Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics

[1]  Steven H. Liang,et al.  Alternative approaches for PET radiotracer development in Alzheimer's disease: imaging beyond plaque. , 2014, Journal of labelled compounds & radiopharmaceuticals.

[2]  M. Yusubov,et al.  Applications of iodonium salts and iodonium ylides as precursors for nucleophilic fluorination in Positron Emission Tomography , 2013 .

[3]  V. Pike,et al.  No-carrier-added [18F]fluoroarenes from the radiofluorination of diaryl sulfoxides. , 2013, Chemical communications.

[4]  M. Carroll,et al.  Evaluation of tetraethylammonium bicarbonate as a phase-transfer agent in the formation of [18F]fluoroarenes , 2012 .

[5]  Eunsung Lee,et al.  Nickel-mediated oxidative fluorination for PET with aqueous [18F] fluoride. , 2012, Journal of the American Chemical Society.

[6]  V. Pike,et al.  Single-step Radiosyntheses of '18F-Labeled Click Synthons' from Azide-functionalized Diaryliodonium Salts. , 2012, European journal of organic chemistry.

[7]  J. Passchier,et al.  Metal-free oxidative fluorination of phenols with [18F]fluoride. , 2012, Angewandte Chemie.

[8]  J. Gelovani,et al.  Synthesis and preliminary evaluation of [18F]-labeled 2-oxoquinoline derivatives for PET imaging of cannabinoid CB2 receptor. , 2012, Nuclear medicine and biology.

[9]  S. Ametamey,et al.  18F‐Radiolabeling of Aromatic Compounds Using Triarylsulfonium Salts , 2012 .

[10]  Jimin Park,et al.  Facile aromatic radiofluorination of [18F]flumazenil from diaryliodonium salts with evaluation of their stability and selectivity. , 2011, Organic & biomolecular chemistry.

[11]  B. Feringa,et al.  Strain-promoted copper-free "click" chemistry for 18F radiolabeling of bombesin. , 2011, Angewandte Chemie.

[12]  Eunsung Lee,et al.  A Fluoride-Derived Electrophilic Late-Stage Fluorination Reagent for PET Imaging , 2011, Science.

[13]  Viktor V. Zhdankin,et al.  Iodonium salts in organic synthesis , 2011 .

[14]  G. Griffiths,et al.  A first synthesis of 18F‐radiolabeled lapatinib: a potential tracer for positron emission tomographic imaging of ErbB1/ErbB2 tyrosine kinase activity , 2011 .

[15]  Linlin Qin,et al.  Unprecedented directing group ability of cyclophanes in arene fluorinations with diaryliodonium salts. , 2011, Organic letters.

[16]  C. Mamat,et al.  Cross‐Coupling Reactions as Valuable Tool for the Preparation of PET Radiotracers , 2011 .

[17]  H. VanBrocklin,et al.  Metabolic stability of 6,7-dialkoxy-4-(2-, 3- and 4-[18F]fluoroanilino)quinazolines, potential EGFR imaging probes. , 2011, Bioorganic & medicinal chemistry.

[18]  Bijia Wang,et al.  Fluoride-Promoted Ligand Exchange in Diaryliodonium Salts. , 2010, Journal of fluorine chemistry.

[19]  F. Wuest,et al.  Synthesis and application of 4-[(18)F]fluorobenzylamine: A versatile building block for the preparation of PET radiotracers. , 2010, Organic & biomolecular chemistry.

[20]  Linlin Qin,et al.  Regiospecific reductive elimination from diaryliodonium salts. , 2010, Angewandte Chemie.

[21]  H. Coenen,et al.  Three-Step, “One-Pot” Radiosynthesis of 6-Fluoro-3,4-Dihydroxy-l-Phenylalanine by Isotopic Exchange , 2009, Journal of Nuclear Medicine.

[22]  A. Luxen,et al.  New strategy for the preparation of clickable peptides and labeling with 1-(azidomethyl)-4-[(18)F]-fluorobenzene for PET. , 2009, Bioconjugate chemistry.

[23]  Nicholas J Long,et al.  Synthesis of 11C, 18F, 15O, and 13N radiolabels for positron emission tomography. , 2008, Angewandte Chemie.

[24]  Lisheng Cai,et al.  Chemistry with [18F]Fluoride Ion , 2008 .

[25]  Pius August Schubiger,et al.  Molecular imaging with PET. , 2008, Chemical reviews.

[26]  H. Coenen,et al.  Nucleophilic 18F-fluorination of heteroaromatic iodonium salts with no-carrier-added [18F]fluoride. , 2007, Journal of the American Chemical Society.

[27]  M. Carroll,et al.  Fluoridation of 2‐thienyliodonium salts , 2007 .

[28]  S. Ametamey,et al.  A new precursor for the preparation of 6-[18F]Fluoro-L-m-tyrosine ([18F]FMT): efficient synthesis and comparison of radiolabeling. , 2004, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.

[29]  M E Phelps,et al.  Positron emission tomography provides molecular imaging of biological processes. , 2000, Proceedings of the National Academy of Sciences of the United States of America.

[30]  V. Pike,et al.  Fluoridation of heteroaromatic iodonium salts—experimental evidence supporting theoretical prediction of the selectivity of the process , 2000 .

[31]  V. Pike,et al.  The synthesis of [18F]fluoroarenes from the reaction of cyclotron-produced [18F]fluoride ion with diaryliodonium salts , 1998 .

[32]  A. Wolf,et al.  Working Against Time: Rapid Radiotracer Synthesis and Imaging the Human Brain , 1997 .

[33]  V. Pike,et al.  Reactions of cyclotron-produced [18F]fluoride with diaryliodonium salts—a novel single-step route to no-carrier-added [18]fluoroarenes , 1995 .

[34]  J. Barrio,et al.  Synthesis of 6-[18F] and 4-[18F]fluoro-L-m-tyrosines via regioselective radiofluorodestannylation. , 1993, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.

[35]  H. Coenen,et al.  Direct electrophilic radiofluorination of phenylalanine, tyrosine and dopa , 1988 .

[36]  C. Lemaire,et al.  A new route for the synthesis of [18F]fluoroaromatic substituted amino acids: no carrier added L-p-[18F]fluorophenylalanine. , 1987, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

[37]  A. Wolf,et al.  The synthesis of 18 F-5-fluorouracil. VII. , 1973, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.

[38]  G. Schiemann,et al.  Über aromatische Fluorverbindungen, I.: Ein neues Verfahren zu ihrer Darstellung , 1927 .

[39]  O. Wallach Ueber das Verhalten einiger Diazo‐ und Diazoamidoverbindungen , 1886 .