Novel sulfamate derivatives of menthol: Synthesis, characterization, and cholinesterases and carbonic anhydrase enzymes inhibition properties
暂无分享,去创建一个
[1] I. Gulcin,et al. Antidiabetic and antiparasitic potentials: Inhibition effects of some natural antioxidant compounds on α-glycosidase, α-amylase and human glutathione S-transferase enzymes. , 2018, International journal of biological macromolecules.
[2] P. Taslimi,et al. Synthesis, characterization and crystal structure of 2-(4-hydroxyphenyl)ethyl and 2-(4-nitrophenyl)ethyl Substituted Benzimidazole Bromide Salts: Their inhibitory properties against carbonic anhydrase and acetylcholinesterase , 2018, Journal of Molecular Structure.
[3] Murat Yiğit,et al. Novel Benzylic Substituted Imidazolinium, Tetrahydropyrimidinium and Tetrahydrodiazepinium Salts: Potent Carbonic Anhydrase and Acetylcholinesterase Inhibitors , 2018, ChemistrySelect.
[4] C. Supuran,et al. Intermolecular amination of allylic and benzylic alcohols leads to effective inhibitions of acetylcholinesterase enzyme and carbonic anhydrase I and II isoenzymes , 2018, Journal of biochemical and molecular toxicology.
[5] I. Gulcin,et al. Sulfonamide inhibitors: a patent review 2013-present , 2018, Expert opinion on therapeutic patents.
[6] P. Taslimi,et al. The rst synthesis and antioxidant and anticholinergic activities of 1-(4,5-dihydroxybenzyl)pyrrolidin-2-one derivative bromophenols including natural products , 2018, TURKISH JOURNAL OF CHEMISTRY.
[7] P. Taslimi,et al. Antioxidant and anticholinergic properties of olivetol , 2018 .
[8] I. Gulcin,et al. Synthesis and discovery of potent carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase, and α‐glycosidase enzymes inhibitors: The novel N,N′‐bis‐cyanomethylamine and alkoxymethylamine derivatives , 2018, Journal of biochemical and molecular toxicology.
[9] I. Gulcin,et al. Synthesis, molecular modeling, and biological evaluation of 4‐[5‐aryl‐3‐(thiophen‐2‐yl)‐4,5‐dihydro‐1H‐pyrazol‐1‐yl] benzenesulfonamides toward acetylcholinesterase, carbonic anhydrase I and II enzymes , 2018, Chemical biology & drug design.
[10] P. Taslimi,et al. 2-Hydroxyethyl substituted NHC precursors: Synthesis, characterization, crystal structure and carbonic anhydrase, α-glycosidase, butyrylcholinesterase, and acetylcholinesterase inhibitory properties , 2018 .
[11] I. Gülçin,et al. The in vivo effects of cefazolin, cefuroxime, and cefoperazon on the carbonic anhydrase in different rat tissues , 2018, Journal of biochemical and molecular toxicology.
[12] I. Gulcin,et al. Synthesis and biological evaluation of phloroglucinol derivatives possessing α‐glycosidase, acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase inhibitory activity , 2018, Archiv der Pharmazie.
[13] I. Gulcin,et al. Synthesis and investigation of the conversion reactions of pyrimidine‐thiones with nucleophilic reagent and evaluation of their acetylcholinesterase, carbonic anhydrase inhibition, and antioxidant activities , 2018, Journal of biochemical and molecular toxicology.
[14] I. Gulcin,et al. The toxicological effects of some avermectins on goat liver carbonic anhydrase enzyme , 2018, Journal of biochemical and molecular toxicology.
[15] P. Taslimi,et al. Synthesis of chalcone-imide derivatives and investigation of their anticancer and antimicrobial activities, carbonic anhydrase and acetylcholinesterase enzymes inhibition profiles , 2018, Archives of physiology and biochemistry.
[16] I. Gulcin,et al. Synthesis and Carbonic Anhydrase Inhibition of Tetrabromo Chalcone Derivatives , 2017, Archiv der Pharmazie.
[17] C. Supuran,et al. The synthesis of novel sulfamides derived from β-benzylphenethylamines as acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase enzymes inhibitors. , 2017, Bioorganic chemistry.
[18] P. Taslimi,et al. Novel antioxidant bromophenols with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions. , 2017, Bioorganic chemistry.
[19] I. Gulcin,et al. The impact of some natural phenolic compounds on carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase, and α‐glycosidase enzymes: An antidiabetic, anticholinergic, and antiepileptic study , 2017, Journal of biochemical and molecular toxicology.
[20] I. Gulcin,et al. Investigation of acetylcholinesterase and mammalian DNA topoisomerases, carbonic anhydrase inhibition profiles, and cytotoxic activity of novel bis(α‐aminoalkyl)phosphinic acid derivatives against human breast cancer , 2017, Journal of biochemical and molecular toxicology.
