Conformational and structural considerations in oxytocin-receptor binding and biological activity.
暂无分享,去创建一个
[1] M. Lebl,et al. Analogs of oxytocin containing a pseudopeptide Leu-Gly bond of cis and trans configuration. , 2009, International journal of peptide and protein research.
[2] L. Kinter,et al. Structure-activity relationships of novel vasopressin antagonists containing C-terminal diaminoalkanes and (aminoalkyl)guanidines. , 1989, Journal of medicinal chemistry.
[3] V. Hruby,et al. Design and synthesis of somatostatin analogues with topographical properties that lead to highly potent and specific mu opioid receptor antagonists with greatly reduced binding at somatostatin receptors. , 1988, Journal of medicinal chemistry.
[4] V. Hruby,et al. Weak oxytocin agonist converted to highly potent oxytocin antagonist through bicyclization , 1988 .
[5] L. Kinter,et al. Potent vasopressin antagonists modified at the carboxy-terminal tripeptide tail. , 1987, Journal of medicinal chemistry.
[6] J. Hempel. Chapter 5 – The Conformation of Neurohypophyseal Hormones , 1987 .
[7] M. Lebl,et al. CRC handbook of neurohypophyseal hormone analogs , 1987 .
[8] M. Manning,et al. No requirement of cyclic conformation of antagonists in binding to vasopressin receptors , 1987, Nature.
[9] G. Gessa,et al. Oxytocin: an extremely potent inducer of penile erection and yawning in male rats. , 1986, European journal of pharmacology.
[10] I. L. Schwartz,et al. Antidiuretic and pressor activities of vasopressin analogs with L-alaninamide and D-alaninamide substitutions at position 9. , 2009, International journal of peptide and protein research.
[11] M. Manning,et al. Carboxy terminus of vasopressin required for activity but not binding , 1984, Nature.
[12] J. Glass,et al. Studies of Hydrogen Bonding in Relation to Oxytocin Activity , 1983 .
[13] G. Kovacs,et al. Oxytocin is a precursor of potent behaviourally active neuropeptides. , 1983, European journal of pharmacology.
[14] V. Hruby,et al. Conformational study of the potent peptide hormone antagonist [1-penicillamine,2-leucine]oxytocin in aqueous solution. , 1981, Biochemistry.
[15] M. Sofroniew,et al. Evidence for a direct projection from oxytocin and vasopressin neurons in the hypothalamic paraventricular nucleus to the medulla oblongata: Immunohistochemical visualization of both the horseradish peroxidase transported and the peptide produced by the same neurons , 1981, Neuroscience Letters.
[16] P. Cordopatis,et al. Effect of changing the COOH-terminal amide group present in the hydrophilic cluster of oxytocin to dimethylamide. , 1980, Journal of medicinal chemistry.
[17] G. Berntson,et al. Antinociceptive effects of intraventricular or systemic administration of vasopressin in the rat. , 1980, Life sciences.
[18] R. Walter,et al. Synthesis and biological activities of arginine-vasopressin analogues designed from a conformation-activity approach. , 1979, Journal of medicinal chemistry.
[19] P. Walter. Indentification of sites in oxytocin involved in uterine receptor recognition and activation. , 1977, Federation proceedings.
[20] V. Hruby,et al. Relative conformational rigidity in oxytocin and (1-penicillamine)-oxytocin: a proposal for the relationship of conformational flexibility to peptide hormone agonism and antagonism. , 1977, Proceedings of the National Academy of Sciences of the United States of America.
[21] M. Manning,et al. Synthesis and some pharmacological properties of deamino(4-threonine,8-D-arginine)vasopressin and deamino(8-D-arginine)vasopressin, highly potent and specific antidiuretic peptides, and (8-D-arginine)vasopressin and deamino-arginine-vasopressin. , 1976, Journal of medicinal chemistry.
[22] R. Walter,et al. Conformational studies on arginine vasopressin and arginine vasotocin by proton magnetic resonance spectroscopy. , 1974, Proceedings of the National Academy of Sciences of the United States of America.
[23] M. Manning,et al. Structural changes in the arginine vasopressin molecule that enhance antidiuretic activity and specificity. , 1974, Endocrinology.
[24] F. Šorm,et al. Synthesis and some biological activities of analogues of deamino-vasopressin with the disulphide bridge altered to a thioether bridge , 1974 .
[25] E. Schillinger,et al. Structure activity relationship of the insulin-like effects of the neurohypophysial peptide hormones. , 1972, European journal of biochemistry.
[26] L. B. Flexner,et al. Effect of corticotropin and desglycinamide 9 -lysine vasopressin on suppression of memory by puromycin. , 1972, Proceedings of the National Academy of Sciences of the United States of America.
[27] C. W. Roberts,et al. THE SYNTHESIS OF AN OCTAPEPTIDE AMIDE WITH THE HORMONAL ACTIVITY OF OXYTOCIN , 1953 .