Novel H3 receptor antagonists. Sulfonamide homologs of histamine.
暂无分享,去创建一个
J. Hey | M. Connolly | R. West | M. Rivelli | R. Wolin | A. Afonso | H. She | S. Willams
[1] P. Carrupt,et al. H3-receptor antagonists: synthesis and structure-activity relationships of para- and meta-substituted 4(5)-phenyl-2-[[2-[4(5)-imidazolyl]ethyl]thio]imidazoles. , 1997, Journal of medicinal chemistry.
[2] J. Schwartz,et al. A novel series of (phenoxyalkyl)imidazoles as potent H3-receptor histamine antagonists. , 1996, Journal of medicinal chemistry.
[3] J. Schwartz,et al. Design of potent non-thiourea H3-receptor histamine antagonists. , 1995, Journal of medicinal chemistry.
[4] R. Leurs,et al. Homologs of histamine as histamine H3 receptor antagonists: a new potent and selective H3 antagonist, 4(5)-(5-aminopentyl)-1H-imidazole. , 1995, Journal of medicinal chemistry.
[5] Gavin Kilpatrick,et al. Histamine H3 receptors modulate the release of [3H]‐acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes , 1992, British journal of pharmacology.
[6] J. Schwartz,et al. Synthesis, absolute configuration, stereoselectivity, and receptor selectivity of (alpha R, beta S)-alpha,beta-dimethylhistamine, a novel high potent histamine H3 receptor agonist. , 1992, Journal of medicinal chemistry.
[7] R. Egan,et al. (R)-alpha-methylhistamine augments neural, cholinergic bronchospasm in guinea pigs by histamine H1 receptor activation. , 1992, European journal of pharmacology.
[8] R. Egan,et al. Characterization and tissue distribution of H3 histamine receptors in guinea pigs by N alpha-methylhistamine. , 1990, Biochemical and biophysical research communications.
[9] H. Timmerman. Histamine H3 ligands: just pharmacological tools or potential therapeutic agents? , 1990, Journal of medicinal chemistry.
[10] J. Schwartz,et al. Highly potent and selective ligands for histamine H3-receptors , 1987, Nature.
[11] R. DiPietro,et al. Improved Syntheses of Vinyl Imidazoles1 , 1986 .
[12] J. Schwartz,et al. Properties and roles of the three subclasses of histamine receptors in brain. , 1986, The Journal of experimental biology.
[13] J. Schwartz,et al. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor , 1983, Nature.
[14] J. Black,et al. Definition and Antagonism of Histamine H2-receptors , 1972, Nature.