[21] I. Gulcin,et al. Inhibitory effects of oxytocin and oxytocin receptor antagonist atosiban on the activities of carbonic anhydrase and acetylcholinesterase enzymes in the liver and kidney tissues of rats , 2017, Journal of biochemical and molecular toxicology.
[22] P. Taslimi,et al. Synephrine and phenylephrine act as α‐amylase, α‐glycosidase, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase enzymes inhibitors , 2017, Journal of biochemical and molecular toxicology.
[23] I. Gulcin,et al. Synthesis of new cyclic thioureas and evaluation of their metal‐chelating activity, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase inhibition profiles , 2017, Journal of biochemical and molecular toxicology.
[24] P. Taslimi,et al. Novel NHC Precursors: Synthesis, Characterization, and Carbonic Anhydrase and Acetylcholinesterase Inhibitory Properties , 2017, Archiv der Pharmazie.
[25] P. Taslimi,et al. The first synthesis of 4-phenylbutenone derivative bromophenols including natural products and their inhibition profiles for carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase enzymes. , 2017, Bioorganic chemistry.
[26] I. Gulcin,et al. Discovery of potent carbonic anhydrase, acetylcholinesterase, and butyrylcholinesterase enzymes inhibitors: The new amides and thiazolidine‐4‐ones synthesized on an acetophenone base , 2017, Journal of biochemical and molecular toxicology.
[27] I. Gülçin,et al. Synthesis of Mannich Bases by Two Different Methods and Evaluation of their Acetylcholine Esterase and Carbonic Anhydrase Inhibitory Activities , 2017 .
[28] I. Gülçin,et al. Inhibition properties of some flavonoids on carbonic anhydrase I and II isoenzymes purified from human erythrocytes , 2017, Journal of biochemical and molecular toxicology.
[29] I. Gulcin,et al. Synthesis and biological evaluation of aminomethyl and alkoxymethyl derivatives as carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase inhibitors , 2017, Journal of enzyme inhibition and medicinal chemistry.
[30] I. Gulcin,et al. Synthesis, carbonic anhydrase I and II inhibition studies of the 1,3,5-trisubstituted-pyrazolines , 2016, Journal of enzyme inhibition and medicinal chemistry.
[31] A. Naderi,et al. Antioxidant Activity, Acetylcholinesterase, and Carbonic Anhydrase Inhibitory Properties of Novel Ureas Derived from Phenethylamines , 2016, Archiv der Pharmazie.
[32] C. Supuran,et al. The effect of caffeic acid phenethyl ester (CAPE) on metabolic enzymes including acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase, lactoperoxidase, and carbonic anhydrase isoenzymes I, II, IX, and XII , 2016, Journal of enzyme inhibition and medicinal chemistry.
[33] I. Gülçin,et al. Discovery of Potent Carbonic Anhydrase and Acetylcholinesterase Inhibitors: 2-Aminoindan β-Lactam Derivatives , 2016, International journal of molecular sciences.
[34] I. Gulcin,et al. Synthesis of 4-(2-substituted hydrazinyl)benzenesulfonamides and their carbonic anhydrase inhibitory effects , 2016, Journal of enzyme inhibition and medicinal chemistry.
[35] C. Supuran,et al. The effects of some bromophenols on human carbonic anhydrase isoenzymes , 2016, Journal of enzyme inhibition and medicinal chemistry.
[36] I. Gulcin,et al. Synthesis of 4,5-disubstituted-2-thioxo-1,2,3,4-tetrahydropyrimidines and investigation of their acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase I/II inhibitory and antioxidant activities , 2016, Journal of enzyme inhibition and medicinal chemistry.
[37] I. Gülçin,et al. Purification and characterization of the carbonic anhydrase enzyme from Black Sea trout (Salmo trutta Labrax Coruhensis) kidney and inhibition effects of some metal ions on enzyme activity. , 2016 .
[38] C. Supuran,et al. Synthesis of diaryl ethers with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions , 2016, Journal of enzyme inhibition and medicinal chemistry.
[39] C. Supuran,et al. Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds. , 2016, Bioorganic & medicinal chemistry.
[40] I. Gulcin,et al. The synthesis of some β-lactams and investigation of their metal-chelating activity, carbonic anhydrase and acetylcholinesterase inhibition profiles , 2016, Journal of enzyme inhibition and medicinal chemistry.
[41] I. Gulcin,et al. Synthesis and bioactivity studies on new 4-(3-(4-Substitutedphenyl)-3a,4-dihydro-3H-indeno[1,2-c]pyrazol-2-yl) benzenesulfonamides , 2016, Journal of enzyme inhibition and medicinal chemistry.
