3-(2-carboxyethyl)-4,6-dichloro-1H-indole-2-carboxylic acid: an allosteric inhibitor of fructose-1,6-bisphosphatase at the AMP site.

[1]  S. Wright,et al.  Allosteric inhibition of fructose-1,6-bisphosphatase by anilinoquinazolines. , 2001, Bioorganic & medicinal chemistry letters.

[2]  B. Spur,et al.  A selective method for the preparation of aliphatic methyl esters in the presence of aromatic carboxylic acids , 1998 .

[3]  M. Erion,et al.  The allosteric site of human liver fructose-1,6-bisphosphatase. Analysis of six AMP site mutants based on the crystal structure. , 1995, The Journal of biological chemistry.

[4]  W. Lipscomb,et al.  Toward a mechanism for the allosteric transition of pig kidney fructose-1,6-bisphosphatase. , 1994, Journal of Molecular Biology.

[5]  J. Navaza,et al.  AMoRe: an automated package for molecular replacement , 1994 .

[6]  S. Pilkis,et al.  Isolation of a human liver fructose-1,6-bisphosphatase cDNA and expression of the protein in Escherichia coli. Role of ASP-118 and ASP-121 in catalysis. , 1993, The Journal of biological chemistry.

[7]  J. Kehne,et al.  3-(2-Carboxyindol-3-yl)propionic acid-based antagonists of the N-methyl-D-aspartic acid receptor associated glycine binding site. , 1992, Journal of medicinal chemistry.

[8]  E. Kantrowitz,et al.  Isolation and sequence analysis of the cDNA for pig kidney fructose 1,6-bisphosphatase. , 1992, Proceedings of the National Academy of Sciences of the United States of America.

[9]  W. Lipscomb,et al.  Conformational transition of fructose-1,6-bisphosphatase: structure comparison between the AMP complex (T form) and the fructose 6-phosphate complex (R form). , 1991, Biochemistry.

[10]  F. Salituro,et al.  3-(2-carboxyindol-3-yl)propionic acid derivatives: antagonists of the strychnine-insensitive glycine receptor associated with the N-methyl-D-aspartate receptor complex. , 1990, Journal of medicinal chemistry.

[11]  C. Melchiorre,et al.  3-Phenyl analogues of 2-[[[2-(2,6-dimethoxyphenoxy)ethyl]amino]-methyl]-1,4-benzodioxan (WB 4101) as highly selective alpha 1-adrenoceptor antagonists. , 1990 .

[12]  W. Lipscomb,et al.  Crystal structure of fructose-1,6-bisphosphatase complexed with fructose 6-phosphate, AMP, and magnesium. , 1990, Proceedings of the National Academy of Sciences of the United States of America.

[13]  H. Ikeda,et al.  Pathogenesis of hyperglycemia in genetically obese-hyperglycemic rats, Wistar fatty: presence of hepatic insulin resistance. , 1989, Endocrinologia japonica.

[14]  S. Pilkis,et al.  cDNA sequence of rat liver fructose-1,6-bisphosphatase and evidence for down-regulation of its mRNA by insulin. , 1988, Proceedings of the National Academy of Sciences of the United States of America.

[15]  A. Baykov,et al.  A malachite green procedure for orthophosphate determination and its use in alkaline phosphatase-based enzyme immunoassay. , 1988, Analytical biochemistry.

[16]  T. Claus,et al.  Inhibition of fructose-1,6-bisphosphatase by fructose 2,6-bisphosphate. , 1981, The Journal of biological chemistry.

[17]  K. Manchester,et al.  A comparison of the effects of diabetes induced with either alloxan or streptozotocin and of starvation on the activities in rat liver of the key enzymes of gluconeogenesis. , 1970, The Biochemical journal.

[18]  S. Pontremoli,et al.  Fructose diphosphatase from rabbit liver. X. Isolation and kinetic properties of the enzyme--adenosine monophosphate complex. , 1968, Biochemistry.

[19]  W. Wood,et al.  Fructose diphosphatase from rabbit liver. I. Purification and properties. , 1965, The Journal of biological chemistry.

[20]  K. Taketa,et al.  ALLOSTERIC INHIBITION OF RAT LIVER FRUCTOSE 1,6-DIPHOSPHATASE BY ADENOSINE 5'-MONOPHOSPHATE. , 1965, The Journal of biological chemistry.

[21]  D. Granner,et al.  Molecular physiology of the regulation of hepatic gluconeogenesis and glycolysis. , 1992, Annual review of physiology.

[22]  T. Claus,et al.  Hormonal regulation of hepatic gluconeogenesis and glycolysis. , 1988, Annual review of biochemistry.

[23]  C. Veneziale.  The Regulation of carbohydrate formation and utilization in mammals , 1981 .