Interconversion into a low active state protects vascular 5-HT2-receptors against irreversible antagonism by phenoxybenzamine
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[1] A. Kaumann,et al. Allosteric properties of the 5-HT2 receptor system of the rat tail artery , 1987, Naunyn-Schmiedeberg's Archives of Pharmacology.
[2] A. Kaumann,et al. Interaction of ketanserin and its metabolite ketanserinol with 5HT2 receptors in pulmonary and coronary arteries of calf , 1984, Naunyn-Schmiedeberg's Archives of Pharmacology.
[3] A. Kaumann. Yohimbine and rauwolscine inhibit 5-hydroxytryptamine-induced contraction of large coronary arteries of calf through blockade of 5 HT2 receptors , 1983, Naunyn-Schmiedeberg's Archives of Pharmacology.
[4] A. Kaumann,et al. 3H-(−)-Bupranolol, a new β-adrenoceptor radioligand: Characterization of its binding to kitten heart β-adrenoceptors , 1981, Naunyn-Schmiedeberg's Archives of Pharmacology.
[5] A. Kaumann,et al. A paradox: the 5-HT2-receptor antagonist ketanserin restores the 5-HT-induced contraction depressed by methysergide in large coronary arteries of calf , 2004, Naunyn-Schmiedeberg's Archives of Pharmacology.
[6] G. Martin,et al. Application of the operational model of agonism to establish conditions when functional antagonism may be used to estimate agonist dissociation constants , 1985, British journal of pharmacology.
[7] S. Maayani,et al. 5-Hydroxytryptamine receptor in isolated rabbit aorta: characterization with tryptamine analogs. , 1985, The Journal of pharmacology and experimental therapeutics.
[8] J. Leysen,et al. [3H]Ketanserin (R 41 468), a selective 3H-ligand for serotonin2 receptor binding sites. Binding properties, brain distribution, and functional role. , 1982, Molecular pharmacology.
[9] J. V. van Beek,et al. Vascular effects of ketanserin (R 41 468), a novel antagonist of 5-HT2 serotonergic receptors. , 1981, The Journal of pharmacology and experimental therapeutics.
[10] J. Leysen,et al. Receptor binding profile of R 41 468, a novel antagonist at 5-HT2 receptors. , 1981, Life sciences.
[11] R. Furchgott,et al. COMPARISON OF DISSOCIATION CONSTANTS AND OF RELATIVE EFFICACIES OF SELECTED AGONISTS ACTING ON PARASYMPATHETIC RECEPTORS * , 1967 .
[12] J. R. Blinks. Convenient apparatus for recording contractions of isolated heart muscle. , 1965, Journal of applied physiology.
[13] R. Furchgott. Dibenamine blockade in strips of rabbit aorta and its use in differentiating receptors. , 1954, The Journal of pharmacology and experimental therapeutics.