[42] I. Gulcin,et al. Synthesis of some tetrahydropyrimidine-5-carboxylates, determination of their metal chelating effects and inhibition profiles against acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase , 2016, Journal of enzyme inhibition and medicinal chemistry.
[43] C. Supuran,et al. Rosmarinic acid inhibits some metabolic enzymes including glutathione S-transferase, lactoperoxidase, acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase isoenzymes , 2016, Journal of enzyme inhibition and medicinal chemistry.
[44] I. Gulcin,et al. The human carbonic anhydrase isoenzymes I and II (hCA I and II) inhibition effects of trimethoxyindane derivatives , 2016, Journal of enzyme inhibition and medicinal chemistry.
[45] C. Supuran,et al. Spirobisnaphthalenes effectively inhibit carbonic anhydrase , 2015, Journal of enzyme inhibition and medicinal chemistry.
[46] I. Gulcin,et al. Purification and characterization of the carbonic anhydrase enzyme from Black Sea trout (Salmo trutta Labrax Coruhensis) kidney and inhibition effects of some metal ions on enzyme activity. , 2016, Environmental toxicology and pharmacology.
[47] C. Supuran,et al. Carbonic anhydrase inhibitors: guaiacol and catechol derivatives effectively inhibit certain human carbonic anhydrase isoenzymes (hCA I, II, IX and XII) , 2015, Journal of enzyme inhibition and medicinal chemistry.
[48] C. Supuran,et al. Discovery of potent carbonic anhydrase and acetylcholine esterase inhibitors: novel sulfamoylcarbamates and sulfamides derived from acetophenones. , 2015, Bioorganic & medicinal chemistry.
[49] Recep Demir,et al. Changes in the anti-oxidant system in adult epilepsy patients receiving anti-epileptic drugs , 2015, Archives of physiology and biochemistry.
[50] C. Supuran,et al. N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II. , 2015, Bioorganic & medicinal chemistry.
[51] P. L. Rosalen,et al. Antibacterial Activity of Essential Oils and Their Isolated Constituents against Cariogenic Bacteria: A Systematic Review , 2015, Molecules.
[52] C. Supuran,et al. Carbonic anhydrase and acetylcholinesterase inhibitory effects of carbamates and sulfamoylcarbamates , 2015, Journal of enzyme inhibition and medicinal chemistry.
[53] C. Supuran,et al. Synthesis and carbonic anhydrase isoenzymes I, II, IX, and XII inhibitory effects of dimethoxybromophenol derivatives incorporating cyclopropane moieties. , 2015, Journal of medicinal chemistry.
[54] I. Gülçin,et al. Synthesis and Carbonic Anhydrase Inhibitory Effects of Novel Sulfamides Derived from 1‐Aminoindanes and Anilines , 2014, Archiv der Pharmazie.
[55] A. Naderi,et al. Carbonic anhydrase inhibitory properties of novel benzylsulfamides using molecular modeling and experimental studies. , 2014, Bioorganic chemistry.
[56] I. Gulcin,et al. Capsaicin: A Potent Inhibitor of Carbonic Anhydrase Isoenzymes , 2014, Molecules.
[57] I. Gülçin,et al. Synthesis and Carbonic Anhydrase Isoenzymes Inhibitory Effects of Brominated Diphenylmethanone and Its Derivatives , 2014, Archiv der Pharmazie.
[58] I. Gülçin,et al. Rosmarinic acid: a potent carbonic anhydrase isoenzymes inhibitor , 2014 .
[59] I. Gülçin,et al. Synthesis and carbonic anhydrase isoenzymes I and II inhibitory effects of novel benzylamine derivatives , 2014, Journal of enzyme inhibition and medicinal chemistry.
[60] I. Gülçin,et al. Novel Sulphamides and Sulphonamides Incorporating the Tetralin Scaffold as Carbonic Anhydrase and Acetylcholine Esterase Inhibitors , 2014, Archiv der Pharmazie.
[61] C. Supuran,et al. In vitro inhibition of α-carbonic anhydrase isozymes by some phenolic compounds. , 2011, Bioorganic & medicinal chemistry letters.
[62] H. Imagawa,et al. Intermolecular Amination of Allyl Alcohols with Sulfamates: Effective Utilization of Mercuric Catalyst , 2011 .
[63] Claudiu T. Supuran,et al. Carbonic anhydrase inhibitors and their therapeutic potential , 2000 .
[64] R. Eccles. Menthol and Related Cooling Compounds , 1994, The Journal of pharmacy and pharmacology.
[65] J. Edsall,et al. Esterase activities of human carbonic anhydrases B and C. , 1967, The Journal of biological chemistry.
[66] K. Courtney,et al. A new and rapid colorimetric determination of acetylcholinesterase activity. , 1961, Biochemical pharmacology.