H. VanBrocklin,et al. Metabolic stability of 6,7-dialkoxy-4-(2-, 3- and 4-[18F]fluoroanilino)quinazolines, potential EGFR imaging probes. , 2011, Bioorganic & medicinal chemistry.
[18] Bijia Wang,et al. Fluoride-Promoted Ligand Exchange in Diaryliodonium Salts. , 2010, Journal of fluorine chemistry.
[19] F. Wuest,et al. Synthesis and application of 4-[(18)F]fluorobenzylamine: A versatile building block for the preparation of PET radiotracers. , 2010, Organic & biomolecular chemistry.
[20] Linlin Qin,et al. Regiospecific reductive elimination from diaryliodonium salts. , 2010, Angewandte Chemie.
[21] H. Coenen,et al. Three-Step, “One-Pot” Radiosynthesis of 6-Fluoro-3,4-Dihydroxy-l-Phenylalanine by Isotopic Exchange , 2009, Journal of Nuclear Medicine.
[22] A. Luxen,et al. New strategy for the preparation of clickable peptides and labeling with 1-(azidomethyl)-4-[(18)F]-fluorobenzene for PET. , 2009, Bioconjugate chemistry.
[23] Nicholas J Long,et al. Synthesis of 11C, 18F, 15O, and 13N radiolabels for positron emission tomography. , 2008, Angewandte Chemie.
[24] Lisheng Cai,et al. Chemistry with [18F]Fluoride Ion , 2008 .
[25] Pius August Schubiger,et al. Molecular imaging with PET. , 2008, Chemical reviews.
[26] H. Coenen,et al. Nucleophilic 18F-fluorination of heteroaromatic iodonium salts with no-carrier-added [18F]fluoride. , 2007, Journal of the American Chemical Society.
[27] M. Carroll,et al. Fluoridation of 2‐thienyliodonium salts , 2007 .
[28] S. Ametamey,et al. A new precursor for the preparation of 6-[18F]Fluoro-L-m-tyrosine ([18F]FMT): efficient synthesis and comparison of radiolabeling. , 2004, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[29] M E Phelps,et al. Positron emission tomography provides molecular imaging of biological processes. , 2000, Proceedings of the National Academy of Sciences of the United States of America.
[30] V. Pike,et al. Fluoridation of heteroaromatic iodonium salts—experimental evidence supporting theoretical prediction of the selectivity of the process , 2000 .
[31] V. Pike,et al. The synthesis of [18F]fluoroarenes from the reaction of cyclotron-produced [18F]fluoride ion with diaryliodonium salts , 1998 .
[32] A. Wolf,et al. Working Against Time: Rapid Radiotracer Synthesis and Imaging the Human Brain , 1997 .
[33] V. Pike,et al. Reactions of cyclotron-produced [18F]fluoride with diaryliodonium salts—a novel single-step route to no-carrier-added [18]fluoroarenes , 1995 .
[34] J. Barrio,et al. Synthesis of 6-[18F] and 4-[18F]fluoro-L-m-tyrosines via regioselective radiofluorodestannylation. , 1993, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[35] H. Coenen,et al. Direct electrophilic radiofluorination of phenylalanine, tyrosine and dopa , 1988 .
[36] C. Lemaire,et al. A new route for the synthesis of [18F]fluoroaromatic substituted amino acids: no carrier added L-p-[18F]fluorophenylalanine. , 1987, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.
[37] A. Wolf,et al. The synthesis of 18 F-5-fluorouracil. VII. , 1973, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[38] G. Schiemann,et al. Über aromatische Fluorverbindungen, I.: Ein neues Verfahren zu ihrer Darstellung , 1927 .
[39] O. Wallach. Ueber das Verhalten einiger Diazo‐ und Diazoamidoverbindungen , 1886 .