Inhibitions of monoamine oxidases by ferulic acid hydrazide derivatives: synthesis, biochemistry, and computational evaluation
暂无分享,去创建一个
M. Ghoneim | B. Mathew | S. Selim | S. Dev | Hoon Kim | M. A. Abdelgawad | Mohamed E. Shaker | Arshida Thottile Peedikayil | Jiseong Lee | Sunil Kumar
[1] M. Abdelgawad,et al. Development of Halogenated-Chalcones Bearing with Dimethoxy Phenyl Head as Monoamine Oxidase-B Inhibitors , 2022, Pharmaceuticals.
[2] Woong-Hee Shin,et al. Synthesis of 4-substituted benzyl-2-triazole-linked-tryptamine-paeonol derivatives and evaluation of their selective inhibitions against butyrylcholinesterase and monoamine oxidase-B. , 2022, International Journal of Biological Macromolecules.
[3] A. Mardinoğlu,et al. Therapeutic Potential of Ferulic Acid in Alzheimer's Disease. , 2021, Current drug delivery.
[4] Hoon Kim,et al. Aldoxime- and Hydroxy-Functionalized Chalcones as Highly Potent and Selective Monoamine Oxidase-B Inhibitors , 2021, Journal of Molecular Structure.
[5] S. Mishra,et al. A review on ferulic acid and analogs based scaffolds for the management of Alzheimer's disease. , 2021, European journal of medicinal chemistry.
[6] E. Uriarte,et al. Combined 3D-QSAR and docking analysis for the design and synthesis of chalcones as potent and selective monoamine oxidase B inhibitors. , 2021, Bioorganic chemistry.
[7] Hoon Kim,et al. A New Potent and Selective Monoamine Oxidase‐B Inhibitor with Extended Conjugation in a Chalcone Framework: 1‐[4‐(Morpholin‐4‐yl)phenyl]‐5‐phenylpenta‐2,4‐dien‐1‐one , 2020 .
[8] B. Mathew. 1-[4-(morpholin-4-yl)phenyl]-5-phenylpenta-2,4-dien-1-one as a new potent and selective monoamine oxidase-B inhibitor with extended conjugation in chalcone framework. , 2020, ChemMedChem.
[9] S. Devenish. The current landscape in Alzheimer's disease research and drug discovery. , 2020, Drug discovery today.
[10] J. P. Lee,et al. Calycosin and 8-O-methylretusin isolated from Maackia amurensis as potent and selective reversible inhibitors of human monoamine oxidase-B. , 2020, International journal of biological macromolecules.
[11] Piyoosh Sharma,et al. Design, synthesis, and biological evaluation of ferulic acid based 1,3,4-oxadiazole hybrids as multifunctional therapeutics for the treatment of Alzheimer's disease. , 2019, Bioorganic chemistry.
[12] J. P. Lee,et al. Design, synthesis and biological evaluation of oxygenated chalcones as potent and selective MAO-B inhibitors. , 2019, Bioorganic chemistry.
[13] S. Carradori,et al. Emerging therapeutic potentials of dual‐acting MAO and AChE inhibitors in Alzheimer's and Parkinson's diseases , 2019, Archiv der Pharmazie.
[14] L. Milella,et al. Carboxamides vs. methanimines: Crystal structures, binding interactions, photophysical studies, and biological evaluation of (indazole-5-yl)methanimines as monoamine oxidase B and acetylcholinesterase inhibitors. , 2019, European journal of medicinal chemistry.
[15] Yue Wang,et al. Discovery of coumarin Mannich base derivatives as multifunctional agents against monoamine oxidase B and neuroinflammation for the treatment of Parkinson's disease. , 2019, European journal of medicinal chemistry.
[16] J. P. Lee,et al. Rhamnocitrin isolated from Prunus padus var. seoulensis: A potent and selective reversible inhibitor of human monoamine oxidase A. , 2019, Bioorganic chemistry.
[17] Daeui Park,et al. Selective inhibition of monoamine oxidase A by hispidol. , 2018, Bioorganic & medicinal chemistry letters.
