WITHDRAWN: 2-Arylquinazolin-4(3H)-ones: A new class of α-glucosidase inhibitors
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M. Choudhary | S. Saad | K. Khan | S. Perveen | I. Fatima | Uzma Salar | Kulsoom Javaid | U. Salar | K. Javaid | Itrat Fatima
[1] M. Choudhary,et al. Synthesis and β-glucuronidase inhibitory activity of 2-arylquinazolin-4(3H)-ones. , 2014, Bioorganic & medicinal chemistry.
[2] Ghada S. Hassan,et al. Nonclassical antifolates, part 3: synthesis, biological evaluation and molecular modeling study of some new 2-heteroarylthio-quinazolin-4-ones. , 2013, European journal of medicinal chemistry.
[3] Tuan-Anh N. Pham,et al. Synthesis and biological evaluation of novel 2,4-disubstituted quinazoline analogues as GPR119 agonists. , 2013, Bioorganic & medicinal chemistry.
[4] Shin-Duk Kim. α-Glucosidase inhibitor from Buthus martensi Karsch. , 2013, Food chemistry.
[5] Can Zhang,et al. Novel oxazolo[4,5-g]quinazolin-2(1H)-ones: dual inhibitors of EGFR and Src protein tyrosine kinases. , 2012, European journal of medicinal chemistry.
[6] P. Crooks,et al. 3-[Benzimidazo- and 3-[benzothiadiazoleimidazo-(1,2-c)quinazolin-5-yl]-2H-chromene-2-ones as potent antimicrobial agents. , 2011, Bioorganic & medicinal chemistry letters.
[7] Mahmud Tareq Hassan Khan,et al. Alpha-glucosidase and tyrosinase inhibitors from fungal hydroxylation of tibolone and hydroxytibolones , 2010, Steroids.
[8] Mahmud Tareq Hassan Khan,et al. Identification of novel quinazolin-4(3H)-ones as inhibitors of thermolysin, the prototype of the M4 family of proteinases. , 2010, Bioorganic & medicinal chemistry.
[9] R. Tundis,et al. Natural Products as α-Amylase and α-Glucosidase Inhibitors and their Hypoglycaemic Potential in the Treatment of Diabetes: An Update , 2010 .
[10] K. Kavitha,et al. Synthesis and pharmacological investigation of novel 4-(2-methylphenyl)-1-substituted-4H-[1,2,4]triazolo[4,3-a]quinazolin-5-ones as new class of H(1)-antihistaminic agents. , 2008, European journal of medicinal chemistry.
[11] S. Murugesan,et al. Synthesis of 4-butyl-1-substituted-4H-[1,2,4]triazolo[4,3-a]quinazolin-5-ones as new class of H(1)-antihistaminic agents. , 2008, Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie.
[12] B. Zinman,et al. Impaired Fasting Glucose and Impaired Glucose Tolerance , 2007, Diabetes Care.
[13] Ivone Carvalho,et al. α- and β-Glucosidase inhibitors: chemical structure and biological activity , 2006 .
[14] Petro Petrides1. Anagrelide: What Was New in 2004 and 2005? , 2006, Seminars in thrombosis and hemostasis.
[15] T. Gefflaut,et al. Synthesis of new nitrogen analogues of salacinol and deoxynojirimycin and their evaluation as glycosidase inhibitors. , 2006, The Journal of organic chemistry.
[16] F. Birke,et al. Pyrrolidinohydroquinazolines--a novel class of CCR3 modulators. , 2005, Bioorganic & medicinal chemistry letters.
[17] R. Wilson,et al. EGF receptor gene mutations are common in lung cancers from "never smokers" and are associated with sensitivity of tumors to gefitinib and erlotinib. , 2004, Proceedings of the National Academy of Sciences of the United States of America.
[18] A. Venkateswarlu,et al. Synthesis and biological evaluation of [4-(2-phenylethenesulfonylmethyl)phenyl]-quinazolin-4-yl-amines as orally active anti-cancer agents. , 2004, Bioorganic & medicinal chemistry letters.
[19] M. Kizaki,et al. Capsaicin-Like Anti-Obese Activities of Evodiamine from Fruits of Evodia rutaecarpa, a Vanilloid Receptor Agonist , 2001, Planta medica.
