An intramolecular Michael reaction strategy for the synthesis of 2,6-disubstituted-3-piperidinols
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[1] B. Lygo. Use of an alamine derived β-ketosulfone in the synthesis of peptide isosteres , 2002 .
[2] S. Sengupta,et al. Diastereoselective reduction of N-phthaloyl α-amino ketones: synthesis of syn-3-amino-1,2-diol derivatives☆ , 2001 .
[3] Somnath Mondal,et al. Zinc Borohydride Reduction of α-Amino Ketones: A Highly Diastereoselective Synthetic Route to anti-γ-Hydroxy-β-amino Alcohols , 2001 .
[4] S. Laschat,et al. Stereoselective Synthesis of Piperidines , 2001 .
[5] P. Stevenson,et al. Synthesis of trans-5-substituted-indolizidin-3-one , 2000 .
[6] A. Moretto,et al. Stereo- and regiocontrolled construction of trisubstituted piperidines using a TpMo(CO)(2)(dihydropyridine) scaffold (Tp = hydridotrispyrazolylborate). , 2000, The Journal of organic chemistry.
[7] S. Haroutounian,et al. Asymmetric total synthesis of (−)-prosophylline , 1999 .
[8] J. Paris,et al. New application of the Julia olefination for the synthesis of Tyr-Gly E-alkene and carba isostere pseudopeptides , 1999 .
[9] Wei-shan Zhou,et al. New concise asymmetric total synthesis of (+)-desoxoprosophylline and prosophylline , 1999 .
[10] N. Toyooka,et al. 2-Piperidone Type of Chiral Building Block for 3-Piperidinol Alkaloid Synthesis. , 1999, The Journal of organic chemistry.
[11] T. Nishio,et al. Hypervalent λn-iodane-mediated fragmentation of tertiary cyclopropanol systems II: Application to asymmetric syntheses of piperidine and indolizidine alkaloids , 1999 .
[12] T. Naito,et al. Total synthesis of (+)-azimic acid, (+)-julifloridine, and proposed structure ofN-methyljulifloridine via cycloaddition of nitrone to a chiral dipolarophile , 1998 .
[13] Wei-shan Zhou,et al. Asymmetric total synthesis of (+)-desoxoprosophylline , 1998 .
[14] Somnath Mondal,et al. A facile synthesis of Enantiopure γ-Amino-And γ-Hydroxy-β-Ketosulfones , 1998 .
[15] I. Ojima,et al. Rhodium-Catalyzed Cyclohydrocarbonylation: Application to the Synthesis of (+)-Prosopinine and (−)-Deoxoprosophylline† , 1998 .
[16] Somnath Mondal,et al. γ-Amino-β-ketosulfones as chiral educts: A facile synthesis of enantiopure α-amino ketones , 1998 .
[17] Hubert Lam,et al. A new access to enantiopure β-hydroxylated piperidines from N-Boc-2-acyloxazolidines. Application to the synthesis of (−)-desoxoprosopinine and (+)-pseudoconhydrine , 1998 .
[18] F. Couty,et al. Total synthesis of (−)-desoxoprosopinine via the diastereoselective reduction of homochiral2-Acyl-N-Boc-oxazolidines , 1998 .
[19] A. Pahl,et al. Synthesis of (−)-(2R,3R,6S)-irnigaine and (+)-(2R,3R,6S)-N-methylirnigaine , 1998 .
[20] H. Takahata,et al. SYMMETRY-ASSISTED SYNTHESIS OF C2-SYMMETRIC TRANS-ALPHA , ALPHA '-BIS(HYDROXYMETHYL)PYRROLIDINE AND -PIPERIDINE DERIVATIVES VIA DOUBLE SHARPLESS ASYMM ETRIC DIHYDROXYLATION OF ALPHA , OMEGA -TERMINAL DIENES , 1998 .
[21] A. Albeck,et al. Functionalized erythro N-protected α-amino epoxides. Stereocontrolled synthesis and biological activity , 1997 .
[22] J. Carretero,et al. Stereoselective synthesis of hydroxypyrrolidines and hydroxypiperidines by cyclization of γ-oxygenated-α,β-unsaturated sulfones , 1996 .
[23] E. Akiyama,et al. Total Synthesis and Absolute Configuration of (-)-Sedacryptine , 1996 .
[24] D. Rotella. Stereoselective synthesis of erythro α-amino epoxides , 1995 .
[25] D. Kingston,et al. BIOACTIVE AND OTHER PIPERIDINE ALKALOIDS FROM CASSIA-LEPTOPHYLLA , 1995 .
[26] C. Rudd,et al. Synthesis of Xaa-Gly-Xaa′ keto-methylene tri-peptide isosteres incorporating phenylalanine, tyrosine and valine units , 1995 .
[27] M. Hirama,et al. Stereoselective Synthesis of (+)-Swainsonine and (-)-8,8a-Di-epi-swainsonine , 1995 .
[28] L. Beholz,et al. Construction of Hydroxylated Alkaloids (.+-.)-Mannonolactam, (.+-.)-Deoxymannojirimycin, and (.+-.)-Prosopinine through Aza-Annulation , 1994 .
[29] R. Persky,et al. Stereocontrolled synthesis of erythro N-protected α-amino epoxides and peptidyl epoxides , 1994 .
[30] T. Ye,et al. Synthesis of chiral n-protected α-amino-β-diketones from α-diazoketones derived from natural amino acids , 1992 .
[31] M. Hirama,et al. Diastereofacial selectivity in the intramolecular conjugate addition of a nitrogen nucleophile; stereocontrolled piperidine synthesis , 1987 .
[32] G. Germain,et al. Sedum alkaloids II: sedacryptine, a new minor base from sedum acre. , 1980 .
[33] I. Christofidis,et al. Spectaline and iso-6 cassine, two new piperidin 3-ol alkaloids from the leaves of cassia spectabilis , 1977 .