Antimalarial quinolones: synthesis, potency, and mechanistic studies.
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David Hinrichs | D. Hinrichs | M. Riscoe | Rolf W Winter | Jane X Kelly | Martin J Smilkstein | Rozalia Dodean | Michael K Riscoe | M. Smilkstein | R. Winter | J. X. Kelly | R. Dodean | J. Kelly | Rozalia A. Dodean
[1] L. Limpach. Über die Bildung von γ‐Oxy‐chinaldinen aus β‐Arylamino‐crotonsäure‐estern , 1931 .
[2] G. Biagini,et al. Resisting resistance: dealing with the irrepressible problem of malaria. , 2006, British journal of clinical pharmacology.
[3] C. Canfield,et al. Interactions of atovaquone with other antimalarial drugs against Plasmodium falciparum in vitro. , 1995, Experimental parasitology.
[4] R. Williams,et al. Potent and selective hydroxynaphthoquinone inhibitors of mitochondrial electron transport in Eimeria tenella (Apicomplexa: Coccidia). , 1984, Biochemical pharmacology.
[5] C. Wang. Studies of the mitochondria from Eimeria tenella and inhibition of the electron transport by quinolone coccidiostats. , 1975, Biochimica et biophysica acta.
[6] J. B. Pitner,et al. Method for determining oxygen consumption rates of static cultures from microplate measurements of pericellular dissolved oxygen concentration , 2004, Biotechnology and bioengineering.
[7] P. Wilairat,et al. Simple and Inexpensive Fluorescence-Based Technique for High-Throughput Antimalarial Drug Screening , 2004, Antimicrobial Agents and Chemotherapy.
[8] M. Conrad,et al. synthesen von Chinolinderivaten mittelst Acetessigester , 1887 .
[9] R. Williams,et al. Effects of decoquinate and clopidol on electron transport in mitochondria of Eimeria tenella (Apicomplexa: Coccidia). , 1984, Biochemical pharmacology.
[10] G. Dutta,et al. Quinoline esters as potential antimalarial drugs: effect on relapses of Plasmodium cynomolgi infections in monkeys. , 1990, Transactions of the Royal Society of Tropical Medicine and Hygiene.
[11] M. Fry,et al. Site of action of the antimalarial hydroxynaphthoquinone, 2-[trans-4-(4'-chlorophenyl) cyclohexyl]-3-hydroxy-1,4-naphthoquinone (566C80). , 1992, Biochemical pharmacology.
[12] Ruth H. Hughes,et al. PfCRT and the trans‐vacuolar proton electrochemical gradient: regulating the access of chloroquine to ferriprotoporphyrin IX , 2006, Molecular microbiology.
[13] M. Conrad,et al. Ueber das γ-Oxychinaldin und dessen Derivate , 2022 .
[14] S. Meshnick,et al. Artemisinin: mechanisms of action, resistance and toxicity. , 2002, International journal for parasitology.
[15] E. Ashley,et al. Artemisinin-based combinations , 2005, Current opinion in infectious diseases.
[16] W. Trager,et al. Human malaria parasites in continuous culture. , 1976, Science.
[17] A. Casey. 4(1H)-quinolones. 2. Antimalarial effect of some 2-methyl-3-(1'-alkenyl)-or-3-alkyl-4(1H)-quinolones. , 1974, Journal of Medicinal Chemistry.
[18] W. Milhous,et al. REDUCED IN-VITRO SUSCEPTIBILITY TO MEFLOQUINE IN WEST AFRICAN ISOLATES OF PLASMODIUM FALCIPARUM , 1987, The Lancet.
[19] B. Greenwood. Review: Intermittent preventive treatment – a new approach to the prevention of malaria in children in areas with seasonal malaria transmission , 2006, Tropical medicine & international health : TM & IH.
[20] Lauer Wm,et al. The synthesis of some chloromethoxyquinolines. , 1946 .
[21] A. Buoniconti,et al. The royal commission and London. , 1968, Lancet.
[22] J. F. Ryley,et al. The antimalarial activity of some quinolone esters. , 1970, Annals of tropical medicine and parasitology.
[23] D. Hinrichs,et al. Evaluation and lead optimization of anti-malarial acridones. , 2006, Experimental parasitology.
[24] Joanne M. Morrisey,et al. Resistance mutations reveal the atovaquone‐binding domain of cytochrome b in malaria parasites , 1999, Molecular microbiology.
[25] J. Brown,et al. New tissue schizontocidal antimalarial drugs. , 1981, Bulletin of the World Health Organization.
[26] Q. Cheng,et al. Mutations in Plasmodium falciparumCytochrome b That Are Associated with Atovaquone Resistance Are Located at a Putative Drug-Binding Site , 2000, Antimicrobial Agents and Chemotherapy.
[27] R. Williams. The mode of action of anticoccidial quinolones (6-decyloxy-4-hydroxyquinoline-3-carboxylates) in chickens. , 1997, International journal for parasitology.
[28] R. Gould,et al. The Synthesis of Certain Substituted Quinolines and 5,6-Benzoquinolines , 1939 .
[29] P. Rosenthal,et al. Comparison of Efficacies of Cysteine Protease Inhibitors against Five Strains of Plasmodium falciparum , 2001, Antimicrobial Agents and Chemotherapy.
[30] S. Hay,et al. The global distribution of clinical episodes of Plasmodium falciparum malaria , 2005, Nature.
[31] H. Timmler,et al. Über einen neuen, gegen Vogelmalaria wirksamen Verbindungstypus† , 1948 .
[32] R. Snow,et al. Averting a malaria disaster , 1999, The Lancet.
[33] Nicholas J White,et al. Antimalarial drug resistance. , 2004, The Journal of clinical investigation.
[34] J. F. Ryley. Lerbek, a synergistic mixture of methyl benzoquate and clopidol for the prevention of chicken coccidiosis , 1975, Parasitology.
[35] K. Kain,et al. Atovaquone-proguanil: report from the CDC expert meeting on malaria chemoprophylaxis (II). , 2007, The American journal of tropical medicine and hygiene.
[36] C. Chong,et al. Inhibition of heme crystal growth by antimalarials and other compounds: implications for drug discovery. , 2003, Biochemical pharmacology.