Synthesis, anti-inflammatory, analgesic and kinase (CDK-1, CDK-5 and GSK-3) inhibition activity evaluation of benzimidazole/benzoxazole derivatives and some Schiff's bases.
暂无分享,去创建一个
[1] N. Curtin,et al. Potentiation of cytotoxic drug activity in human tumour cell lines, by amine-substituted 2-arylbenzimidazole-4-carboxamide PARP-1 inhibitors. , 2004, Bioorganic & medicinal chemistry letters.
[2] T. Inoue,et al. Synthesis and biological activities of novel antiallergic agents with 5-lipoxygenase inhibiting action. , 2000, Bioorganic & medicinal chemistry.
[3] F. Costantini,et al. Purification of GSK-3 by affinity chromatography on immobilized axin. , 2000, Protein expression and purification.
[4] J. Lown,,et al. SYNTHESIS OF AMIDINE AND BIS AMIDINE PERCURSORS , 2001 .
[5] Ashok Kumar,et al. Synthesis, anti-inflammatory and analgesic activities evaluation of some mono, bi and tricyclic pyrimidine derivatives. , 2005, Bioorganic & medicinal chemistry.
[6] J. Lown,,et al. Heterocyclic Compounds as Inflammation Inhibitors , 2002 .
[7] A. Sparatore,et al. Synthesis and biological investigations of 2-(tetrahydropyran-2'-yl) and 2-(tetrahydrofuran-2'-yl)benzimidazoles. , 1997, Farmaco.
[8] Sung-Yu Hong,et al. Synthesis and biological evaluation of benzimidazole-4,7-diones that inhibit vascular smooth muscle cell proliferation. , 2004, Bioorganic & medicinal chemistry letters.
[9] J. Lown,,et al. Anticancer, Anti-inflammatory and Analgesic Activity Evaluation of Heterocyclic Compounds Synthesized by the Reaction of 4-Isothiocyanato-4-methylpentan-2-one with Substituted o-Phenylenediamines, o-Diaminopyridine and (Un)Substituted o , 2001 .
[10] J. W. COOK,et al. A Text-Book of Practical Organic Chemistry , 1948, Nature.
[11] G L Snyder,et al. Paullones are potent inhibitors of glycogen synthase kinase-3beta and cyclin-dependent kinase 5/p25. , 2000, European journal of biochemistry.
[12] R. Goyal,et al. Synthesis and biological evaluation of 2-thiopyrimidine derivatives. , 2005, Bioorganic & medicinal chemistry.
[13] A. Pession,et al. Differential antiproliferative activity of new benzimidazole-4,7-diones. , 2004, Farmaco.
[14] G L Snyder,et al. Indirubins inhibit glycogen synthase kinase-3 beta and CDK5/p25, two protein kinases involved in abnormal tau phosphorylation in Alzheimer's disease. A property common to most cyclin-dependent kinase inhibitors? , 2001, The Journal of biological chemistry.
[15] P. Singh,et al. Acetic acid and phenylquinone writhing test: a critical study in mice. , 1983, Methods and findings in experimental and clinical pharmacology.
[16] E. Yeşilada,et al. Studies on Novel 7‐Acyl‐5‐chloro‐2‐oxo‐3H‐benzoxazole Derivatives as Potential Analgesic and Anti‐Inflammatory Agents , 2003, Archiv der Pharmazie.
[17] J. Kočí,et al. Heterocyclic benzazole derivatives with antimycobacterial in vitro activity. , 2002, Bioorganic & medicinal chemistry letters.
[18] A. Brukštus,et al. Synthesis and Antiinflammatory Activity of Some New 1-Acyl Derivatives of 2-Methylthio-5,6-Diethoxybenzimidazole , 2004, Pharmaceutical Chemistry Journal.
[19] S. Sondhi,et al. Synthesis, Hydrolysis over Silica Column, Anticancer, Antiinflammatory and Analgesic Activity Evaluation of Some Pyridine (I) and Pyrazine Derivatives (II). , 2005 .
[20] H. Homma,et al. Studies on the synthesis and anti-inflammatory activity of 2,6-di-tert-butylphenols with a heterocyclic group at the 4-position. I. , 1983, Chemical & pharmaceutical bulletin.
[21] C A WINTER,et al. Carrageenin-Induced Edema in Hind Paw of the Rat as an Assay for Antiinflammatory Drugs , 1962, Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine.
[22] M. Andrzejewska,et al. Synthesis and antimycobacterial activity of 2-substituted halogenobenzimidazoles. , 2005, European journal of medicinal chemistry.
[23] L. Meijer,et al. Synthesis of acridinyl-thiazolino derivatives and their evaluation for anti-inflammatory, analgesic and kinase inhibition activities. , 2005, Bioorganic & medicinal chemistry.