[20] K. Schrör,et al. Inhibition of platelet-derived growth factor-induced mitogenesis by phosphodiesterase 3 inhibitors: role of protein kinase A in vascular smooth muscle cell mitogenesis. , 2000, Biochemical pharmacology.
[21] N Zitzmann,et al. Imino sugars inhibit the formation and secretion of bovine viral diarrhea virus, a pestivirus model of hepatitis C virus: implications for the development of broad spectrum anti-hepatitis virus agents. , 1999, Proceedings of the National Academy of Sciences of the United States of America.
[22] D. Riendeau,et al. Phosphodiesterase 4-dependent regulation of cyclic AMP levels and leukotriene B4 biosynthesis in human polymorphonuclear leukocytes. , 1999, European journal of pharmacology.
[23] Y. Kurogi,et al. Synthesis and hypolipidemic activities of novel 2-[4-[diethoxyphosphoryl)methyl]phenyl]quinazolines and 4(3H)-quinazolinones. , 1996, Journal of medicinal chemistry.
[24] M. Davies,et al. Impaired glucose tolerance , 1996, BMJ.
[25] M. Poli,et al. Prophylaxis and treatment with a monoclonal antibody of tetrodotoxin poisoning in mice. , 1995, Toxicon : official journal of the International Society on Toxinology.
[26] M. Niimura,et al. Photoleukomelanodermatitis (Kobori) Induced by Afloqualone , 1994, The Journal of dermatology.
[27] H. Holmsen. Significance of testing platelet functions in vitro , 1994, European journal of clinical investigation.
[28] F. Rousseau. The fragile X syndrome: implications of molecular genetics for the clinical syndrome , 1994, European journal of clinical investigation.
[29] J. Groopman. Current advances in the diagnosis and treatment of AIDS: an introduction. , 1990, Reviews of infectious diseases.
[30] V. Ram,et al. Chemotherapeutic agents XI: synthesis of pyrimidines and azolopyrimidines as leishmanicides☆ , 1990 .
[31] M. Scheinbaum,et al. R013-6438, a new inotrope-vasodilator: Systemic and coronary hemodynamic effects in congestive heart failure , 1985 .
[32] G. Belz,et al. Dose‐Response Following Single Administrations of a New Cardiac Performance Enhancer RO 13–6438 in Normal Volunteers , 1985, Journal of cardiovascular pharmacology.
[33] M. Gerold,et al. Cardiovascular Profile of Ro 13–6438, a Novel Positive Inotropic Agent with Vasodilating Properties , 1984, Journal of cardiovascular pharmacology.
[34] Amer Ms,et al. Effect of quazodine on phosphodiesterase. , 1971 .
[35] J. R. Vaughan,et al. Quinazolinone Sulfonamides. A New Class of Diuretic Agents1 , 1960 .
[36] Ji Young Kim,et al. Synthesis and antifungal activity of 6,7-bis(arylthio)-quinazoline-5,8-diones and furo[2,3-f]quinazolin-5-ols. , 2012, Bioorganic & medicinal chemistry letters.
[37] C. S. Rajput,et al. Synthesis and anti-inflammatory activity of newer quinazolin-4-one derivatives. , 2009, European journal of medicinal chemistry.
[38] T. Kurtz,et al. Type 2 diabetes and oral antihyperglycemic drugs. , 2008, Current medicinal chemistry.
[39] J. Blessing,et al. Trimetrexate in the treatment of recurrent or advanced leiomyosarcoma of the uterus: a phase II study of the Gynecologic Oncology Group. , 2002, Gynecologic oncology.
[40] A. Boddy,et al. Phase I studies with the nonclassical antifolate nolatrexed dihydrochloride (AG337, THYMITAQ) administered orally for 5 days. , 1999, Clinical cancer research : an official journal of the American Association for Cancer Research.
[41] A. Caruso,et al. Synthesis and pharmacological study of ethyl 1-methyl-5-[2-substituted-4-oxo-3(4H)-quinazolinyl]-1H-pyrazole-4-acetates , 1994 .
[42] R. Ishida,et al. Pharmacological studies on 6-amino-2-fluoromethyl-3-(O-tolyl)-4(3H)-quinazolinone (afloqualone), a new centrally acting muscle relaxant. (II) Effects on the spinal reflex potential and the rigidity. , 1982, Japanese journal of pharmacology.