Macrocyclic BACE inhibitors: Optimization of a micromolar hit to nanomolar leads.
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M. Vandermeeren | M. Mercken | C. Ho | R. Alexander | G. Yohrling | C. Reynolds | D. Brenneman | B. Tounge | K. Conway | A. Reitz | Yifang Huang | E. W. Baxter | D. Rosenthal | J. Piesvaux | M. H. Parker | E. Strobel | H. Moore Arnold | Chih Ho