[18] A. Tripathi,et al. Privileged scaffolds as MAO inhibitors: Retrospect and prospects. , 2018, European journal of medicinal chemistry.
[19] B. Korkut,et al. Design, Synthesis and Biological Evaluation of Novel N-Pyridyl-Hydrazone Derivatives as Potential Monoamine Oxidase (MAO) Inhibitors , 2018, Molecules.
[20] S. Ilgın,et al. Synthesis of New Hydrazone Derivatives for MAO Enzymes Inhibitory Activity , 2017, Molecules.
[21] B. Winblad,et al. Monoamine oxidase B is elevated in Alzheimer disease neurons, is associated with γ-secretase and regulates neuronal amyloid β-peptide levels , 2017, Alzheimer's Research & Therapy.
[22] Daeui Park,et al. Potent inhibition of monoamine oxidase A by decursin from Angelica gigas Nakai and by wogonin from Scutellaria baicalensis Georgi. , 2017, International journal of biological macromolecules.
[23] N. Tzvetkov,et al. Crystal structures, binding interactions, and ADME evaluation of brain penetrant N-substituted indazole-5-carboxamides as subnanomolar, selective monoamine oxidase B and dual MAO-A/B inhibitors. , 2017, European journal of medicinal chemistry.
[24] Hong Jiang,et al. Novel ferulic amide derivatives with tertiary amine side chain as acetylcholinesterase and butyrylcholinesterase inhibitors: The influence of carbon spacer length, alkylamine and aromatic group. , 2017, European journal of medicinal chemistry.
[25] B. Kumar,et al. A Perspective on Monoamine Oxidase Enzyme as Drug Target: Challenges and Opportunities. , 2016, Current drug targets.
[26] Oscar M. Bautista-Aguilera,et al. The Antioxidant Additive Approach for Alzheimer's Disease Therapy: New Ferulic (Lipoic) Acid Plus Melatonin Modified Tacrines as Cholinesterases Inhibitors, Direct Antioxidants, and Nuclear Factor (Erythroid-Derived 2)-Like 2 Activators. , 2016, Journal of medicinal chemistry.
[27] Daeui Park,et al. Potent selective monoamine oxidase B inhibition by maackiain, a pterocarpan from the roots of Sophora flavescens. , 2016, Bioorganic & medicinal chemistry letters.
[28] R. Ramsay. Molecular aspects of monoamine oxidase B , 2016, Progress in Neuro-Psychopharmacology and Biological Psychiatry.
[29] B. Mathew,et al. Monoamine Oxidase Inhibitors: Perspective Design for the Treatment of Depression and Neurological Disorders , 2016 .
[30] B. Mathew,et al. Synthesis, Biochemistry, and Computational Studies of Brominated Thienyl Chalcones: A New Class of Reversible MAO‐B Inhibitors , 2016, ChemMedChem.
[31] M. Di Carlo,et al. Ferulic Acid: A Hope for Alzheimer’s Disease Therapy from Plants , 2015, Nutrients.
[32] A. Sureda,et al. Ferulic Acid and Alzheimer’s Disease: Promises and Pitfalls , 2015 .
[33] L. Profire,et al. New hydrazones of ferulic acid: synthesis, characterization and biological activity. , 2014, Revista medico-chirurgicala a Societatii de Medici si Naturalisti din Iasi.
[34] Naresh Kumar,et al. Potential applications of ferulic acid from natural sources , 2014, Biotechnology reports.
[35] C. Mancuso,et al. Ferulic acid: pharmacological and toxicological aspects. , 2014, Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association.
[36] S. Vilar,et al. Monoamine oxidase inhibitors: ten years of docking studies. , 2012, Current topics in medicinal chemistry.
[37] Angelo Carotti,et al. Structures of human monoamine oxidase B complexes with selective noncovalent inhibitors: safinamide and coumarin analogs. , 2007, Journal of medicinal chemistry.
[38] J. N. Dixit. Retrospect and Prospects , 2003 .
[39] Hilde van der Togt,et al. Publisher's Note , 2003, J. Netw. Comput. Appl..