Design, synthesis, and characterization of a series of cytochrome P(450) 3A-activated prodrugs (HepDirect prodrugs) useful for targeting phosph(on)ate-based drugs to the liver.
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M. Erion | P. D. van Poelje | K. R. Reddy | B. Ugarkar | Michael C. Matelich | J. Schanzer | S. Boyer | R. Lemus | Jorge E. Gomez-Galeno | T. Colby | K. Raja Reddy | Serge H. Boyer