Selective functionalization of 1,2-dihydronaphthalenols leads to a concise, stereoselective synthesis of sertraline
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[1] M. Lautens,et al. Scope of the nickel catalyzed asymmetric reductive ring opening reaction. Synthesis of enantiomerically enriched cyclohexenols , 1998 .
[2] M. Lautens,et al. Metal catalyzed hydrometalations and their applications in synthesis , 1998 .
[3] M. Lautens,et al. A New Route to the Enantioselective Synthesis of Cycloheptenols. Temperature Effects in the Asymmetric Reductive Ring Opening of [3.2.1] Oxabicycloalkenes , 1997 .
[4] M. Lautens,et al. General Strategy toward the Tetrahydronaphthalene Skeleton. An Expedient Total Synthesis of Sertraline , 1997 .
[5] A. Kamal,et al. An efficient method for 4β-anilino-4′-demethylepipodophyllotoxins: Synthesis of NPF and W-68 , 1996 .
[6] Jonathan A. Ellman,et al. Synthesis and Applications of Small Molecule Libraries. , 1996, Chemical reviews.
[7] V. Farina. New perspectives in the cross-coupling reactions of organostannanes , 1996 .
[8] G. Sulikowski,et al. Application of Glycosyltetrazoles in Oligosaccharide Synthesis: Assembly of the C3 Trisaccharide Component of the Antibiotic PI-080 , 1996 .
[9] T. Honda,et al. Enantiodivergent Synthesis of the Key Intermediate for Aphanorphine by Chemoenzymatic Process , 1995 .
[10] Norio Miyaura,et al. Palladium-Catalyzed Cross-Coupling Reactions of Organoboron Compounds , 1995 .
[11] R. Mailman,et al. Synthesis and evaluation of 6,7-dihydroxy-2,3,4,8,9,13b-hexahydro-1H- benzo[6,7]cyclohepta[1,2,3-ef][3]benzazepine, 6,7-dihydroxy- 1,2,3,4,8,12b-hexahydroanthr[10,4a,4-cd]azepine, and 10-(aminomethyl)-9,10- dihydro-1,2-dihydroxyanthracene as conformationally restricted analogs of beta-phenyldopamine , 1995, Journal of medicinal chemistry.
[12] W. Cabri,et al. Recent Developments and New Perspectives in the Heck Reaction , 1995 .
[13] M. Leopoldo,et al. High affinity and selectivity on 5-HT1A receptor of 1-aryl-4-[1-tetralin)alkyl]piperazines. 2. , 1995, Journal of medicinal chemistry.
[14] A. Meijere,et al. Fine Feathers Make Fine Birds: The Heck Reaction in Modern Garb† , 1995 .
[15] M. Lautens,et al. Nickel-Catalyzed Hydroalumination of Oxabicyclic Alkenes. Ligand Effects on the Regio- and Enantioselectivity , 1995 .
[16] S. Wright,et al. Fluoride-Mediated Boronic Acid Coupling Reactions , 1994 .
[17] K. Houk,et al. Stereoselective epoxidations and electrophilic additions to partial ergot alkaloids and conformationally-fixed styrenes. Experimental and theoretical modeling evidence for the importance of torsional steering as a stereocontrol element , 1994 .
[18] Anil Kumar,et al. Asymmetric Synthesis of the AB Ring Segments of Daunomycin and 4-Demethoxydaunomycin , 1994 .
[19] W. Cabri,et al. 1,10-Phenanthroline derivatives: a new ligand class in the Heck reaction. Mechanistic aspects , 1993 .
[20] D. Mathre,et al. Direct conversion of activated alcohols to azides using diphenyl phosphorazidate. A practical alternative to mitsunobu conditions , 1993 .
[21] A. M. Myers,et al. Synthesis and pharmacological evaluation of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for a novel receptor with sigma-like neuromodulatory activity. , 1993, Journal of medicinal chemistry.
[22] Davidr . Evans,et al. Substrate-directable chemical reactions , 1993 .
[23] N. Miyaura,et al. Palladium-catalyzed inter- and intramolecular cross-coupling reactions of B-alkyl-9-borabicyclo[3.3.1]nonane derivatives with 1-halo-1-alkenes or haloarenes. Syntheses of functionalized alkenes, arenes, and cycloalkenes via a hydroboration-coupling sequence , 1989 .
[24] R. Larock,et al. Palladium-catalyzed intermolecular allylic arylation of cyloalkenes , 1988 .
[25] L. Arvidsson,et al. Resolved cis- and trans-2-amino-5-methoxy-1-methyltetralins: central dopamine receptor agonists and antagonists. , 1987, Journal of medicinal chemistry.
[26] John M. Brown. Directed Homogeneous Hydrogenation [New Synthetic Methods (65)] , 1987 .
[27] H. Wong,et al. Total synthesis of (±) podophyllotoxin , 1987 .
[28] C. P. Vandermaelen,et al. Buspirone analogues. 2. Structure-activity relationships of aromatic imide derivatives. , 1986, Journal of medicinal chemistry.
[29] R. Crabtree,et al. Directing effects in homogeneous hydrogenation with [Ir(cod)(PCy3)(py)]PF6 , 1986 .
[30] William Bauta,et al. A regioselective entry to vinyllithiums from unsymmetrical ketones via enol triflates , 1986 .
[31] R. Sarges,et al. Nontricyclic antidepressant agents derived from cis- and trans-1-amino-4-aryltetralins. , 1984, Journal of medicinal chemistry.
[32] D. Kahne,et al. Stereocontrol in homogeneous catalytic hydrogenation via hydroxyl group coordination , 1983 .
[33] A. Takénaka,et al. Synthesis and immunological activity of 5,6,6a,8,9,11a-hexahydronaphth[1',2':4,5]imidazo[2,1-b]thiazoles and 5,6,6a,9,10,11a-hexahydroanaphth[2',1':4,5]imidazo[2,1-b]thiazoles. , 1980, Journal of medicinal chemistry.